| Compound name | Brutto | MW | CAS | PubChem CID | Action | Reference | Reference |
|---|---|---|---|---|---|---|---|
| SB-203580 | C21H16N3OSF | 377.40 | 152121-47-6 | 176155 | p38 MAPK | Powell D.J. (2003) Mol. Cell Biol. 23 7794 | Davies S.P. (2000) Biochem. J. 351 95 |
| Kinase | % Activity Remaining | Standard Deviation |
|---|---|---|
| AMPK | 80 | 0 |
| Aurora B | 85 | 1 |
| Aurora C | 92 | 0 |
| BRSK2 | 85 | 11 |
| CAMK1 | 86 | 5 |
| CAMKK alpha | 105 | 13 |
| CAMKK beta | 98 | 4 |
| CDK2-Cyclin A | 103 | 2 |
| CHK1 | 66 | 6 |
| CHK2 | 91 | 4 |
| CK1 delta |
8
|
0 |
| CK2 | 97 | 2 |
| CSK | 68 | 0 |
| DYRK1A | 84 | 0 |
| DYRK2 | 96 | 1 |
| DYRK3 | 112 | 0 |
| EF2K | 97 | 0 |
| ERK1 | 88 | 0 |
| ERK2 | 83 | 7 |
| ERK8 | 93 | 8 |
| GSK3 beta | 34 | 2 |
| HIPK2 | 85 | 6 |
| HIPK3 | 96 | 1 |
| IKK beta | 94 | 2 |
| JNK1 | 95 | 0 |
| JNK2 | 60 | 3 |
| JNK3 | 72 | 6 |
| Lck | 56 | 3 |
| MAPKAP-K2 | 84 | 2 |
| MAPKAP-K3 | 119 | 5 |
| MARK3 | 98 | 1 |
| MELK | 82 | 8 |
| MKK1 | 85 | 7 |
| MNK1 | 108 | 10 |
| MNK2 | 106 | 1 |
| MSK1 | 90 | 10 |
| MST2 | 85 | 5 |
| NEK2a | 80 | 5 |
| NEK6 | 98 | 0 |
| NEK7 | 95 | 6 |
| p38 alpha MAPK |
9
|
0 |
| p38 beta MAPK | 12 | 0 |
| p38 delta MAPK | 106 | 3 |
| p38 gamma MAPK | 104 | 0 |
| PAK4 | 86 | 12 |
| PAK5 | 88 | 0 |
| PAK6 | 82 | 10 |
| PDK1 | 81 | 2 |
| PHK | 104 | 2 |
| PIM1 | 82 | 4 |
| PIM2 | 97 | 2 |
| PIM3 | 81 | 4 |
| PKA | 89 | 3 |
| PKB alpha | 89 | 11 |
| PKB beta | 89 | 0 |
| PKC alpha | 86 | 6 |
| PKC zeta | 88 | 0 |
| PKD1 | 77 | 7 |
| PLK1 | 108 | 0 |
| PRAK | 95 | 5 |
| PRK2 | 95 | 7 |
| ROCK 2 | 72 | 13 |
| RSK1 | 52 | 7 |
| RSK2 | 93 | 6 |
| S6K1 | 79 | 5 |
| SGK1 | 90 | 0 |
| SmMLCK | 85 | 1 |
| Src | 72 | 3 |
| SRPK1 | 90 | 2 |
| Kinase | % Activity Remaining | Standard Deviation |
|---|---|---|
| AMPK | 20 | 3 |
| Aurora B | 63 | 4 |
| Aurora C | 68 | 4 |
| BRSK2 | 58 | 4 |
| CAMK1 | 79 | 4 |
| CAMKK alpha | 72 | 4 |
| CAMKK beta | 78 | 0 |
| CDK2-Cyclin A | 81 | 2 |
| CHK1 | 67 | 3 |
| CHK2 | 107 | 5 |
| CK1 delta |
0
|
0 |
| CK2 | 89 | 3 |
| CSK | 37 | 2 |
| DYRK1A | 91 | 1 |
| DYRK2 | 88 | 8 |
| DYRK3 | 75 | 5 |
| EF2K | 101 | 1 |
| ERK1 | 82 | 1 |
| ERK2 | 85 | 1 |
| ERK8 | 80 | 8 |
| GSK3 beta | 12 | 2 |
| HIPK2 | 90 | 1 |
| HIPK3 | 99 | 7 |
| IKK beta | 87 | 4 |
| JNK1 | 77 | 5 |
| JNK2 | 16 | 0 |
| JNK3 | 29 | 0 |
| Lck | 24 | 4 |
| MAPKAP-K2 | 111 | 4 |
| MAPKAP-K3 | 88 | 8 |
| MARK3 | 66 | 3 |
| MELK | 53 | 0 |
| MKK1 | 85 | 4 |
| MNK1 | 63 | 0 |
| MNK2 | 92 | 1 |
| MSK1 | 78 | 5 |
| MST2 | 75 | 6 |
| NEK2a | 83 | 2 |
| NEK6 | 85 | 1 |
| NEK7 | 108 | 3 |
| p38 alpha MAPK |
2
|
0 |
| p38 beta MAPK |
3
|
1 |
| p38 delta MAPK | 83 | 3 |
| p38 gamma MAPK | 83 | 4 |
| PAK4 | 80 | 6 |
| PAK5 | 88 | 4 |
| PAK6 | 82 | 1 |
| PDK1 | 67 | 2 |
| PHK | 62 | 2 |
| PIM1 | 81 | 0 |
| PIM2 | 106 | 8 |
| PIM3 | 54 | 3 |
| PKA | 53 | 4 |
| PKB alpha | 77 | 7 |
| PKB beta | 80 | 4 |
| PKC alpha | 42 | 0 |
| PKC zeta | 65 | 8 |
| PKD1 | 60 | 3 |
| PLK1 | 83 | 6 |
| PRAK | 64 | 6 |
| PRK2 | 67 | 1 |
| ROCK 2 | 65 | 1 |
| RSK1 | 34 | 6 |
| RSK2 | 60 | 7 |
| S6K1 | 78 | 4 |
| SGK1 | 66 | 1 |
| SmMLCK | 73 | 3 |
| Src | 47 | 5 |
| SRPK1 | 81 | 7 |