

Compound name | Brutto | MW | CAS | PubChem CID | Action | Reference | Reference |
---|---|---|---|---|---|---|---|
Zearalenone | C18H22O5 | 318.40 | 17924-92-4 | 5281576 | Estrogen receptor (ER) | Powell-Jones W. (1981) Mol. Pharmacol. 20 35-42 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
AMPK | 94 | 13 |
Aurora B | 37 | 1 |
BRSK2 | 54 | 1 |
BTK | 107 | 12 |
CAMK1 | 101 | 1 |
CAMKK beta | 90 | 5 |
CDK2-Cyclin A | 82 | 10 |
CHK1 | 92 | 5 |
CHK2 | 93 | 3 |
CK1 delta | 99 | 4 |
CK2 | 97 | 15 |
CSK | 80 | 6 |
DYRK1A | 72 | 22 |
DYRK2 | 90 | 3 |
DYRK3 | 100 | 3 |
EF2K | 101 | 3 |
EPH-A2 | 69 | 4 |
EPH-B3 | 85 | 11 |
ERK1 | 113 | 10 |
ERK2 | 98 | 3 |
ERK8 | 77 | 13 |
FGF-R1 | 90 | 16 |
GSK3 beta | 47 | 3 |
HIPK2 | 100 | 0 |
IGF-1R | 93 | 13 |
IKK beta | 101 | 12 |
IKK epsilon | 95 | 5 |
IR | 107 | 13 |
IRR | 75 | 18 |
JNK1 | 88 | 5 |
JNK2 | 46 | 2 |
Lck | 69 | 2 |
MAPKAP-K2 | 101 | 7 |
MARK3 | 102 | 4 |
MELK | 97 | 6 |
MKK1 | 66 | 4 |
MNK1 | 89 | 15 |
MNK2 | 64 | 4 |
MSK1 | 69 | 29 |
MST2 | 119 | 2 |
MST4 | 103 | 25 |
NEK2a | 93 | 9 |
NEK6 | 91 | 1 |
p38 alpha MAPK | 93 | 8 |
p38 beta MAPK | 108 | 11 |
p38 delta MAPK | 84 | 1 |
p38 gamma MAPK | 97 | 4 |
PAK4 | 95 | 6 |
PAK5 | 93 | 11 |
PAK6 | 99 | 10 |
PDK1 | 91 | 5 |
PHK | 102 | 6 |
PIM1 | 51 | 6 |
PIM2 | 86 | 2 |
PIM3 | 49 | 3 |
PKA | 97 | 7 |
PKB alpha | 111 | 23 |
PKB beta | 97 | 4 |
PKC alpha | 54 | 4 |
PKC zeta | 98 | 10 |
PKD1 | 86 | 1 |
PLK1 | 76 | 5 |
PRAK | 97 | 5 |
PRK2 | 70 | 5 |
ROCK 2 | 82 | 5 |
RSK1 | 89 | 1 |
RSK2 | 80 | 13 |
S6K1 | 106 | 18 |
SGK1 | 93 | 6 |
SmMLCK | 104 | 11 |
Src | 89 | 13 |
SRPK1 | 95 | 19 |
SYK | 93 | 12 |
TBK1 | 82 | 5 |
VEGFR1 | 95 | 8 |
YES1 | 79 | 8 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
AMPK | 60 | 9 |
Aurora B | 23 | 4 |
BRSK2 | 17 | 1 |
BTK | 69 | 3 |
CAMK1 | 75 | 11 |
CAMKK beta | 52 | 3 |
CDK2-Cyclin A | 32 | 1 |
CHK1 | 81 | 5 |
CHK2 | 73 | 7 |
CK1 delta | 83 | 3 |
CK2 | 96 | 5 |
CSK | 64 | 5 |
DYRK1A | 32 | 8 |
DYRK2 | 62 | 1 |
DYRK3 | 62 | 4 |
EF2K | 85 | 15 |
EPH-A2 | 26 | 1 |
EPH-B3 | 85 | 3 |
ERK1 | 107 | 7 |
ERK2 | 96 | 17 |
ERK8 | 26 | 5 |
FGF-R1 | 51 | 4 |
GSK3 beta | 11 | 1 |
HIPK2 | 63 | 6 |
IGF-1R | 64 | 6 |
IKK beta | 78 | 15 |
IKK epsilon | 82 | 5 |
IR | 102 | 3 |
IRR | 41 | 1 |
JNK1 | 80 | 2 |
JNK2 | 65 | 9 |
Lck | 26 | 0 |
MAPKAP-K2 | 92 | 1 |
MARK3 | 99 | 4 |
MELK | 66 | 0 |
MKK1 | 55 | 0 |
MNK1 | 46 | 5 |
MNK2 | 23 | 1 |
MSK1 | 36 | 2 |
MST2 | 113 | 12 |
MST4 | 66 | 9 |
NEK2a | 96 | 11 |
NEK6 | 91 | 3 |
p38 alpha MAPK | 85 | 2 |
p38 beta MAPK | 101 | 2 |
p38 delta MAPK | 87 | 2 |
p38 gamma MAPK | 93 | 10 |
PAK4 | 90 | 2 |
PAK5 | 80 | 6 |
PAK6 | 94 | 10 |
PDK1 | 80 | 2 |
PHK | 86 | 5 |
PIM1 | 11 | 0 |
PIM2 | 45 | 11 |
PIM3 | 18 | 2 |
PKA | 91 | 5 |
PKB alpha | 95 | 9 |
PKB beta | 89 | 4 |
PKC alpha | 69 | 2 |
PKC zeta | 86 | 9 |
PKD1 | 64 | 17 |
PLK1 | 63 | 5 |
PRAK | 79 | 4 |
PRK2 | 33 | 5 |
ROCK 2 | 81 | 4 |
RSK1 | 41 | 1 |
RSK2 | 52 | 3 |
S6K1 | 61 | 9 |
SGK1 | 93 | 13 |
SmMLCK | 59 | 1 |
Src | 34 | 5 |
SRPK1 | 89 | 17 |
SYK | 84 | 6 |
TBK1 | 80 | 4 |
VEGFR1 | 69 | 10 |
YES1 | 35 | 1 |