Compound name | Brutto | MW | CAS | PubChem CID | Action | Reference | Reference |
---|---|---|---|---|---|---|---|
PP3 | C11H9N5 | 211.22 | 5334-30-5 | 4879 | Src | Hou (2007) Neurosci Lett 420 235 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
AMPK | 105 | 1 |
Aurora A | 83 | 9 |
Aurora B | 83 | 10 |
BRSK1 | 60 | 1 |
BRSK2 | 69 | 4 |
BTK | 83 | 22 |
CAMK1 | 87 | 18 |
CAMKK beta | 116 | 11 |
CDK2-Cyclin A | 91 | 10 |
CHK1 | 96 | 7 |
CHK2 | 115 | 6 |
CK1 delta | 19 | 1 |
CK2 | 38 | 1 |
CSK | 111 | 3 |
DYRK1A | 52 | 8 |
DYRK2 | 53 | 7 |
DYRK3 | 47 | 4 |
EF2K | 64 | 6 |
EPH-A2 | 113 | 10 |
EPH-B3 | 108 | 7 |
ERK1 | 84 | 8 |
ERK2 | 85 | 24 |
ERK8 | 68 | 7 |
FGF-R1 | 101 | 18 |
GCK | 67 | 10 |
GSK3 beta | 93 | 2 |
HER4 | 67 | 5 |
HIPK1 | 112 | 5 |
HIPK2 | 76 | 4 |
HIPK3 | 110 | 6 |
IGF-1R | 77 | 6 |
IKK beta | 82 | 3 |
IKK epsilon | 95 | 8 |
IR | 87 | 13 |
IRAK4 | 83 | 5 |
IRR | 60 | 3 |
JNK1 | 95 | 3 |
JNK2 | 128 | 4 |
JNK3 | 100 | 1 |
Lck | 75 | 11 |
LKB1 | 100 | 14 |
MAPKAP-K2 | 108 | 2 |
MAPKAP-K3 | 97 | 11 |
MARK2 | 100 | 2 |
MARK3 | 88 | 10 |
MARK4 | 82 | 3 |
MELK | 94 | 17 |
MINK1 | 77 | 15 |
MKK1 | 118 | 32 |
MLK1 | 83 | 0 |
MLK3 | 83 | 10 |
MNK1 | 34 | 1 |
MNK2 | 88 | 9 |
MSK1 | 90 | 2 |
MST2 | 96 | 13 |
MST4 | 124 | 8 |
NEK2a | 121 | 1 |
NEK6 | 80 | 2 |
NUAK1 | 69 | 0 |
p38 alpha MAPK | 94 | 2 |
p38 beta MAPK | 96 | 8 |
p38 delta MAPK | 91 | 1 |
p38 gamma MAPK | 102 | 7 |
PAK2 | 104 | 1 |
PAK4 | 83 | 9 |
PAK5 | 92 | 1 |
PAK6 | 109 | 14 |
PDK1 | 104 | 5 |
PHK | 89 | 0 |
PIM1 | 85 | 12 |
PIM2 | 89 | 1 |
PIM3 | 90 | 1 |
PKA | 91 | 4 |
PKB alpha | 105 | 7 |
PKB beta | 113 | 11 |
PKC alpha | 95 | 3 |
PKC zeta | 96 | 6 |
PKD1 | 121 | 23 |
PLK1 | 96 | 11 |
PRAK | 80 | 10 |
PRK2 | 70 | 11 |
RIPK2 | 42 | 4 |
ROCK 2 | 65 | 8 |
RSK1 | 108 | 13 |
RSK2 | 79 | 7 |
S6K1 | 73 | 2 |
SGK1 | 86 | 1 |
SmMLCK | 94 | 12 |
Src | 81 | 13 |
SRPK1 | 121 | 14 |
SYK | 110 | 11 |
TBK1 | 103 | 2 |
TTK | 83 | 5 |
VEGFR1 | 114 | 10 |
YES1 | 80 | 4 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
AMPK | 98 | 6 |
Aurora A | 66 | 0 |
Aurora B | 61 | 4 |
BRSK1 | 40 | 0 |
BRSK2 | 52 | 5 |
BTK | 59 | 5 |
CAMK1 | 89 | 4 |
CAMKK beta | 96 | 10 |
CDK2-Cyclin A | 91 | 6 |
CHK1 | 97 | 8 |
CHK2 | 107 | 20 |
CK1 delta | 14 | 4 |
CK2 | 26 | 6 |
CSK | 98 | 9 |
DYRK1A | 30 | 4 |
DYRK2 | 30 | 3 |
DYRK3 | 32 | 1 |
EF2K | 53 | 4 |
EPH-A2 | 102 | 14 |
EPH-B3 | 95 | 10 |
ERK1 | 96 | 22 |
ERK2 | 77 | 2 |
ERK8 | 56 | 5 |
FGF-R1 | 96 | 1 |
GCK | 57 | 4 |
GSK3 beta | 104 | 18 |
HER4 | 50 | 4 |
HIPK1 | 95 | 4 |
HIPK2 | 64 | 1 |
HIPK3 | 117 | 3 |
IGF-1R | 66 | 9 |
IKK beta | 77 | 7 |
IKK epsilon | 92 | 6 |
IR | 60 | 6 |
IRAK4 | 72 | 0 |
IRR | 48 | 5 |
JNK1 | 88 | 8 |
JNK2 | 111 | 2 |
JNK3 | 97 | 12 |
Lck | 48 | 7 |
LKB1 | 81 | 0 |
MAPKAP-K2 | 110 | 4 |
MAPKAP-K3 | 101 | 4 |
MARK2 | 88 | 4 |
MARK3 | 78 | 0 |
MARK4 | 90 | 6 |
MELK | 67 | 25 |
MINK1 | 54 | 6 |
MKK1 | 94 | 13 |
MLK1 | 54 | 1 |
MLK3 | 57 | 0 |
MNK1 | 24 | 4 |
MNK2 | 81 | 15 |
MSK1 | 88 | 12 |
MST2 | 81 | 11 |
MST4 | 119 | 3 |
NEK2a | 115 | 4 |
NEK6 | 92 | 18 |
NUAK1 | 55 | 0 |
p38 alpha MAPK | 89 | 8 |
p38 beta MAPK | 84 | 6 |
p38 delta MAPK | 93 | 7 |
p38 gamma MAPK | 108 | 4 |
PAK2 | 107 | 11 |
PAK4 | 74 | 5 |
PAK5 | 78 | 8 |
PAK6 | 103 | 6 |
PDK1 | 92 | 6 |
PHK | 73 | 0 |
PIM1 | 77 | 3 |
PIM2 | 93 | 5 |
PIM3 | 69 | 1 |
PKA | 74 | 6 |
PKB alpha | 94 | 3 |
PKB beta | 98 | 34 |
PKC alpha | 77 | 5 |
PKC zeta | 99 | 1 |
PKD1 | 83 | 0 |
PLK1 | 91 | 2 |
PRAK | 94 | 17 |
PRK2 | 58 | 4 |
RIPK2 | 31 | 3 |
ROCK 2 | 52 | 0 |
RSK1 | 103 | 7 |
RSK2 | 92 | 19 |
S6K1 | 65 | 1 |
SGK1 | 83 | 0 |
SmMLCK | 69 | 33 |
Src | 61 | 0 |
SRPK1 | 92 | 33 |
SYK | 120 | 15 |
TBK1 | 91 | 4 |
TTK | 75 | 2 |
VEGFR1 | 95 | 7 |
YES1 | 64 | 12 |