Inhibitor | AG1296 (Tyrphostin)
Screening Results Tables
Screen Conc: 10.00µM
| Kinase |
% Activity Remaining |
Standard Deviation |
| AMPK |
80
|
1 |
| Aurora B |
15
|
1 |
| BRSK2 |
99
|
2 |
| BTK |
80
|
10 |
| CAMK1 |
104
|
3 |
| CAMKK beta |
88
|
1 |
| CDK2-Cyclin A |
91
|
8 |
| CHK1 |
95
|
0 |
| CHK2 |
93
|
9 |
| CK1 delta |
54
|
2 |
| CK2 |
80
|
2 |
| CSK |
105
|
0 |
| DYRK1A |
93
|
4 |
| DYRK2 |
84
|
5 |
| DYRK3 |
91
|
22 |
| EF2K |
103
|
10 |
| EPH-A2 |
98
|
14 |
| EPH-B3 |
86
|
10 |
| ERK1 |
101
|
17 |
| ERK2 |
105
|
3 |
| ERK8 |
86
|
12 |
| FGF-R1 |
94
|
18 |
| GSK3 beta |
113
|
4 |
| HIPK2 |
98
|
0 |
| IGF-1R |
102
|
7 |
| IKK beta |
101
|
3 |
| IKK epsilon |
85
|
2 |
| IR |
70
|
7 |
| IRR |
75
|
9 |
| JNK1 |
101
|
11 |
| JNK2 |
113
|
10 |
| Lck |
82
|
1 |
| MAPKAP-K2 |
107
|
11 |
| MARK3 |
103
|
9 |
| MELK |
64
|
6 |
| MKK1 |
92
|
10 |
| MNK1 |
83
|
11 |
| MNK2 |
74
|
0 |
| MSK1 |
102
|
1 |
| MST2 |
79
|
6 |
| MST4 |
105
|
10 |
| NEK2a |
65
|
5 |
| NEK6 |
116
|
27 |
| p38 alpha MAPK |
91
|
5 |
| p38 beta MAPK |
95
|
4 |
| p38 delta MAPK |
102
|
11 |
| p38 gamma MAPK |
110
|
6 |
| PAK4 |
69
|
1 |
| PAK5 |
74
|
2 |
| PAK6 |
97
|
2 |
| PDK1 |
110
|
5 |
| PHK |
101
|
10 |
| PIM1 |
104
|
8 |
| PIM2 |
108
|
1 |
| PIM3 |
79
|
1 |
| PKA |
96
|
5 |
| PKB alpha |
104
|
2 |
| PKB beta |
98
|
0 |
| PKC alpha |
103
|
5 |
| PKC zeta |
94
|
1 |
| PKD1 |
103
|
9 |
| PLK1 |
96
|
3 |
| PRAK |
88
|
13 |
| PRK2 |
95
|
9 |
| ROCK 2 |
85
|
3 |
| RSK1 |
75
|
2 |
| RSK2 |
97
|
6 |
| S6K1 |
106
|
17 |
| SGK1 |
88
|
3 |
| SmMLCK |
84
|
26 |
| Src |
72
|
2 |
| SRPK1 |
95
|
0 |
| SYK |
100
|
2 |
| TBK1 |
64
|
4 |
| VEGFR1 |
50
|
1 |
| YES1 |
85
|
7 |
