Inhibitor | SRC Inhibitor 1  

Screen Conc: 1.00µM

Kinase	% Activity Remaining	Standard Deviation
AMPK	87	11
Aurora B	35	1
Aurora C	71	1
BRSK2	92	11
CAMK1	86	9
CAMKK beta	94	1
CDK2-Cyclin A	97	13
CHK1	86	8
CHK2	11	1
CK1 delta	101	4
CK2	92	2
CSK	12	3
DYRK1A	102	5
DYRK2	100	1
DYRK3	81	2
EF2K	89	1
EPH-A2	85	9
ERK1	103	8
ERK2	74	9
ERK8	82	7
FGF-R1	40	7
GSK3 beta	89	1
HIPK2	88	1
HIPK3	83	13
IKK beta	97	7
IKK epsilon	81	12
IRR	108	5
JNK1	84	3
JNK2	94	9
JNK3	81	7
Lck	11	1
MAPKAP-K2	81	3
MAPKAP-K3	88	4
MARK3	92	10
MELK	76	7
MKK1	50	8
MNK1	81	1
MNK2	61	7
MSK1	81	3
MST2	87	4
MST4	72	7
NEK2a	83	1
NEK6	97	14
NEK7	81	7
p38 alpha MAPK	83	4
p38 beta MAPK	90	8
p38 delta MAPK	86	2
p38 gamma MAPK	104	2
PAK4	95	1
PAK5	81	2
PAK6	102	12
PDK1	88	3
PHK	80	5
PIM1	82	0
PIM2	85	6
PIM3	81	8
PKA	95	9
PKB alpha	80	12
PKB beta	86	7
PKC alpha	95	2
PKC zeta	95	4
PKD1	81	4
PLK1	95	13
PRAK	94	5
PRK2	81	4
ROCK 2	84	10
RSK1	73	5
RSK2	80	2
S6K1	92	4
SGK1	106	4
SmMLCK	85	14
Src	12	1
SRPK1	69	0
SYK	91	5
TBK1	93	15
YES1	5	1

Screen Conc: 10.00µM

Kinase	% Activity Remaining	Standard Deviation
AMPK	74	4
Aurora B	23	2
Aurora C	42	5
BRSK2	88	6
CAMK1	61	10
CAMKK beta	93	0
CDK2-Cyclin A	103	14
CHK1	84	4
CHK2	2	1
CK1 delta	81	5
CK2	105	3
CSK	2	0
DYRK1A	95	0
DYRK2	94	14
DYRK3	68	11
EF2K	111	7
EPH-A2	103	4
ERK1	103	7
ERK2	68	7
ERK8	80	1
FGF-R1	20	5
GSK3 beta	74	14
HIPK2	79	8
HIPK3	84	5
IKK beta	98	1
IKK epsilon	81	9
IRR	101	10
JNK1	75	0
JNK2	77	7
JNK3	74	13
Lck	4	0
MAPKAP-K2	81	5
MAPKAP-K3	100	6
MARK3	102	3
MELK	74	6
MKK1	25	3
MNK1	61	2
MNK2	50	1
MSK1	75	9
MST2	72	10
MST4	70	11
NEK2a	70	7
NEK6	96	4
NEK7	87	9
p38 alpha MAPK	82	2
p38 beta MAPK	67	7
p38 delta MAPK	70	4
p38 gamma MAPK	96	1
PAK4	52	2
PAK5	65	5
PAK6	82	6
PDK1	89	7
PHK	70	3
PIM1	86	11
PIM2	95	6
PIM3	69	7
PKA	94	10
PKB alpha	91	6
PKB beta	88	14
PKC alpha	87	9
PKC zeta	89	2
PKD1	91	6
PLK1	87	1
PRAK	89	6
PRK2	75	10
ROCK 2	71	15
RSK1	41	3
RSK2	81	7
S6K1	77	10
SGK1	94	4
SmMLCK	49	0
Src	2	0
SRPK1	66	11
SYK	86	4
TBK1	75	8
YES1	1	0