Inhibitor | AG1478 (Tyrphostin)  

Screen Conc: 10.00µM

Kinase Sort ascending	% Activity Remaining	Standard Deviation
YES1	5	0
VEGFR1	5	0
TTK	79	1
TBK1	40	7
SYK	107	3
SRPK1	98	2
Src	8	1
SmMLCK	14	0
SGK1	83	6
S6K1	86	1
RSK2	82	1
RSK1	74	14
ROCK 2	61	9
RIPK2	14	3
PRK2	111	3
PRAK	88	12
PLK1	74	10
PKD1	32	2
PKC zeta	106	7
PKC alpha	74	3
PKB beta	93	10
PKB alpha	86	10
PKA	107	7
PIM3	29	4
PIM2	96	3
PIM1	40	5
PHK	23	3
PDK1	79	5
PAK6	98	1
PAK5	81	2
PAK4	87	6
PAK2	85	0
p38 gamma MAPK	105	9
p38 delta MAPK	97	6
p38 beta MAPK	38	0
p38 alpha MAPK	12	1
NUAK1	39	4
NEK6	100	1
NEK2a	82	3
MST4	62	21
MST2	35	0
MSK1	96	2
MNK2	36	5
MNK1	7	0
MLK3	75	14
MLK1	24	0
MKK1	52	0
MINK1	14	0
MELK	55	0
MARK4	79	4
MARK3	61	0
MARK2	102	3
MAPKAP-K3	98	4
MAPKAP-K2	89	4
LKB1	99	19
Lck	34	0
JNK3	73	8
JNK2	78	7
JNK1	105	7
IRR	78	0
IRAK4	11	0
IR	81	2
IKK epsilon	67	3
IKK beta	89	0
IGF-1R	95	7
HIPK3	96	2
HIPK2	76	2
HIPK1	120	59
HER4	3	1
GSK3 beta	75	5
GCK	43	2
FGF-R1	44	5
ERK8	61	9
ERK2	39	6
ERK1	75	0
EPH-B3	63	0
EPH-A2	18	0
EF2K	113	6
DYRK3	23	3
DYRK2	33	3
DYRK1A	45	2
CSK	57	13
CK2	90	2
CK1 delta	65	11
CHK2	23	0
CHK1	78	4
CDK2-Cyclin A	91	8
CAMKK beta	52	2
CAMK1	94	1
BTK	15	0
BRSK2	41	3
BRSK1	40	2
Aurora B	46	5
Aurora A	15	0
AMPK	68	1

Screen Conc: 1.00µM

Kinase Sort ascending	% Activity Remaining	Standard Deviation
YES1	42	4
VEGFR1	31	0
TTK	83	2
TrkA	65	9
TBK1	83	1
TAO1	93	8
TAK1	91	7
SYK	110	3
SRPK1	98	5
Src	39	1
SmMLCK	49	0
SGK1	106	3
S6K1	82	2
RSK2	83	7
RSK1	82	2
ROCK 2	86	2
RIPK2	10	1
PRK2	86	3
PRAK	87	0
PLK1	104	3
PKD1	87	3
PKC zeta	104	6
PKC alpha	79	7
PKB beta	69	11
PKB alpha	102	9
PKA	97	15
PIM3	75	12
PIM2	102	2
PIM1	79	14
PHK	85	3
PDK1	92	5
PAK6	99	4
PAK5	90	0
PAK4	98	5
PAK2	101	11
p38 gamma MAPK	98	3
p38 delta MAPK	99	4
p38 beta MAPK	68	10
p38 alpha MAPK	37	2
NUAK1	80	5
NEK6	90	2
NEK2a	86	6
MST4	100	12
MST2	76	0
MSK1	87	7
MNK2	47	4
MNK1	44	3
MLK3	53	5
MLK1	63	3
MKK6	103	4
MKK2	84	7
MKK1	94	1
MINK1	62	4
MELK	91	7
MEKK1	88	5
MARK4	104	14
MARK3	83	3
MARK2	79	6
MARK1	101	4
MAPKAP-K3	88	2
MAPKAP-K2	81	6
LKB1	93	11
Lck	54	2
JNK3	76	6
JNK2	79	3
JNK1	100	0
JAK2	61	1
IRR	93	5
IRAK4	38	0
IR	105	5
IKK epsilon	82	4
IKK beta	90	4
IGF-1R	104	13
HIPK3	101	0
HIPK2	100	4
HIPK1	93	7
HER4	25	0
GSK3 beta	90	13
GCK	82	2
FGF-R1	75	1
ERK8	96	9
ERK2	94	5
ERK1	84	11
EPH-B4	67	2
EPH-B3	63	11
EPH-B2	57	10
EPH-B1	107	13
EPH-A4	58	1
EPH-A2	77	1
EF2K	88	3
DYRK3	76	6
DYRK2	74	3
DYRK1A	90	5
DAPK1	88	2
CSK	86	9
CLK2	95	3
CK2	99	0
CK1 delta	100	5
CHK2	81	5
CHK1	81	4
CDK2-Cyclin A	112	7
CAMKK beta	97	1
CAMK1	106	6
BTK	69	0
BRSK2	79	4
BRSK1	74	9
Aurora B	53	3
Aurora A	82	6
ASK1	104	1
AMPK	80	8