Inhibitor | KU 0063794  

Screen Conc: 1.00µM

Kinase	% Activity Remaining	Standard Deviation
AMPK	97	1
BRSK2	90	1
BTK	85	7
CAMK1	96	1
CAMKK beta	108	5
CDK2-Cyclin A	89	5
CHK1	87	8
CHK2	97	2
CK1 delta	112	15
CK2	104	0
CSK	90	1
DYRK1A	94	10
DYRK2	92	1
DYRK3	88	9
EF2K	88	7
EPH-A2	108	8
EPH-B3	100	8
ERK1	102	0
ERK2	102	8
ERK8	88	1
FGF-R1	102	8
GSK3 beta	95	11
HIPK2	89	5
IGF-1R	117	0
IKK beta	104	3
IKK epsilon	99	1
IR	81	1
IRR	105	7
JNK1	80	5
JNK2	101	4
Lck	69	5
MAPKAP-K2	98	3
MARK3	93	6
MELK	91	6
MKK1	96	4
MNK1	111	0
MNK2	87	5
MSK1	101	6
MST2	81	10
MST4	87	5
NEK2a	92	10
NEK6	74	4
p38 alpha MAPK	101	6
p38 beta MAPK	106	7
p38 delta MAPK	72	1
p38 gamma MAPK	89	8
PAK4	110	1
PAK5	101	1
PAK6	75	3
PDK1	89	5
PHK	89	2
PIM1	89	4
PIM2	86	11
PIM3	114	12
PKA	115	7
PKB alpha	98	8
PKB beta	97	8
PKC alpha	106	13
PKC zeta	87	9
PKD1	80	4
PLK1	76	2
PRAK	67	4
PRK2	95	5
ROCK 2	75	4
RSK1	100	4
RSK2	103	7
S6K1	104	11
SGK1	76	6
SmMLCK	82	4
SRPK1	101	1
SYK	88	3
TBK1	97	8
VEGFR1	92	8
YES1	94	10

Screen Conc: 10.00µM

Kinase	% Activity Remaining	Standard Deviation
AMPK	106	3
Aurora B	86	6
BRSK2	72	7
BTK	81	21
CAMK1	101	6
CAMKK beta	94	0
CDK2-Cyclin A	90	6
CHK1	86	7
CHK2	96	9
CK1 delta	109	12
CK2	85	12
CSK	99	3
DYRK1A	80	7
DYRK2	96	12
DYRK3	84	1
EF2K	108	0
EPH-A2	96	2
EPH-B3	78	4
ERK1	87	1
ERK2	92	9
ERK8	92	5
FGF-R1	87	10
GSK3 beta	91	5
HIPK2	89	1
IGF-1R	89	1
IKK beta	89	3
IKK epsilon	100	5
IR	67	5
IRR	71	4
JNK1	93	4
JNK2	103	13
Lck	104	9
MAPKAP-K2	81	10
MARK3	93	15
MELK	72	4
MKK1	43	7
MNK1	75	12
MNK2	92	1
MSK1	11	7
MST2	102	3
MST4	86	8
NEK2a	86	2
NEK6	83	10
p38 alpha MAPK	96	5
p38 beta MAPK	83	5
p38 delta MAPK	87	4
p38 gamma MAPK	91	1
PAK4	75	4
PAK5	81	3
PAK6	100	24
PDK1	91	2
PHK	116	3
PIM1	98	15
PIM2	78	0
PIM3	75	7
PKA	85	12
PKB alpha	90	1
PKB beta	107	9
PKC alpha	86	18
PKC zeta	84	0
PKD1	101	3
PLK1	94	2
PRAK	87	8
PRK2	105	12
ROCK 2	86	5
RSK1	86	2
RSK2	104	1
S6K1	98	4
SGK1	64	6
SmMLCK	104	3
Src	86	5
SRPK1	94	2
SYK	83	5
TBK1	89	4
VEGFR1	92	8
YES1	90	1