Inhibitor | AG1296 (Tyrphostin)  

Compound name Brutto MW CAS PubChem CID Action Reference Reference
AG1296 (Tyrphostin)   C16H14N2O2 266.29 146535-11-7 2049 PDGF Kovalenko M. (1994) Cancer Res. 54 6106 https://pubmed.ncbi.nlm.nih.gov/[pmid2]

Screening Results Chart

Screening Results Tables

Screen Conc: 10.00µM
Kinase % Activity Remaining Standard Deviation
AMPK 80 1
Aurora B 15 1
BRSK2 99 2
BTK 80 10
CAMK1 104 3
CAMKK beta 88 1
CDK2-Cyclin A 91 8
CHK1 95 0
CHK2 93 9
CK1 delta 54 2
CK2 80 2
CSK 105 0
DYRK1A 93 4
DYRK2 84 5
DYRK3 91 22
EF2K 103 10
EPH-A2 98 14
EPH-B3 86 10
ERK1 101 17
ERK2 105 3
ERK8 86 12
FGF-R1 94 18
GSK3 beta 113 4
HIPK2 98 0
IGF-1R 102 7
IKK beta 101 3
IKK epsilon 85 2
IR 70 7
IRR 75 9
JNK1 101 11
JNK2 113 10
Lck 82 1
MAPKAP-K2 107 11
MARK3 103 9
MELK 64 6
MKK1 92 10
MNK1 83 11
MNK2 74 0
MSK1 102 1
MST2 79 6
MST4 105 10
NEK2a 65 5
NEK6 116 27
p38 alpha MAPK 91 5
p38 beta MAPK 95 4
p38 delta MAPK 102 11
p38 gamma MAPK 110 6
PAK4 69 1
PAK5 74 2
PAK6 97 2
PDK1 110 5
PHK 101 10
PIM1 104 8
PIM2 108 1
PIM3 79 1
PKA 96 5
PKB alpha 104 2
PKB beta 98 0
PKC alpha 103 5
PKC zeta 94 1
PKD1 103 9
PLK1 96 3
PRAK 88 13
PRK2 95 9
ROCK 2 85 3
RSK1 75 2
RSK2 97 6
S6K1 106 17
SGK1 88 3
SmMLCK 84 26
Src 72 2
SRPK1 95 0
SYK 100 2
TBK1 64 4
VEGFR1 50 1
YES1 85 7