Inhibitor | TG003  

Screen Conc: 1.00µM

Kinase	% Activity Remaining	Standard Deviation
AMPK	114	8
ASK1	97	0
Aurora A	105	9
Aurora B	98	10
BRSK1	113	5
BRSK2	98	4
BTK	115	8
CAMK1	82	1
CAMKK beta	100	6
CDK2-Cyclin A	129	3
CHK1	117	3
CHK2	109	0
CK1 delta	19	0
CK2	107	6
CLK2	18	1
CSK	112	5
DAPK1	80	10
DYRK1A	16	0
DYRK2	12	3
DYRK3	23	10
EF2K	115	10
EPH-A2	116	10
EPH-A4	116	13
EPH-B1	105	9
EPH-B2	128	4
EPH-B3	91	14
EPH-B4	116	1
ERK1	114	15
ERK2	74	1
ERK8	93	9
FGF-R1	86	9
GCK	112	3
GSK3 beta	86	10
HER4	94	11
HIPK1	104	5
HIPK2	98	7
HIPK3	114	10
IGF-1R	120	11
IKK beta	98	1
IKK epsilon	106	2
IR	123	14
IRAK4	112	4
IRR	45	2
JAK2	110	11
JNK1	92	4
JNK2	104	10
JNK3	105	6
Lck	105	14
LKB1	113	2
MAPKAP-K2	116	6
MAPKAP-K3	119	5
MARK1	91	10
MARK2	89	4
MARK3	94	7
MARK4	94	13
MEKK1	109	10
MELK	119	3
MINK1	122	14
MKK1	99	4
MKK2	107	6
MKK6	92	7
MLK1	108	14
MLK3	93	6
MNK1	95	10
MNK2	109	4
MSK1	115	4
MST2	104	9
MST4	106	1
NEK2a	77	1
NEK6	105	6
NUAK1	82	3
p38 alpha MAPK	80	0
p38 beta MAPK	97	2
p38 delta MAPK	104	1
p38 gamma MAPK	128	3
PAK2	105	2
PAK4	94	1
PAK5	113	0
PAK6	105	12
PDK1	101	3
PHK	108	2
PIM1	21	2
PIM2	105	7
PIM3	30	1
PKA	91	5
PKB alpha	107	7
PKB beta	88	8
PKC alpha	109	8
PKC zeta	106	6
PKD1	57	2
PLK1	119	6
PRAK	117	12
PRK2	97	2
RIPK2	100	5
ROCK 2	88	1
RSK1	101	7
RSK2	79	2
S6K1	99	3
SGK1	101	6
SmMLCK	82	3
Src	79	3
SRPK1	91	2
SYK	109	8
TAK1	118	4
TAO1	70	9
TBK1	118	1
TrkA	111	7
TTK	72	4
VEGFR1	89	5
YES1	100	4

Screen Conc: 10.00µM

Kinase	% Activity Remaining	Standard Deviation
AMPK	92	9
ASK1	98	1
Aurora A	106	13
Aurora B	97	11
BRSK1	84	5
BRSK2	99	4
BTK	91	2
CAMK1	82	5
CAMKK beta	91	0
CDK2-Cyclin A	103	9
CHK1	99	5
CHK2	72	1
CK1 delta	9	0
CK2	73	5
CLK2	3	0
CSK	88	10
DAPK1	74	6
DYRK1A	3	0
DYRK2	2	0
DYRK3	6	0
EF2K	96	4
EPH-A2	104	11
EPH-A4	118	10
EPH-B1	112	9
EPH-B2	110	5
EPH-B3	105	7
EPH-B4	100	14
ERK1	104	11
ERK2	80	8
ERK8	23	3
FGF-R1	116	11
GCK	72	6
GSK3 beta	41	3
HER4	95	9
HIPK1	86	3
HIPK2	60	3
HIPK3	87	6
IGF-1R	113	13
IKK beta	92	9
IKK epsilon	105	6
IR	118	2
IRAK4	98	3
IRR	39	6
JAK2	95	6
JNK1	92	1
JNK2	95	5
JNK3	96	8
Lck	109	9
LKB1	79	7
MAPKAP-K2	101	4
MAPKAP-K3	97	7
MARK1	86	7
MARK2	85	12
MARK3	95	9
MARK4	86	3
MEKK1	101	12
MELK	61	11
MINK1	82	8
MKK1	98	4
MKK2	80	4
MKK6	119	11
MLK1	105	2
MLK3	85	2
MNK1	99	14
MNK2	103	2
MSK1	79	9
MST2	101	14
MST4	120	15
NEK2a	81	12
NEK6	108	6
NUAK1	88	14
p38 alpha MAPK	83	2
p38 beta MAPK	93	0
p38 delta MAPK	69	3
p38 gamma MAPK	82	5
PAK2	97	10
PAK4	99	1
PAK5	89	2
PAK6	93	2
PDK1	104	4
PHK	105	3
PIM1	11	2
PIM2	47	5
PIM3	12	1
PKA	93	4
PKB alpha	87	6
PKB beta	83	5
PKC alpha	109	4
PKC zeta	97	7
PKD1	22	2
PLK1	108	1
PRAK	97	3
PRK2	74	10
RIPK2	63	11
ROCK 2	90	0
RSK1	73	4
RSK2	89	9
S6K1	94	5
SGK1	103	1
SmMLCK	82	6
Src	83	2
SRPK1	94	0
SYK	110	12
TAK1	82	1
TAO1	49	2
TBK1	87	9
TrkA	98	12
TTK	68	5
VEGFR1	85	13
YES1	100	6