| Compound name | Brutto | MW | CAS | PubChem CID | Action | Reference | Reference |
|---|---|---|---|---|---|---|---|
| SB-216763 | C19H12Cl2N2O2 | 371.22 | 280744-09-4 | 176158 | GSK3 | Coghlan (2000) Chem.Biol. 7 793 | Liang (2006) J.Biol.Chem. 282 3904 |
| Kinase | % Activity Remaining | Standard Deviation |
|---|---|---|
| AMPK | 69 | 0 |
| Aurora B | 83 | 4 |
| Aurora C | 52 | 1 |
| BRSK2 | 82 | 4 |
| CAMK1 | 86 | 3 |
| CAMKK alpha | 85 | 3 |
| CAMKK beta | 43 | 12 |
| CDK2-Cyclin A | 57 | 9 |
| CHK1 | 92 | 8 |
| CHK2 | 83 | 7 |
| CK1 delta | 73 | 5 |
| CK2 | 91 | 6 |
| CSK | 91 | 1 |
| DYRK1A |
4
|
0 |
| DYRK2 | 104 | 3 |
| DYRK3 | 59 | 1 |
| EF2K | 96 | 4 |
| EPH-A2 | 84 | 4 |
| ERK1 | 88 | 13 |
| ERK2 | 76 | 5 |
| ERK8 |
0
|
0 |
| FGF-R1 | 94 | 11 |
| GSK3 beta |
-3
|
1 |
| HIPK2 | 14 | 7 |
| HIPK3 | 41 | 4 |
| IKK beta | 91 | 0 |
| IKK epsilon | 55 | 4 |
| IRR | 31 | 3 |
| JNK1 | 95 | 5 |
| JNK2 | 81 | 1 |
| JNK3 | 77 | 6 |
| Lck | 88 | 11 |
| MAPKAP-K2 | 71 | 10 |
| MAPKAP-K3 | 117 | 3 |
| MARK3 | 68 | 10 |
| MELK | 59 | 3 |
| MKK1 | 61 | 4 |
| MNK1 | 79 | 1 |
| MNK2 | 81 | 4 |
| MSK1 | 73 | 4 |
| MST2 | 31 | 7 |
| MST4 | 49 | 7 |
| NEK2a | 60 | 7 |
| NEK6 | 42 | 8 |
| NEK7 | 79 | 1 |
| p38 alpha MAPK | 72 | 3 |
| p38 beta MAPK | 61 | 12 |
| p38 delta MAPK | 67 | 11 |
| p38 gamma MAPK | 95 | 5 |
| PAK4 | 63 | 4 |
| PAK5 | 58 | 1 |
| PAK6 | 86 | 14 |
| PDK1 | 95 | 2 |
| PHK | 73 | 5 |
| PIM1 | 62 | 11 |
| PIM2 | 44 | 3 |
| PIM3 | 31 | 5 |
| PKA | 92 | 5 |
| PKB alpha | 84 | 7 |
| PKB beta | 81 | 14 |
| PKC alpha | 58 | 7 |
| PKC zeta | 75 | 6 |
| PKD1 | 86 | 12 |
| PLK1 | 51 | 2 |
| PRAK | 84 | 3 |
| PRK2 | 69 | 1 |
| ROCK 2 | 71 | 6 |
| RSK1 | 33 | 0 |
| RSK2 | 40 | 2 |
| S6K1 | 96 | 10 |
| SGK1 | 84 | 2 |
| SmMLCK | 40 | 6 |
| Src | 85 | 6 |
| SRPK1 | 12 | 2 |
| SYK | 89 | 13 |
| TBK1 | 82 | 8 |
| YES1 | 43 | 11 |