

Compound name | Brutto | MW | CAS | PubChem CID | Action | Reference | Reference |
---|---|---|---|---|---|---|---|
ARA014418 | C12H12N4O4S | 308.30 | 487021-52-3 | 448014 | GSK3 | Noble W. (2005) Proc. Natl. Acad. Sci. USA 102 6990 | Bhat R. (2003) J. Biol. Chem. 278 45937 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
AMPK | 72 | 1 |
Aurora B | 71 | 3 |
Aurora C | 84 | 3 |
BRSK2 | 76 | 4 |
CAMK1 | 76 | 3 |
CAMKK alpha | 79 | 5 |
CAMKK beta | 73 | 9 |
CDK2-Cyclin A | 23 | 2 |
CHK1 | 83 | 2 |
CHK2 | 93 | 2 |
CK1 delta | 89 | 6 |
CK2 | 79 | 1 |
CSK | 82 | 2 |
DYRK1A | 50 | 6 |
DYRK2 | 81 | 7 |
DYRK3 | 71 | 1 |
EF2K | 98 | 5 |
EPH-A2 | 101 | 5 |
ERK1 | 101 | 1 |
ERK2 | 94 | 7 |
ERK8 | 37 | 3 |
FGF-R1 | 91 | 8 |
GSK3 beta |
3
|
0 |
HIPK2 | 53 | 3 |
HIPK3 | 88 | 1 |
IKK beta | 75 | 3 |
IKK epsilon | 83 | 3 |
IRR | 45 | 1 |
JNK1 | 80 | 1 |
JNK2 | 72 | 5 |
JNK3 | 91 | 0 |
Lck | 80 | 1 |
MAPKAP-K2 | 103 | 2 |
MAPKAP-K3 | 81 | 4 |
MARK3 | 75 | 4 |
MELK | 75 | 4 |
MKK1 | 77 | 9 |
MNK1 | 80 | 2 |
MNK2 | 94 | 5 |
MSK1 | 80 | 4 |
MST2 | 80 | 7 |
MST4 | 99 | 14 |
NEK2a | 81 | 2 |
NEK6 | 91 | 1 |
NEK7 | 96 | 2 |
p38 alpha MAPK | 109 | 8 |
p38 beta MAPK | 102 | 8 |
p38 delta MAPK | 80 | 2 |
p38 gamma MAPK | 89 | 1 |
PAK4 | 66 | 2 |
PAK5 | 76 | 0 |
PAK6 | 74 | 2 |
PDK1 | 74 | 1 |
PHK | 90 | 4 |
PIM1 | 83 | 3 |
PIM2 | 92 | 5 |
PIM3 | 69 | 0 |
PKA | 68 | 4 |
PKB alpha | 95 | 2 |
PKB beta | 85 | 2 |
PKC alpha | 80 | 3 |
PKC zeta | 70 | 1 |
PKD1 | 92 | 4 |
PLK1 | 78 | 0 |
PRAK | 67 | 5 |
PRK2 | 85 | 2 |
ROCK 2 | 83 | 2 |
RSK1 | 79 | 4 |
RSK2 | 84 | 1 |
S6K1 | 75 | 2 |
SGK1 | 87 | 3 |
SmMLCK | 90 | 2 |
Src | 81 | 1 |
SRPK1 | 74 | 5 |
SYK | 107 | 10 |
TBK1 | 78 | 2 |
YES1 | 111 | 7 |