Inhibitor | Akt Inhibitor IV
Screening Results Tables
Screen Conc: 1.00µM
Kinase |
% Activity Remaining |
Standard Deviation |
AMPK |
98
|
0 |
Aurora B |
96
|
7 |
BRSK2 |
79
|
10 |
BTK |
98
|
4 |
CAMK1 |
94
|
2 |
CAMKK beta |
109
|
0 |
CDK2-Cyclin A |
88
|
1 |
CHK1 |
89
|
4 |
CHK2 |
99
|
11 |
CK1 delta |
98
|
2 |
CK2 |
104
|
12 |
CSK |
94
|
11 |
DYRK1A |
99
|
6 |
DYRK2 |
88
|
0 |
DYRK3 |
99
|
1 |
EF2K |
123
|
13 |
EPH-A2 |
86
|
11 |
EPH-B3 |
74
|
3 |
ERK1 |
104
|
11 |
ERK2 |
93
|
5 |
ERK8 |
91
|
5 |
FGF-R1 |
90
|
14 |
GCK |
80
|
1 |
GSK3 beta |
102
|
7 |
HER4 |
70
|
1 |
HIPK2 |
101
|
1 |
IGF-1R |
95
|
6 |
IKK beta |
72
|
0 |
IKK epsilon |
97
|
11 |
IR |
93
|
10 |
IRAK4 |
83
|
2 |
IRR |
102
|
1 |
JNK1 |
100
|
6 |
JNK2 |
95
|
6 |
Lck |
74
|
0 |
LKB1 |
97
|
9 |
MAPKAP-K2 |
93
|
1 |
MARK3 |
99
|
10 |
MELK |
109
|
2 |
MINK1 |
97
|
15 |
MKK1 |
68
|
0 |
MLK1 |
80
|
10 |
MLK3 |
126
|
3 |
MNK1 |
93
|
2 |
MNK2 |
89
|
3 |
MSK1 |
91
|
6 |
MST2 |
106
|
0 |
MST4 |
94
|
12 |
NEK2a |
102
|
7 |
NEK6 |
92
|
6 |
NUAK1 |
139
|
11 |
p38 alpha MAPK |
99
|
1 |
p38 beta MAPK |
105
|
6 |
p38 delta MAPK |
95
|
8 |
p38 gamma MAPK |
99
|
6 |
PAK4 |
104
|
1 |
PAK5 |
109
|
1 |
PAK6 |
99
|
1 |
PDK1 |
128
|
0 |
PHK |
90
|
0 |
PIM1 |
90
|
10 |
PIM2 |
99
|
1 |
PIM3 |
79
|
9 |
PKA |
104
|
6 |
PKB alpha |
99
|
16 |
PKB beta |
93
|
1 |
PKC alpha |
97
|
2 |
PKC zeta |
99
|
4 |
PKD1 |
102
|
4 |
PLK1 |
107
|
3 |
PRAK |
94
|
8 |
PRK2 |
99
|
1 |
ROCK 2 |
99
|
3 |
RSK1 |
80
|
4 |
RSK2 |
103
|
19 |
S6K1 |
83
|
4 |
SGK1 |
65
|
16 |
SmMLCK |
89
|
5 |
Src |
90
|
10 |
SRPK1 |
80
|
36 |
SYK |
89
|
9 |
TBK1 |
91
|
8 |
TTK |
109
|
10 |
VEGFR1 |
116
|
0 |
YES1 |
101
|
9 |
Screen Conc: 10.00µM
Kinase |
% Activity Remaining |
Standard Deviation |
AMPK |
92
|
8 |
Aurora B |
82
|
6 |
BRSK2 |
101
|
4 |
BTK |
148
|
30 |
CAMK1 |
22
|
1 |
CAMKK beta |
91
|
4 |
CDK2-Cyclin A |
89
|
0 |
CHK1 |
70
|
6 |
CHK2 |
90
|
4 |
CK1 delta |
108
|
10 |
CK2 |
95
|
3 |
CSK |
74
|
2 |
DYRK1A |
71
|
7 |
DYRK2 |
64
|
2 |
DYRK3 |
90
|
0 |
EF2K |
130
|
1 |
EPH-A2 |
72
|
6 |
EPH-B3 |
79
|
0 |
ERK1 |
100
|
7 |
ERK2 |
96
|
1 |
ERK8 |
85
|
4 |
FGF-R1 |
91
|
2 |
GCK |
64
|
0 |
GSK3 beta |
95
|
5 |
HER4 |
104
|
5 |
HIPK2 |
80
|
1 |
IGF-1R |
62
|
0 |
IKK beta |
65
|
0 |
IKK epsilon |
91
|
16 |
IR |
88
|
18 |
IRAK4 |
64
|
0 |
IRR |
88
|
2 |
JNK1 |
100
|
9 |
JNK2 |
91
|
3 |
Lck |
45
|
3 |
LKB1 |
89
|
6 |
MAPKAP-K2 |
85
|
4 |
MARK3 |
89
|
1 |
MELK |
63
|
9 |
MINK1 |
65
|
0 |
MKK1 |
42
|
0 |
MLK1 |
54
|
9 |
MLK3 |
88
|
1 |
MNK1 |
99
|
8 |
MNK2 |
75
|
2 |
MSK1 |
61
|
6 |
MST2 |
88
|
5 |
MST4 |
68
|
7 |
NEK2a |
63
|
12 |
NEK6 |
52
|
14 |
NUAK1 |
111
|
4 |
p38 alpha MAPK |
88
|
6 |
p38 beta MAPK |
100
|
4 |
p38 delta MAPK |
95
|
11 |
p38 gamma MAPK |
80
|
1 |
PAK4 |
94
|
11 |
PAK5 |
116
|
4 |
PAK6 |
113
|
3 |
PDK1 |
126
|
3 |
PHK |
74
|
5 |
PIM1 |
64
|
0 |
PIM2 |
90
|
12 |
PIM3 |
50
|
0 |
PKA |
91
|
4 |
PKB alpha |
53
|
24 |
PKB beta |
79
|
2 |
PKC alpha |
75
|
0 |
PKC zeta |
78
|
2 |
PKD1 |
50
|
12 |
PLK1 |
144
|
2 |
PRAK |
96
|
20 |
PRK2 |
76
|
7 |
ROCK 2 |
77
|
9 |
RSK1 |
47
|
4 |
RSK2 |
99
|
7 |
S6K1 |
44
|
9 |
SGK1 |
40
|
10 |
SmMLCK |
56
|
3 |
Src |
103
|
8 |
SRPK1 |
78
|
33 |
SYK |
59
|
16 |
TBK1 |
76
|
2 |
TTK |
92
|
1 |
VEGFR1 |
126
|
15 |
YES1 |
112
|
6 |