Inhibitor | Uo126  

Screen Conc: 5.00µM

Kinase	% Activity Remaining	Standard Deviation
AMPK	58	6
Aurora B	71	3
Aurora C	87	9
BRSK2	58	2
CAMK1	81	1
CAMKK alpha	76	1
CAMKK beta	91	1
CDK2-Cyclin A	89	0
CHK1	98	3
CHK2	85	8
CK1 delta	102	2
CK2	85	1
CSK	77	6
DYRK1A	92	2
DYRK2	71	1
DYRK3	54	5
EF2K	75	5
ERK1	79	2
ERK2	81	6
ERK8	71	4
GSK3 beta	62	5
HIPK2	106	5
HIPK3	87	2
IKK beta	74	1
JNK1	77	1
JNK2	84	2
JNK3	78	2
Lck	63	6
MAPKAP-K2	98	5
MAPKAP-K3	79	2
MARK3	82	7
MELK	75	4
MKK1	66	2
MNK1	56	7
MNK2	74	1
MSK1	76	5
MST2	70	8
NEK2a	90	6
NEK6	90	3
NEK7	77	9
p38 alpha MAPK	48	1
p38 beta MAPK	64	1
p38 delta MAPK	96	4
p38 gamma MAPK	87	4
PAK4	64	3
PAK5	66	1
PAK6	63	3
PDK1	91	6
PHK	75	4
PIM1	86	7
PIM2	65	9
PIM3	74	2
PKA	52	0
PKB alpha	94	6
PKB beta	81	6
PKC alpha	83	8
PKC zeta	65	4
PKD1	73	0
PLK1	68	8
PRAK	67	0
PRK2	97	4
ROCK 2	64	5
RSK1	94	9
RSK2	83	0
S6K1	82	1
SGK1	70	3
SmMLCK	81	6
Src	83	7
SRPK1	91	0

Screen Conc: 10.00µM

Kinase	% Activity Remaining	Standard Deviation
AMPK	76	12
Aurora B	86	3
Aurora C	88	11
BRSK2	87	12
CAMK1	69	4
CAMKK alpha	99	11
CAMKK beta	92	6
CDK2-Cyclin A	86	1
CHK1	83	3
CHK2	98	3
CK1 delta	90	10
CK2	99	4
CSK	88	12
DYRK1A	69	4
DYRK2	84	3
DYRK3	77	4
EF2K	116	5
ERK1	72	5
ERK2	68	3
ERK8	67	3
GSK3 beta	82	5
HIPK2	97	3
HIPK3	87	7
IKK beta	118	7
JNK1	90	2
JNK2	73	4
JNK3	98	4
Lck	84	4
MAPKAP-K2	95	2
MAPKAP-K3	97	15
MARK3	95	5
MELK	83	11
MKK1	24	1
MNK1	78	2
MNK2	85	8
MSK1	85	7
MST2	96	5
NEK2a	89	7
NEK6	90	3
NEK7	97	6
p38 alpha MAPK	77	6
p38 beta MAPK	91	9
p38 delta MAPK	93	7
p38 gamma MAPK	90	1
PAK4	94	4
PAK5	86	2
PAK6	85	11
PDK1	77	3
PHK	94	7
PIM1	87	0
PIM2	101	3
PIM3	63	8
PKA	93	5
PKB alpha	76	8
PKB beta	98	1
PKC alpha	95	5
PKC zeta	78	2
PKD1	77	6
PLK1	92	7
PRAK	92	2
PRK2	85	9
ROCK 2	81	6
RSK1	83	6
RSK2	81	1
S6K1	93	5
SGK1	72	6
SmMLCK	95	5
Src	84	6
SRPK1	102	6