Inhibitor | KU 0063794  

Compound name Brutto MW CAS PubChem CID Action Reference Reference
KU 0063794   C25H31N5O4 465.54 938440-64-3 16736978 mTOR Juan M. García-Martínez (2009) Biochem J. 421 29–42

Screening Results Chart

Screening Results Tables

Screen Conc: 10.00µM
Kinase % Activity Remaining Sort descending Standard Deviation
MSK1 11 7
MKK1 43 7
SGK1 64 6
IR 67 5
IRR 71 4
BRSK2 72 7
MELK 72 4
PIM3 75 7
MNK1 75 12
PAK4 75 4
PIM2 78 0
EPH-B3 78 4
DYRK1A 80 7
MAPKAP-K2 81 10
PAK5 81 3
BTK 81 21
NEK6 83 10
SYK 83 5
p38 beta MAPK 83 5
DYRK3 84 1
PKC zeta 84 0
CK2 85 12
PKA 85 12
RSK1 86 2
Src 86 5
NEK2a 86 2
CHK1 86 7
ROCK 2 86 5
MST4 86 8
PKC alpha 86 18
Aurora B 86 6
PRAK 87 8
FGF-R1 87 10
ERK1 87 1
p38 delta MAPK 87 4
TBK1 89 4
IKK beta 89 3
IGF-1R 89 1
HIPK2 89 1
PKB alpha 90 1
CDK2-Cyclin A 90 6
YES1 90 1
PDK1 91 2
GSK3 beta 91 5
p38 gamma MAPK 91 1
ERK2 92 9
VEGFR1 92 8
ERK8 92 5
MNK2 92 1
JNK1 93 4
MARK3 93 15
CAMKK beta 94 0
PLK1 94 2
SRPK1 94 2
DYRK2 96 12
CHK2 96 9
EPH-A2 96 2
p38 alpha MAPK 96 5
S6K1 98 4
PIM1 98 15
CSK 99 3
PAK6 100 24
IKK epsilon 100 5
CAMK1 101 6
PKD1 101 3
MST2 102 3
JNK2 103 13
RSK2 104 1
Lck 104 9
SmMLCK 104 3
PRK2 105 12
AMPK 106 3
PKB beta 107 9
EF2K 108 0
CK1 delta 109 12
PHK 116 3
Screen Conc: 1.00µM
Kinase % Activity Remaining Sort descending Standard Deviation
PRAK 67 4
Lck 69 5
p38 delta MAPK 72 1
NEK6 74 4
PAK6 75 3
ROCK 2 75 4
PLK1 76 2
SGK1 76 6
PKD1 80 4
JNK1 80 5
MST2 81 10
IR 81 1
SmMLCK 82 4
BTK 85 7
PIM2 86 11
PKC zeta 87 9
MNK2 87 5
CHK1 87 8
MST4 87 5
EF2K 88 7
ERK8 88 1
DYRK3 88 9
SYK 88 3
p38 gamma MAPK 89 8
HIPK2 89 5
PDK1 89 5
PHK 89 2
PIM1 89 4
CDK2-Cyclin A 89 5
BRSK2 90 1
CSK 90 1
MELK 91 6
VEGFR1 92 8
DYRK2 92 1
NEK2a 92 10
MARK3 93 6
DYRK1A 94 10
YES1 94 10
GSK3 beta 95 11
PRK2 95 5
CAMK1 96 1
MKK1 96 4
AMPK 97 1
TBK1 97 8
PKB beta 97 8
CHK2 97 2
MAPKAP-K2 98 3
PKB alpha 98 8
IKK epsilon 99 1
EPH-B3 100 8
RSK1 100 4
JNK2 101 4
SRPK1 101 1
p38 alpha MAPK 101 6
MSK1 101 6
PAK5 101 1
FGF-R1 102 8
ERK1 102 0
ERK2 102 8
RSK2 103 7
CK2 104 0
S6K1 104 11
IKK beta 104 3
IRR 105 7
PKC alpha 106 13
p38 beta MAPK 106 7
CAMKK beta 108 5
EPH-A2 108 8
PAK4 110 1
MNK1 111 0
CK1 delta 112 15
PIM3 114 12
PKA 115 7
IGF-1R 117 0