Compound name | Brutto | MW | CAS | PubChem CID | Action | Reference | Reference |
---|---|---|---|---|---|---|---|
BAY-11-7082 | C10H9NO2S | 207.20 | 19542-67-7 | 5353431 | NFKBIA | Kamthong P.J. (2001) Biochem. J. 356 | Izban K.F. (2000) Hum. Pathol. 31 1482 |
Kinase | % Activity Remaining Sort descending | Standard Deviation |
---|---|---|
RSK2 |
8
|
0 |
PKB beta |
8
|
1 |
Aurora A | 14 | 0 |
CAMK1 | 19 | 2 |
NUAK1 | 20 | 1 |
MINK1 | 27 | 4 |
IKK epsilon | 35 | 1 |
VEGFR1 | 40 | 9 |
BRSK2 | 41 | 7 |
MST2 | 51 | 5 |
MARK4 | 58 | 3 |
BTK | 58 | 6 |
MST4 | 61 | 6 |
GCK | 67 | 6 |
HER4 | 68 | 2 |
MARK2 | 70 | 1 |
PRK2 | 70 | 5 |
PIM1 | 71 | 3 |
PKD1 | 72 | 5 |
BRSK1 | 73 | 6 |
DAPK1 | 73 | 6 |
TBK1 | 75 | 6 |
EPH-A2 | 75 | 7 |
LKB1 | 75 | 4 |
PKC alpha | 75 | 0 |
MAPKAP-K3 | 75 | 0 |
PRAK | 76 | 3 |
AMPK | 76 | 4 |
DYRK2 | 78 | 5 |
SYK | 78 | 1 |
MLK1 | 78 | 2 |
JNK2 | 78 | 5 |
ERK2 | 79 | 2 |
MSK1 | 79 | 5 |
CHK1 | 79 | 2 |
PAK6 | 80 | 7 |
RIPK2 | 80 | 0 |
TAO1 | 81 | 3 |
ROCK 2 | 82 | 7 |
PIM3 | 82 | 1 |
HIPK1 | 82 | 4 |
PAK2 | 83 | 5 |
PIM2 | 83 | 7 |
JNK3 | 83 | 0 |
S6K1 | 84 | 2 |
JAK2 | 84 | 3 |
SmMLCK | 85 | 9 |
EF2K | 85 | 4 |
MKK6 | 85 | 1 |
RSK1 | 86 | 1 |
TTK | 86 | 3 |
CHK2 | 86 | 0 |
DYRK1A | 86 | 3 |
CDK2-Cyclin A | 87 | 8 |
p38 beta MAPK | 87 | 4 |
IKK beta | 87 | 2 |
EPH-B4 | 87 | 5 |
IRR | 87 | 3 |
TrkA | 87 | 7 |
p38 alpha MAPK | 88 | 7 |
NEK2a | 88 | 10 |
HIPK3 | 88 | 7 |
PAK5 | 89 | 8 |
PKA | 89 | 6 |
MNK1 | 89 | 1 |
MELK | 89 | 13 |
MKK2 | 89 | 7 |
PDK1 | 90 | 4 |
PKB alpha | 90 | 4 |
SRPK1 | 90 | 2 |
PKC zeta | 92 | 2 |
NEK6 | 92 | 1 |
CSK | 92 | 10 |
FGF-R1 | 92 | 11 |
MKK1 | 92 | 11 |
MAPKAP-K2 | 92 | 0 |
IRAK4 | 92 | 2 |
PLK1 | 93 | 5 |
p38 delta MAPK | 93 | 1 |
MLK3 | 93 | 8 |
EPH-B1 | 94 | 3 |
MEKK1 | 94 | 6 |
PAK4 | 95 | 10 |
EPH-A4 | 95 | 4 |
MARK3 | 95 | 7 |
IGF-1R | 95 | 2 |
DYRK3 | 96 | 3 |
MNK2 | 96 | 11 |
HIPK2 | 96 | 5 |
CLK2 | 96 | 6 |
EPH-B3 | 97 | 6 |
p38 gamma MAPK | 97 | 6 |
CK1 delta | 97 | 6 |
CAMKK beta | 99 | 1 |
JNK1 | 99 | 1 |
TAK1 | 99 | 6 |
SGK1 | 99 | 6 |
MARK1 | 100 | 1 |
GSK3 beta | 101 | 3 |
Aurora B | 101 | 14 |
ASK1 | 101 | 5 |
ERK8 | 101 | 6 |
ERK1 | 102 | 8 |
CK2 | 104 | 4 |
IR | 105 | 10 |
PHK | 106 | 5 |
Lck | 107 | 4 |
EPH-B2 | 112 | 4 |
YES1 | 158 | 14 |
Src | 162 | 6 |
Kinase | % Activity Remaining Sort descending | Standard Deviation |
---|---|---|
CAMK1 | 59 | 13 |
PIM3 | 74 | 6 |
IGF-1R | 77 | 40 |
RSK2 | 79 | 2 |
VEGFR1 | 80 | 1 |
MARK2 | 80 | 11 |
BRSK1 | 80 | 11 |
p38 beta MAPK | 81 | 15 |
BTK | 81 | 3 |
Aurora B | 82 | 12 |
PKD1 | 83 | 1 |
PAK4 | 83 | 10 |
ERK2 | 84 | 5 |
CDK2-Cyclin A | 84 | 4 |
JNK2 | 85 | 3 |
PKB beta | 86 | 15 |
MLK1 | 86 | 13 |
PAK6 | 87 | 4 |
MEKK1 | 88 | 2 |
SGK1 | 88 | 10 |
MST4 | 89 | 6 |
MAPKAP-K3 | 89 | 8 |
MST2 | 90 | 16 |
FGF-R1 | 90 | 5 |
MARK3 | 90 | 3 |
HIPK3 | 90 | 3 |
PKA | 91 | 0 |
PDK1 | 91 | 4 |
JNK1 | 91 | 7 |
PHK | 91 | 3 |
EPH-B3 | 92 | 1 |
LKB1 | 93 | 1 |
MLK3 | 93 | 7 |
NUAK1 | 93 | 5 |
GSK3 beta | 93 | 6 |
MAPKAP-K2 | 93 | 7 |
SYK | 94 | 3 |
AMPK | 94 | 5 |
TBK1 | 94 | 1 |
MSK1 | 95 | 6 |
IRAK4 | 95 | 1 |
p38 delta MAPK | 95 | 8 |
MARK4 | 95 | 1 |
MNK2 | 95 | 3 |
PKC alpha | 95 | 6 |
ROCK 2 | 96 | 7 |
DYRK1A | 96 | 16 |
DYRK2 | 96 | 0 |
PAK2 | 96 | 15 |
HIPK2 | 97 | 4 |
PAK5 | 97 | 7 |
EPH-A2 | 98 | 6 |
PRAK | 98 | 13 |
CSK | 98 | 2 |
RSK1 | 98 | 11 |
IRR | 99 | 1 |
CHK2 | 99 | 6 |
IR | 99 | 7 |
JAK2 | 99 | 9 |
NEK6 | 100 | 12 |
p38 alpha MAPK | 100 | 13 |
PKC zeta | 100 | 10 |
S6K1 | 100 | 16 |
PRK2 | 100 | 0 |
MELK | 101 | 6 |
IKK beta | 101 | 10 |
CK1 delta | 101 | 3 |
EPH-B2 | 101 | 8 |
PKB alpha | 102 | 4 |
CAMKK beta | 102 | 6 |
IKK epsilon | 103 | 1 |
GCK | 103 | 1 |
MINK1 | 103 | 3 |
PIM2 | 103 | 9 |
CK2 | 103 | 2 |
EF2K | 103 | 13 |
CLK2 | 103 | 1 |
Aurora A | 103 | 14 |
PIM1 | 104 | 5 |
MARK1 | 104 | 2 |
SmMLCK | 104 | 13 |
NEK2a | 104 | 0 |
MKK1 | 105 | 8 |
EPH-A4 | 106 | 1 |
BRSK2 | 106 | 4 |
DAPK1 | 107 | 13 |
SRPK1 | 107 | 6 |
JNK3 | 107 | 20 |
TTK | 107 | 14 |
Lck | 108 | 10 |
TAK1 | 108 | 24 |
HIPK1 | 108 | 18 |
PLK1 | 108 | 1 |
DYRK3 | 108 | 3 |
RIPK2 | 109 | 1 |
ERK8 | 110 | 7 |
p38 gamma MAPK | 112 | 9 |
CHK1 | 113 | 18 |
HER4 | 117 | 11 |
MNK1 | 117 | 16 |
ERK1 | 121 | 5 |
TrkA | 124 | 5 |
EPH-B4 | 125 | 4 |
YES1 | 127 | 34 |
Src | 177 | 4 |