

Compound name | Brutto | MW | CAS | PubChem CID | Action | Reference | Reference |
---|---|---|---|---|---|---|---|
(5Z)-7-Oxozeaenol | C19H22O7 | 362.37 | 66018-38-0 | 53442201 | TAK1 | Ninomiya-Tsuji (2003) J.Biol.Chem. 278 18485 | Windheim et al (2007) Biochem.J. 404 179 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
ABL | 108 | 5 |
AMPK | 100 | 7 |
ASK1 | 91 | 1 |
Aurora A | 106 | 20 |
Aurora B | 94 | 1 |
BRK | 65 | 13 |
BRSK1 | 113 | 12 |
BRSK2 | 84 | 11 |
BTK | 90 | 5 |
CAMK1 | 88 | 2 |
CAMKK beta | 87 | 4 |
CDK2-Cyclin A | 119 | 7 |
CHK1 | 114 | 13 |
CHK2 | 110 | 1 |
CK1 delta | 102 | 4 |
CK2 | 106 | 15 |
CLK2 | 96 | 17 |
CSK | 118 | 16 |
DAPK1 | 108 | 1 |
DYRK1A | 117 | 0 |
DYRK2 | 114 | 5 |
DYRK3 | 94 | 7 |
EF2K | 48 | 57 |
EPH-A2 | 99 | 8 |
EPH-A4 | 91 | 4 |
EPH-B1 | 99 | 11 |
EPH-B2 | 96 | 21 |
EPH-B3 | 111 | 8 |
EPH-B4 | 87 | 6 |
ERK1 | 106 | 15 |
ERK2 | 103 | 2 |
ERK8 | 40 | 2 |
FGF-R1 | 105 | 24 |
GCK | 121 | 3 |
GSK3 beta | 102 | 13 |
HER4 | 100 | 2 |
HIPK1 | 102 | 11 |
HIPK2 | 98 | 9 |
HIPK3 | 90 | 2 |
IGF-1R | 100 | 16 |
IKK beta | 102 | 17 |
IKK epsilon | 120 | 4 |
IR | 110 | 10 |
IRAK4 | 99 | 4 |
IRR | 107 | 52 |
JAK2 | 108 | 11 |
JNK1 | 90 | 0 |
JNK2 | 109 | 12 |
JNK3 | 107 | 2 |
Lck | 78 | 1 |
LKB1 | 138 | 6 |
MAPKAP-K2 | 124 | 4 |
MAPKAP-K3 | 113 | 18 |
MARK1 | 112 | 16 |
MARK2 | 109 | 1 |
MARK3 | 116 | 11 |
MARK4 | 107 | 1 |
MEKK1 | 107 | 5 |
MELK | 95 | 11 |
MINK1 | 101 | 9 |
MKK1 | 13 | 2 |
MKK2 | 12 | 2 |
MKK6 | 12 | 4 |
MLK1 | 109 | 4 |
MLK3 | 114 | 16 |
MNK1 | 55 | 0 |
MNK2 | 41 | 3 |
MPSK1 | 103 | 6 |
MSK1 | 107 | 25 |
MST2 | 120 | 14 |
MST4 | 129 | 6 |
NEK2a | 108 | 0 |
NEK6 | 122 | 5 |
NUAK1 | 113 | 9 |
p38 alpha MAPK | 103 | 3 |
p38 beta MAPK | 90 | 9 |
p38 delta MAPK | 99 | 2 |
p38 gamma MAPK | 99 | 1 |
PAK2 | 104 | 5 |
PAK4 | 94 | 11 |
PAK5 | 96 | 9 |
PAK6 | 100 | 5 |
PDK1 | 99 | 10 |
PHK | 100 | 2 |
PIM1 | 102 | 1 |
PIM2 | 91 | 7 |
PIM3 | 126 | 6 |
PKA | 99 | 7 |
PKB alpha | 111 | 9 |
PKB beta | 86 | 9 |
PKC alpha | 107 | 3 |
PKC gamma | 87 | 4 |
PKC zeta | 105 | 1 |
PKD1 | 71 | 6 |
PLK1 | 103 | 1 |
PRAK | 66 | 7 |
PRK2 | 102 | 2 |
RIPK2 | 103 | 5 |
ROCK 2 | 116 | 13 |
RSK1 | 113 | 1 |
RSK2 | 106 | 6 |
S6K1 | 112 | 8 |
SGK1 | 106 | 2 |
SmMLCK | 108 | 4 |
Src | 106 | 4 |
SRPK1 | 104 | 10 |
STK33 | 120 | 13 |
SYK | 88 | 3 |
TAK1 |
5
|
1 |
TAO1 | 103 | 3 |
TBK1 | 105 | 1 |
TIE2 | 103 | 16 |
TrkA | 46 | 0 |
TTK | 104 | 2 |
VEGFR1 |
8
|
0 |
YES1 | 105 | 40 |
ZAP70 | 110 | 4 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
ABL | 71 | 6 |
AMPK | 92 | 5 |
ASK1 | 95 | 6 |
Aurora A | 105 | 2 |
Aurora B | 74 | 6 |
BRK | 25 | 0 |
BRSK1 | 90 | 4 |
BRSK2 | 88 | 11 |
BTK | 93 | 0 |
CAMK1 | 105 | 11 |
CAMKK beta | 57 | 2 |
CDK2-Cyclin A | 88 | 3 |
CHK1 | 92 | 3 |
CHK2 | 87 | 1 |
CK1 delta | 104 | 6 |
CK2 | 77 | 1 |
CLK2 | 90 | 2 |
CSK | 56 | 7 |
DAPK1 | 94 | 2 |
DYRK1A | 97 | 1 |
DYRK2 | 89 | 5 |
DYRK3 | 101 | 2 |
EF2K | 85 | 3 |
EPH-A2 | 55 | 2 |
EPH-A4 | 46 | 8 |
EPH-B1 | 81 | 8 |
EPH-B2 | 75 | 5 |
EPH-B3 | 100 | 4 |
EPH-B4 | 90 | 5 |
ERK1 | 64 | 0 |
ERK2 | 65 | 7 |
ERK8 |
4
|
4 |
FGF-R1 | 87 | 7 |
GCK | 80 | 0 |
GSK3 beta | 74 | 5 |
HER4 | 95 | 1 |
HIPK1 | 98 | 9 |
HIPK2 | 82 | 4 |
HIPK3 | 103 | 10 |
IGF-1R | 93 | 8 |
IKK beta | 95 | 6 |
IKK epsilon | 92 | 10 |
IR | 94 | 7 |
IRAK4 | 28 | 2 |
IRR | 96 | 14 |
JAK2 | 75 | 0 |
JNK1 | 52 | 14 |
JNK2 | 81 | 4 |
JNK3 | 90 | 11 |
Lck | 30 | 4 |
LKB1 | 65 | 1 |
MAPKAP-K2 | 79 | 4 |
MAPKAP-K3 | 94 | 5 |
MARK1 | 99 | 0 |
MARK2 | 114 | 3 |
MARK3 | 77 | 14 |
MARK4 | 86 | 4 |
MEKK1 | 92 | 2 |
MELK | 94 | 4 |
MINK1 | 83 | 1 |
MKK1 |
2
|
1 |
MKK2 |
3
|
2 |
MKK6 |
10
|
2 |
MLK1 | 75 | 1 |
MLK3 | 79 | 18 |
MNK1 | 13 | 5 |
MNK2 | 26 | 1 |
MPSK1 | 101 | 10 |
MSK1 | 100 | 1 |
MST2 | 89 | 4 |
MST4 | 72 | 9 |
NEK2a | 89 | 1 |
NEK6 | 93 | 5 |
NUAK1 | 78 | 3 |
p38 alpha MAPK | 85 | 4 |
p38 beta MAPK | 72 | 0 |
p38 delta MAPK | 114 | 14 |
p38 gamma MAPK | 92 | 6 |
PAK2 | 110 | 8 |
PAK4 | 81 | 6 |
PAK5 | 103 | 6 |
PAK6 | 87 | 1 |
PDK1 | 76 | 3 |
PHK | 89 | 5 |
PIM1 | 72 | 9 |
PIM2 | 106 | 4 |
PIM3 | 80 | 3 |
PKA | 93 | 1 |
PKB alpha | 91 | 1 |
PKB beta | 84 | 10 |
PKC alpha | 85 | 3 |
PKC gamma | 87 | 10 |
PKC zeta | 99 | 12 |
PKD1 | 31 | 11 |
PLK1 | 100 | 6 |
PRAK | 14 | 11 |
PRK2 | 91 | 15 |
RIPK2 | 39 | 2 |
ROCK 2 | 83 | 6 |
RSK1 | 90 | 2 |
RSK2 | 70 | 13 |
S6K1 | 82 | 4 |
SGK1 | 95 | 1 |
SmMLCK | 80 | 5 |
Src | 43 | 3 |
SRPK1 | 88 | 5 |
STK33 | 85 | 2 |
SYK | 77 | 5 |
TAK1 |
3
|
1 |
TAO1 | 66 | 5 |
TBK1 | 102 | 13 |
TIE2 | 93 | 9 |
TrkA | 24 | 11 |
TTK | 91 | 8 |
VEGFR1 | 13 | 6 |
YES1 | 60 | 2 |
ZAP70 | 96 | 6 |