Inhibitor | PP3  

Compound name Brutto MW CAS PubChem CID Action Reference Reference
PP3   C11H9N5 211.22 5334-30-5 4879 Src Hou (2007) Neurosci Lett 420 235

Screening Results Chart

Screening Results Tables

Screen Conc: 10.00µM
Kinase % Activity Remaining Standard Deviation
AMPK 105 1
Aurora A 83 9
Aurora B 83 10
BRSK1 60 1
BRSK2 69 4
BTK 83 22
CAMK1 87 18
CAMKK beta 116 11
CDK2-Cyclin A 91 10
CHK1 96 7
CHK2 115 6
CK1 delta 19 1
CK2 38 1
CSK 111 3
DYRK1A 52 8
DYRK2 53 7
DYRK3 47 4
EF2K 64 6
EPH-A2 113 10
EPH-B3 108 7
ERK1 84 8
ERK2 85 24
ERK8 68 7
FGF-R1 101 18
GCK 67 10
GSK3 beta 93 2
HER4 67 5
HIPK1 112 5
HIPK2 76 4
HIPK3 110 6
IGF-1R 77 6
IKK beta 82 3
IKK epsilon 95 8
IR 87 13
IRAK4 83 5
IRR 60 3
JNK1 95 3
JNK2 128 4
JNK3 100 1
Lck 75 11
LKB1 100 14
MAPKAP-K2 108 2
MAPKAP-K3 97 11
MARK2 100 2
MARK3 88 10
MARK4 82 3
MELK 94 17
MINK1 77 15
MKK1 118 32
MLK1 83 0
MLK3 83 10
MNK1 34 1
MNK2 88 9
MSK1 90 2
MST2 96 13
MST4 124 8
NEK2a 121 1
NEK6 80 2
NUAK1 69 0
p38 alpha MAPK 94 2
p38 beta MAPK 96 8
p38 delta MAPK 91 1
p38 gamma MAPK 102 7
PAK2 104 1
PAK4 83 9
PAK5 92 1
PAK6 109 14
PDK1 104 5
PHK 89 0
PIM1 85 12
PIM2 89 1
PIM3 90 1
PKA 91 4
PKB alpha 105 7
PKB beta 113 11
PKC alpha 95 3
PKC zeta 96 6
PKD1 121 23
PLK1 96 11
PRAK 80 10
PRK2 70 11
RIPK2 42 4
ROCK 2 65 8
RSK1 108 13
RSK2 79 7
S6K1 73 2
SGK1 86 1
SmMLCK 94 12
Src 81 13
SRPK1 121 14
SYK 110 11
TBK1 103 2
TTK 83 5
VEGFR1 114 10
YES1 80 4
Screen Conc: 20.00µM
Kinase % Activity Remaining Standard Deviation
AMPK 98 6
Aurora A 66 0
Aurora B 61 4
BRSK1 40 0
BRSK2 52 5
BTK 59 5
CAMK1 89 4
CAMKK beta 96 10
CDK2-Cyclin A 91 6
CHK1 97 8
CHK2 107 20
CK1 delta 14 4
CK2 26 6
CSK 98 9
DYRK1A 30 4
DYRK2 30 3
DYRK3 32 1
EF2K 53 4
EPH-A2 102 14
EPH-B3 95 10
ERK1 96 22
ERK2 77 2
ERK8 56 5
FGF-R1 96 1
GCK 57 4
GSK3 beta 104 18
HER4 50 4
HIPK1 95 4
HIPK2 64 1
HIPK3 117 3
IGF-1R 66 9
IKK beta 77 7
IKK epsilon 92 6
IR 60 6
IRAK4 72 0
IRR 48 5
JNK1 88 8
JNK2 111 2
JNK3 97 12
Lck 48 7
LKB1 81 0
MAPKAP-K2 110 4
MAPKAP-K3 101 4
MARK2 88 4
MARK3 78 0
MARK4 90 6
MELK 67 25
MINK1 54 6
MKK1 94 13
MLK1 54 1
MLK3 57 0
MNK1 24 4
MNK2 81 15
MSK1 88 12
MST2 81 11
MST4 119 3
NEK2a 115 4
NEK6 92 18
NUAK1 55 0
p38 alpha MAPK 89 8
p38 beta MAPK 84 6
p38 delta MAPK 93 7
p38 gamma MAPK 108 4
PAK2 107 11
PAK4 74 5
PAK5 78 8
PAK6 103 6
PDK1 92 6
PHK 73 0
PIM1 77 3
PIM2 93 5
PIM3 69 1
PKA 74 6
PKB alpha 94 3
PKB beta 98 34
PKC alpha 77 5
PKC zeta 99 1
PKD1 83 0
PLK1 91 2
PRAK 94 17
PRK2 58 4
RIPK2 31 3
ROCK 2 52 0
RSK1 103 7
RSK2 92 19
S6K1 65 1
SGK1 83 0
SmMLCK 69 33
Src 61 0
SRPK1 92 33
SYK 120 15
TBK1 91 4
TTK 75 2
VEGFR1 95 7
YES1 64 12