Inhibitor | ARA014418  

Compound name Brutto MW CAS PubChem CID Action Reference Reference
ARA014418   C12H12N4O4S 308.30 487021-52-3 448014 GSK3 Noble W. (2005) Proc. Natl. Acad. Sci. USA 102 6990 Bhat R. (2003) J. Biol. Chem. 278 45937

Screening Results Chart

Screening Results Tables

Screen Conc: 10.00µM
Kinase % Activity Remaining Sort ascending Standard Deviation
YES1 111 7
p38 alpha MAPK 109 8
SYK 107 10
MAPKAP-K2 103 2
p38 beta MAPK 102 8
ERK1 101 1
EPH-A2 101 5
MST4 99 14
EF2K 98 5
NEK7 96 2
PKB alpha 95 2
MNK2 94 5
ERK2 94 7
CHK2 93 2
PKD1 92 4
PIM2 92 5
NEK6 91 1
JNK3 91 0
FGF-R1 91 8
SmMLCK 90 2
PHK 90 4
CK1 delta 89 6
p38 gamma MAPK 89 1
HIPK3 88 1
SGK1 87 3
PKB beta 85 2
PRK2 85 2
RSK2 84 1
Aurora C 84 3
IKK epsilon 83 3
ROCK 2 83 2
CHK1 83 2
PIM1 83 3
CSK 82 2
MAPKAP-K3 81 4
DYRK2 81 7
Src 81 1
NEK2a 81 2
MST2 80 7
JNK1 80 1
Lck 80 1
PKC alpha 80 3
MSK1 80 4
p38 delta MAPK 80 2
MNK1 80 2
RSK1 79 4
CAMKK alpha 79 5
CK2 79 1
TBK1 78 2
PLK1 78 0
MKK1 77 9
BRSK2 76 4
CAMK1 76 3
PAK5 76 0
MARK3 75 4
MELK 75 4
S6K1 75 2
IKK beta 75 3
SRPK1 74 5
PDK1 74 1
PAK6 74 2
CAMKK beta 73 9
AMPK 72 1
JNK2 72 5
DYRK3 71 1
Aurora B 71 3
PKC zeta 70 1
PIM3 69 0
PKA 68 4
PRAK 67 5
PAK4 66 2
HIPK2 53 3
DYRK1A 50 6
IRR 45 1
ERK8 37 3
CDK2-Cyclin A 23 2
GSK3 beta
3
0