

Compound name | Brutto | MW | CAS | PubChem CID | Action | Reference | Reference |
---|---|---|---|---|---|---|---|
SB-203580 | C21H16N3OSF | 377.40 | 152121-47-6 | 176155 | p38 MAPK | Powell D.J. (2003) Mol. Cell Biol. 23 7794 | Davies S.P. (2000) Biochem. J. 351 95 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
AMPK | 80 | 0 |
Aurora B | 85 | 1 |
Aurora C | 92 | 0 |
BRSK2 | 85 | 11 |
CAMK1 | 86 | 5 |
CAMKK alpha | 105 | 13 |
CAMKK beta | 98 | 4 |
CDK2-Cyclin A | 103 | 2 |
CHK1 | 66 | 6 |
CHK2 | 91 | 4 |
CK1 delta |
8
|
0 |
CK2 | 97 | 2 |
CSK | 68 | 0 |
DYRK1A | 84 | 0 |
DYRK2 | 96 | 1 |
DYRK3 | 112 | 0 |
EF2K | 97 | 0 |
ERK1 | 88 | 0 |
ERK2 | 83 | 7 |
ERK8 | 93 | 8 |
GSK3 beta | 34 | 2 |
HIPK2 | 85 | 6 |
HIPK3 | 96 | 1 |
IKK beta | 94 | 2 |
JNK1 | 95 | 0 |
JNK2 | 60 | 3 |
JNK3 | 72 | 6 |
Lck | 56 | 3 |
MAPKAP-K2 | 84 | 2 |
MAPKAP-K3 | 119 | 5 |
MARK3 | 98 | 1 |
MELK | 82 | 8 |
MKK1 | 85 | 7 |
MNK1 | 108 | 10 |
MNK2 | 106 | 1 |
MSK1 | 90 | 10 |
MST2 | 85 | 5 |
NEK2a | 80 | 5 |
NEK6 | 98 | 0 |
NEK7 | 95 | 6 |
p38 alpha MAPK |
9
|
0 |
p38 beta MAPK | 12 | 0 |
p38 delta MAPK | 106 | 3 |
p38 gamma MAPK | 104 | 0 |
PAK4 | 86 | 12 |
PAK5 | 88 | 0 |
PAK6 | 82 | 10 |
PDK1 | 81 | 2 |
PHK | 104 | 2 |
PIM1 | 82 | 4 |
PIM2 | 97 | 2 |
PIM3 | 81 | 4 |
PKA | 89 | 3 |
PKB alpha | 89 | 11 |
PKB beta | 89 | 0 |
PKC alpha | 86 | 6 |
PKC zeta | 88 | 0 |
PKD1 | 77 | 7 |
PLK1 | 108 | 0 |
PRAK | 95 | 5 |
PRK2 | 95 | 7 |
ROCK 2 | 72 | 13 |
RSK1 | 52 | 7 |
RSK2 | 93 | 6 |
S6K1 | 79 | 5 |
SGK1 | 90 | 0 |
SmMLCK | 85 | 1 |
Src | 72 | 3 |
SRPK1 | 90 | 2 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
AMPK | 20 | 3 |
Aurora B | 63 | 4 |
Aurora C | 68 | 4 |
BRSK2 | 58 | 4 |
CAMK1 | 79 | 4 |
CAMKK alpha | 72 | 4 |
CAMKK beta | 78 | 0 |
CDK2-Cyclin A | 81 | 2 |
CHK1 | 67 | 3 |
CHK2 | 107 | 5 |
CK1 delta |
0
|
0 |
CK2 | 89 | 3 |
CSK | 37 | 2 |
DYRK1A | 91 | 1 |
DYRK2 | 88 | 8 |
DYRK3 | 75 | 5 |
EF2K | 101 | 1 |
ERK1 | 82 | 1 |
ERK2 | 85 | 1 |
ERK8 | 80 | 8 |
GSK3 beta | 12 | 2 |
HIPK2 | 90 | 1 |
HIPK3 | 99 | 7 |
IKK beta | 87 | 4 |
JNK1 | 77 | 5 |
JNK2 | 16 | 0 |
JNK3 | 29 | 0 |
Lck | 24 | 4 |
MAPKAP-K2 | 111 | 4 |
MAPKAP-K3 | 88 | 8 |
MARK3 | 66 | 3 |
MELK | 53 | 0 |
MKK1 | 85 | 4 |
MNK1 | 63 | 0 |
MNK2 | 92 | 1 |
MSK1 | 78 | 5 |
MST2 | 75 | 6 |
NEK2a | 83 | 2 |
NEK6 | 85 | 1 |
NEK7 | 108 | 3 |
p38 alpha MAPK |
2
|
0 |
p38 beta MAPK |
3
|
1 |
p38 delta MAPK | 83 | 3 |
p38 gamma MAPK | 83 | 4 |
PAK4 | 80 | 6 |
PAK5 | 88 | 4 |
PAK6 | 82 | 1 |
PDK1 | 67 | 2 |
PHK | 62 | 2 |
PIM1 | 81 | 0 |
PIM2 | 106 | 8 |
PIM3 | 54 | 3 |
PKA | 53 | 4 |
PKB alpha | 77 | 7 |
PKB beta | 80 | 4 |
PKC alpha | 42 | 0 |
PKC zeta | 65 | 8 |
PKD1 | 60 | 3 |
PLK1 | 83 | 6 |
PRAK | 64 | 6 |
PRK2 | 67 | 1 |
ROCK 2 | 65 | 1 |
RSK1 | 34 | 6 |
RSK2 | 60 | 7 |
S6K1 | 78 | 4 |
SGK1 | 66 | 1 |
SmMLCK | 73 | 3 |
Src | 47 | 5 |
SRPK1 | 81 | 7 |