Inhibitor | AG1478 (Tyrphostin)  

Screen Conc: 10.00µM

Kinase	% Activity Remaining Sort descending	Standard Deviation
HER4	3	1
VEGFR1	5	0
YES1	5	0
MNK1	7	0
Src	8	1
IRAK4	11	0
p38 alpha MAPK	12	1
RIPK2	14	3
SmMLCK	14	0
MINK1	14	0
BTK	15	0
Aurora A	15	0
EPH-A2	18	0
DYRK3	23	3
PHK	23	3
CHK2	23	0
MLK1	24	0
PIM3	29	4
PKD1	32	2
DYRK2	33	3
Lck	34	0
MST2	35	0
MNK2	36	5
p38 beta MAPK	38	0
NUAK1	39	4
ERK2	39	6
TBK1	40	7
BRSK1	40	2
PIM1	40	5
BRSK2	41	3
GCK	43	2
FGF-R1	44	5
DYRK1A	45	2
Aurora B	46	5
CAMKK beta	52	2
MKK1	52	0
MELK	55	0
CSK	57	13
MARK3	61	0
ERK8	61	9
ROCK 2	61	9
MST4	62	21
EPH-B3	63	0
CK1 delta	65	11
IKK epsilon	67	3
AMPK	68	1
JNK3	73	8
RSK1	74	14
PKC alpha	74	3
PLK1	74	10
ERK1	75	0
GSK3 beta	75	5
MLK3	75	14
HIPK2	76	2
CHK1	78	4
IRR	78	0
JNK2	78	7
PDK1	79	5
MARK4	79	4
TTK	79	1
IR	81	2
PAK5	81	2
RSK2	82	1
NEK2a	82	3
SGK1	83	6
PAK2	85	0
PKB alpha	86	10
S6K1	86	1
PAK4	87	6
PRAK	88	12
MAPKAP-K2	89	4
IKK beta	89	0
CK2	90	2
CDK2-Cyclin A	91	8
PKB beta	93	10
CAMK1	94	1
IGF-1R	95	7
HIPK3	96	2
PIM2	96	3
MSK1	96	2
p38 delta MAPK	97	6
MAPKAP-K3	98	4
PAK6	98	1
SRPK1	98	2
LKB1	99	19
NEK6	100	1
MARK2	102	3
JNK1	105	7
p38 gamma MAPK	105	9
PKC zeta	106	7
PKA	107	7
SYK	107	3
PRK2	111	3
EF2K	113	6
HIPK1	120	59

Screen Conc: 1.00µM

Kinase	% Activity Remaining Sort descending	Standard Deviation
RIPK2	10	1
HER4	25	0
VEGFR1	31	0
p38 alpha MAPK	37	2
IRAK4	38	0
Src	39	1
YES1	42	4
MNK1	44	3
MNK2	47	4
SmMLCK	49	0
Aurora B	53	3
MLK3	53	5
Lck	54	2
EPH-B2	57	10
EPH-A4	58	1
JAK2	61	1
MINK1	62	4
MLK1	63	3
EPH-B3	63	11
TrkA	65	9
EPH-B4	67	2
p38 beta MAPK	68	10
BTK	69	0
PKB beta	69	11
BRSK1	74	9
DYRK2	74	3
FGF-R1	75	1
PIM3	75	12
DYRK3	76	6
MST2	76	0
JNK3	76	6
EPH-A2	77	1
MARK2	79	6
PIM1	79	14
BRSK2	79	4
JNK2	79	3
PKC alpha	79	7
AMPK	80	8
NUAK1	80	5
MAPKAP-K2	81	6
CHK1	81	4
CHK2	81	5
Aurora A	82	6
RSK1	82	2
IKK epsilon	82	4
GCK	82	2
S6K1	82	2
TTK	83	2
RSK2	83	7
MARK3	83	3
TBK1	83	1
MKK2	84	7
ERK1	84	11
PHK	85	3
NEK2a	86	6
CSK	86	9
ROCK 2	86	2
PRK2	86	3
MSK1	87	7
PRAK	87	0
PKD1	87	3
MAPKAP-K3	88	2
MEKK1	88	5
DAPK1	88	2
EF2K	88	3
NEK6	90	2
IKK beta	90	4
PAK5	90	0
GSK3 beta	90	13
DYRK1A	90	5
MELK	91	7
TAK1	91	7
PDK1	92	5
LKB1	93	11
IRR	93	5
TAO1	93	8
HIPK1	93	7
ERK2	94	5
MKK1	94	1
CLK2	95	3
ERK8	96	9
CAMKK beta	97	1
PKA	97	15
p38 gamma MAPK	98	3
PAK4	98	5
SRPK1	98	5
p38 delta MAPK	99	4
PAK6	99	4
CK2	99	0
MST4	100	12
JNK1	100	0
CK1 delta	100	5
HIPK2	100	4
HIPK3	101	0
PAK2	101	11
MARK1	101	4
PKB alpha	102	9
PIM2	102	2
MKK6	103	4
IGF-1R	104	13
MARK4	104	14
ASK1	104	1
PKC zeta	104	6
PLK1	104	3
IR	105	5
CAMK1	106	6
SGK1	106	3
EPH-B1	107	13
SYK	110	3
CDK2-Cyclin A	112	7