| Compound name | Brutto | MW | CAS | PubChem CID | Action | Reference | Reference |
|---|---|---|---|---|---|---|---|
| ARA014418 | C12H12N4O4S | 308.30 | 487021-52-3 | 448014 | GSK3 | Noble W. (2005) Proc. Natl. Acad. Sci. USA 102 6990 | Bhat R. (2003) J. Biol. Chem. 278 45937 |
| Kinase Sort ascending | % Activity Remaining | Standard Deviation |
|---|---|---|
| YES1 | 111 | 7 |
| TBK1 | 78 | 2 |
| SYK | 107 | 10 |
| SRPK1 | 74 | 5 |
| Src | 81 | 1 |
| SmMLCK | 90 | 2 |
| SGK1 | 87 | 3 |
| S6K1 | 75 | 2 |
| RSK2 | 84 | 1 |
| RSK1 | 79 | 4 |
| ROCK 2 | 83 | 2 |
| PRK2 | 85 | 2 |
| PRAK | 67 | 5 |
| PLK1 | 78 | 0 |
| PKD1 | 92 | 4 |
| PKC zeta | 70 | 1 |
| PKC alpha | 80 | 3 |
| PKB beta | 85 | 2 |
| PKB alpha | 95 | 2 |
| PKA | 68 | 4 |
| PIM3 | 69 | 0 |
| PIM2 | 92 | 5 |
| PIM1 | 83 | 3 |
| PHK | 90 | 4 |
| PDK1 | 74 | 1 |
| PAK6 | 74 | 2 |
| PAK5 | 76 | 0 |
| PAK4 | 66 | 2 |
| p38 gamma MAPK | 89 | 1 |
| p38 delta MAPK | 80 | 2 |
| p38 beta MAPK | 102 | 8 |
| p38 alpha MAPK | 109 | 8 |
| NEK7 | 96 | 2 |
| NEK6 | 91 | 1 |
| NEK2a | 81 | 2 |
| MST4 | 99 | 14 |
| MST2 | 80 | 7 |
| MSK1 | 80 | 4 |
| MNK2 | 94 | 5 |
| MNK1 | 80 | 2 |
| MKK1 | 77 | 9 |
| MELK | 75 | 4 |
| MARK3 | 75 | 4 |
| MAPKAP-K3 | 81 | 4 |
| MAPKAP-K2 | 103 | 2 |
| Lck | 80 | 1 |
| JNK3 | 91 | 0 |
| JNK2 | 72 | 5 |
| JNK1 | 80 | 1 |
| IRR | 45 | 1 |
| IKK epsilon | 83 | 3 |
| IKK beta | 75 | 3 |
| HIPK3 | 88 | 1 |
| HIPK2 | 53 | 3 |
| GSK3 beta |
3
|
0 |
| FGF-R1 | 91 | 8 |
| ERK8 | 37 | 3 |
| ERK2 | 94 | 7 |
| ERK1 | 101 | 1 |
| EPH-A2 | 101 | 5 |
| EF2K | 98 | 5 |
| DYRK3 | 71 | 1 |
| DYRK2 | 81 | 7 |
| DYRK1A | 50 | 6 |
| CSK | 82 | 2 |
| CK2 | 79 | 1 |
| CK1 delta | 89 | 6 |
| CHK2 | 93 | 2 |
| CHK1 | 83 | 2 |
| CDK2-Cyclin A | 23 | 2 |
| CAMKK beta | 73 | 9 |
| CAMKK alpha | 79 | 5 |
| CAMK1 | 76 | 3 |
| BRSK2 | 76 | 4 |
| Aurora C | 84 | 3 |
| Aurora B | 71 | 3 |
| AMPK | 72 | 1 |