Inhibitor | IKK-2 Inhibitor VIII  

Compound name Brutto MW CAS PubChem CID Action Reference Reference
IKK-2 Inhibitor VIII   C21H24N4O2 364.40 406208-42-2 66576999 IKK2 Murata T. (2004) Bioorg. Med. Chem. Lett. 14 4019

Screening Results Chart

Screening Results Tables

Screen Conc: 1.00µM
Kinase % Activity Remaining Sort ascending Standard Deviation
HIPK3 129 2
IRAK4 124 2
BTK 122 13
EPH-B2 119 12
MARK3 118 10
PKC alpha 117 7
IRR 117 7
MKK1 117 2
MAPKAP-K2 115 1
MARK4 115 6
HIPK1 113 8
MST4 113 0
MNK2 113 3
PAK4 112 13
Aurora A 111 1
JNK1 110 1
BRSK1 107 5
MKK2 107 5
EPH-A4 107 14
PKD1 106 9
CAMKK beta 106 1
MSK1 105 5
ASK1 102 14
p38 alpha MAPK 102 15
ERK2 101 4
MNK1 101 3
VEGFR1 101 11
NEK6 99 7
DYRK1A 99 4
EPH-A2 99 13
FGF-R1 97 0
SGK1 96 4
EPH-B1 96 9
CHK1 95 14
EPH-B3 94 15
PRK2 94 7
p38 gamma MAPK 94 3
BRSK2 92 11
SRPK1 92 8
CK2 91 2
DYRK2 91 3
EF2K 90 3
EPH-B4 90 11
PRAK 90 12
PDK1 90 1
TTK 89 10
MARK2 89 1
Src 89 8
PAK6 89 9
S6K1 88 8
MELK 88 1
ROCK 2 88 13
MARK1 88 11
PKC zeta 88 6
p38 beta MAPK 88 11
SYK 88 12
MLK3 87 12
IKK epsilon 87 1
MAPKAP-K3 87 12
CK1 delta 86 6
IGF-1R 86 12
ERK1 85 10
AMPK 85 2
p38 delta MAPK 85 12
CAMK1 85 6
PKB beta 85 2
NEK2a 85 5
PAK5 84 5
DYRK3 84 1
PKA 83 1
JNK2 83 4
PLK1 83 5
PAK2 83 12
CSK 83 11
MST2 83 7
Lck 82 8
PKB alpha 81 9
GSK3 beta 80 3
HIPK2 80 5
RIPK2 80 13
TBK1 80 9
YES1 79 0
LKB1 78 8
TAO1 77 1
GCK 77 3
PHK 77 4
MKK6 76 4
TAK1 73 3
JNK3 73 6
MLK1 73 0
HER4 71 1
SmMLCK 70 1
TrkA 68 1
DAPK1 68 8
Aurora B 67 12
MINK1 66 11
PIM1 63 7
MEKK1 62 1
CHK2 60 4
ERK8 59 2
PIM3 56 3
NUAK1 53 3
IR 51 13
RSK1 45 6
CLK2 43 10
RSK2 39 6
PIM2 34 2
CDK2-Cyclin A 32 1
JAK2 27 5
IKK beta
6
0
Screen Conc: 10.00µM
Kinase % Activity Remaining Sort ascending Standard Deviation
EPH-B2 113 6
MST4 102 5
MARK4 102 5
NEK6 101 5
SRPK1 101 5
EPH-B1 100 10
IKK epsilon 96 8
MARK2 96 11
MAPKAP-K2 95 4
MARK1 95 5
PKA 95 7
NEK2a 94 6
PDK1 94 8
CK2 93 5
CHK1 92 10
DYRK2 91 5
p38 alpha MAPK 91 7
Aurora A 91 7
MNK1 90 13
MNK2 89 4
PRAK 88 8
PLK1 87 14
TBK1 86 9
EPH-B4 86 12
MAPKAP-K3 85 9
EPH-A4 84 3
PAK6 83 2
MKK6 83 13
ASK1 83 6
MARK3 82 6
SYK 81 8
JNK1 80 4
DYRK1A 80 5
ERK1 80 4
HIPK3 79 5
PAK2 78 8
EPH-A2 78 2
CK1 delta 78 3
MKK2 77 8
PKC zeta 76 2
ERK2 76 1
PAK5 75 8
CSK 74 3
EPH-B3 74 2
GSK3 beta 73 8
FGF-R1 72 8
p38 gamma MAPK 72 6
JNK2 71 3
p38 beta MAPK 71 4
IRAK4 70 6
PAK4 69 2
SGK1 69 2
JNK3 68 11
Src 68 3
p38 delta MAPK 68 8
HER4 67 12
TTK 66 3
MLK1 66 5
LKB1 65 3
PKB alpha 63 1
PKB beta 62 5
HIPK1 62 2
ROCK 2 61 4
IRR 61 3
PHK 59 5
HIPK2 59 2
BTK 58 10
BRSK1 58 7
RIPK2 57 3
CAMKK beta 57 8
TAO1 57 6
EF2K 56 3
PKC alpha 55 3
MSK1 55 7
PRK2 53 2
VEGFR1 53 3
S6K1 53 9
MINK1 52 2
MKK1 51 4
AMPK 50 0
MEKK1 50 11
BRSK2 46 1
DAPK1 46 0
PKD1 45 4
MLK3 44 4
Aurora B 42 3
GCK 41 4
DYRK3 40 3
TAK1 39 2
YES1 38 13
IGF-1R 35 7
CHK2 34 4
MST2 34 1
Lck 33 1
IR 33 7
MELK 29 4
CAMK1 27 0
PIM3 27 5
SmMLCK 25 1
NUAK1 24 3
TrkA 20 8
PIM1 18 3
PIM2 12 2
RSK2 11 1
ERK8
9
0
CLK2
7
5
CDK2-Cyclin A
6
2
RSK1
6
0
IKK beta
4
2
JAK2
4
2