Inhibitor | AG1296 (Tyrphostin)
Screening Results Tables
Screen Conc: 10.00µM
Kinase |
% Activity Remaining |
Standard Deviation |
AMPK |
80
|
1 |
Aurora B |
15
|
1 |
BRSK2 |
99
|
2 |
BTK |
80
|
10 |
CAMK1 |
104
|
3 |
CAMKK beta |
88
|
1 |
CDK2-Cyclin A |
91
|
8 |
CHK1 |
95
|
0 |
CHK2 |
93
|
9 |
CK1 delta |
54
|
2 |
CK2 |
80
|
2 |
CSK |
105
|
0 |
DYRK1A |
93
|
4 |
DYRK2 |
84
|
5 |
DYRK3 |
91
|
22 |
EF2K |
103
|
10 |
EPH-A2 |
98
|
14 |
EPH-B3 |
86
|
10 |
ERK1 |
101
|
17 |
ERK2 |
105
|
3 |
ERK8 |
86
|
12 |
FGF-R1 |
94
|
18 |
GSK3 beta |
113
|
4 |
HIPK2 |
98
|
0 |
IGF-1R |
102
|
7 |
IKK beta |
101
|
3 |
IKK epsilon |
85
|
2 |
IR |
70
|
7 |
IRR |
75
|
9 |
JNK1 |
101
|
11 |
JNK2 |
113
|
10 |
Lck |
82
|
1 |
MAPKAP-K2 |
107
|
11 |
MARK3 |
103
|
9 |
MELK |
64
|
6 |
MKK1 |
92
|
10 |
MNK1 |
83
|
11 |
MNK2 |
74
|
0 |
MSK1 |
102
|
1 |
MST2 |
79
|
6 |
MST4 |
105
|
10 |
NEK2a |
65
|
5 |
NEK6 |
116
|
27 |
p38 alpha MAPK |
91
|
5 |
p38 beta MAPK |
95
|
4 |
p38 delta MAPK |
102
|
11 |
p38 gamma MAPK |
110
|
6 |
PAK4 |
69
|
1 |
PAK5 |
74
|
2 |
PAK6 |
97
|
2 |
PDK1 |
110
|
5 |
PHK |
101
|
10 |
PIM1 |
104
|
8 |
PIM2 |
108
|
1 |
PIM3 |
79
|
1 |
PKA |
96
|
5 |
PKB alpha |
104
|
2 |
PKB beta |
98
|
0 |
PKC alpha |
103
|
5 |
PKC zeta |
94
|
1 |
PKD1 |
103
|
9 |
PLK1 |
96
|
3 |
PRAK |
88
|
13 |
PRK2 |
95
|
9 |
ROCK 2 |
85
|
3 |
RSK1 |
75
|
2 |
RSK2 |
97
|
6 |
S6K1 |
106
|
17 |
SGK1 |
88
|
3 |
SmMLCK |
84
|
26 |
Src |
72
|
2 |
SRPK1 |
95
|
0 |
SYK |
100
|
2 |
TBK1 |
64
|
4 |
VEGFR1 |
50
|
1 |
YES1 |
85
|
7 |