Compound name | Brutto | MW | CAS | PubChem CID | Action | Reference | Reference |
---|---|---|---|---|---|---|---|
Resveratrol | C14H12O3 | 228.20 | 501-36-0 | 445154 | cyclo-oxygenase 1 | Lin H.Y. (2002) J. Urol. 168 748 | Klabunde T. (2000) Nat. Struct. Biol. 7 312 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
AMPK | 103 | 9 |
Aurora B | 97 | 8 |
Aurora C | 75 | 2 |
BRSK2 | 54 | 5 |
CAMK1 | 75 | 9 |
CAMKK alpha | 98 | 1 |
CAMKK beta | 107 | 2 |
CDK2-Cyclin A | 103 | 9 |
CHK1 | 95 | 5 |
CHK2 | 84 | 6 |
CK1 delta | 84 | 6 |
CK2 | 101 | 1 |
CSK | 102 | 9 |
DYRK1A | 94 | 6 |
DYRK2 | 40 | 5 |
DYRK3 | 38 | 2 |
EF2K | 95 | 8 |
ERK1 | 101 | 11 |
ERK2 | 102 | 9 |
ERK8 | 36 | 6 |
GSK3 beta | 100 | 1 |
HIPK2 | 60 | 0 |
HIPK3 | 93 | 11 |
IKK beta | 99 | 0 |
JNK1 | 96 | 10 |
JNK2 | 95 | 10 |
JNK3 | 80 | 8 |
Lck | 115 | 8 |
MAPKAP-K2 | 118 | 9 |
MAPKAP-K3 | 121 | 12 |
MARK3 | 99 | 2 |
MELK | 49 | 3 |
MKK1 | 99 | 6 |
MNK1 | 102 | 13 |
MNK2 | 74 | 0 |
MSK1 | 80 | 0 |
MST2 | 84 | 9 |
NEK2a | 96 | 1 |
NEK6 | 104 | 9 |
NEK7 | 94 | 9 |
p38 alpha MAPK | 95 | 6 |
p38 beta MAPK | 112 | 2 |
p38 delta MAPK | 95 | 6 |
p38 gamma MAPK | 106 | 8 |
PAK4 | 85 | 8 |
PAK5 | 102 | 0 |
PAK6 | 108 | 1 |
PDK1 | 74 | 6 |
PHK | 58 | 13 |
PIM1 | 50 | 10 |
PIM2 | 78 | 9 |
PIM3 | 48 | 1 |
PKA | 106 | 6 |
PKB alpha | 82 | 6 |
PKB beta | 108 | 8 |
PKC alpha | 96 | 3 |
PKC zeta | 128 | 12 |
PKD1 | 96 | 2 |
PLK1 | 90 | 9 |
PRAK | 105 | 8 |
PRK2 | 95 | 9 |
ROCK 2 | 125 | 3 |
RSK1 | 77 | 0 |
RSK2 | 77 | 8 |
S6K1 | 93 | 9 |
SGK1 | 79 | 3 |
SmMLCK | 78 | 9 |
Src | 108 | 2 |
SRPK1 | 111 | 1 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
AMPK | 73 | 7 |
ASK1 | 77 | 2 |
Aurora A | 100 | 11 |
Aurora B | 62 | 11 |
BRSK1 | 56 | 5 |
BRSK2 | 50 | 9 |
BTK | 75 | 2 |
CAMK1 | 73 | 7 |
CAMKK beta | 74 | 6 |
CDK2-Cyclin A | 59 | 3 |
CHK1 | 79 | 2 |
CHK2 | 79 | 13 |
CK1 delta | 94 | 8 |
CK2 | 82 | 6 |
CLK2 | 55 | 4 |
CSK | 87 | 3 |
DAPK1 | 62 | 0 |
DYRK1A | 61 | 8 |
DYRK2 | 15 | 2 |
DYRK3 |
8
|
0 |
EF2K | 69 | 11 |
EPH-A2 | 81 | 8 |
EPH-A4 | 107 | 5 |
EPH-B1 | 97 | 13 |
EPH-B2 | 116 | 7 |
EPH-B3 | 88 | 12 |
EPH-B4 | 99 | 6 |
ERK1 | 88 | 10 |
ERK2 | 79 | 1 |
ERK8 |
10
|
1 |
FGF-R1 | 85 | 3 |
GCK | 73 | 0 |
GSK3 beta | 80 | 5 |
HER4 | 59 | 3 |
HIPK1 | 48 | 8 |
HIPK2 | 30 | 11 |
HIPK3 | 41 | 3 |
IGF-1R | 59 | 5 |
IKK beta | 70 | 1 |
IKK epsilon | 59 | 2 |
IR | 50 | 10 |
IRAK4 | 73 | 3 |
IRR | 62 | 2 |
JAK2 | 27 | 2 |
JNK1 | 108 | 5 |
JNK2 | 86 | 12 |
JNK3 | 87 | 8 |
Lck | 97 | 7 |
LKB1 | 69 | 2 |
MAPKAP-K2 | 88 | 3 |
MAPKAP-K3 | 64 | 2 |
MARK1 | 96 | 3 |
MARK2 | 86 | 3 |
MARK3 | 82 | 4 |
MARK4 | 99 | 6 |
MEKK1 | 90 | 10 |
MELK | 50 | 6 |
MINK1 | 66 | 8 |
MKK1 | 81 | 9 |
MKK2 | 91 | 4 |
MKK6 | 87 | 9 |
MLK1 | 44 | 3 |
MLK3 | 35 | 2 |
MNK1 | 66 | 6 |
MNK2 | 96 | 10 |
MSK1 | 65 | 7 |
MST2 | 69 | 9 |
MST4 | 68 | 5 |
NEK2a | 91 | 1 |
NEK6 | 96 | 3 |
NUAK1 | 68 | 5 |
p38 alpha MAPK | 97 | 6 |
p38 beta MAPK | 93 | 3 |
p38 delta MAPK | 91 | 2 |
p38 gamma MAPK | 78 | 6 |
PAK2 | 83 | 2 |
PAK4 | 80 | 7 |
PAK5 | 83 | 3 |
PAK6 | 106 | 8 |
PDK1 | 97 | 4 |
PHK | 21 | 4 |
PIM1 | 30 | 5 |
PIM2 | 37 | 3 |
PIM3 | 44 | 2 |
PKA | 101 | 5 |
PKB alpha | 89 | 5 |
PKB beta | 67 | 13 |
PKC alpha | 82 | 3 |
PKC zeta | 105 | 1 |
PKD1 | 105 | 8 |
PLK1 | 87 | 2 |
PRAK | 85 | 1 |
PRK2 | 70 | 6 |
RIPK2 | 51 | 0 |
ROCK 2 | 83 | 2 |
RSK1 | 63 | 1 |
RSK2 | 72 | 3 |
S6K1 | 69 | 10 |
SGK1 | 94 | 3 |
SmMLCK | 63 | 8 |
Src | 81 | 6 |
SRPK1 | 87 | 12 |
SYK | 92 | 14 |
TAK1 | 83 | 1 |
TAO1 | 32 | 1 |
TBK1 | 79 | 2 |
TrkA | 67 | 8 |
TTK | 83 | 3 |
VEGFR1 | 51 | 5 |
YES1 | 77 | 3 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
AMPK | 16 | 1 |
Aurora B | 22 | 2 |
Aurora C | 32 | 1 |
BRSK2 | 13 | 2 |
CAMK1 | 38 | 9 |
CAMKK alpha | 30 | 3 |
CAMKK beta | 28 | 6 |
CDK2-Cyclin A | 34 | 5 |
CHK1 | 29 | 8 |
CHK2 | 14 | 0 |
CK1 delta | 46 | 2 |
CK2 | 49 | 0 |
CSK | 68 | 1 |
DYRK1A | 17 | 0 |
DYRK2 |
1
|
0 |
DYRK3 |
2
|
0 |
EF2K | 87 | 3 |
ERK1 | 92 | 0 |
ERK2 | 100 | 2 |
ERK8 | 12 | 4 |
GSK3 beta | 37 | 1 |
HIPK2 |
3
|
0 |
HIPK3 | 12 | 0 |
IKK beta | 46 | 2 |
JNK1 | 101 | 7 |
JNK2 | 103 | 5 |
JNK3 | 114 | 15 |
Lck | 59 | 9 |
MAPKAP-K2 | 71 | 9 |
MAPKAP-K3 | 97 | 13 |
MARK3 | 41 | 9 |
MELK |
8
|
3 |
MKK1 | 75 | 3 |
MNK1 | 125 | 1 |
MNK2 | 34 | 8 |
MSK1 | 16 | 6 |
MST2 | 28 | 2 |
NEK2a | 83 | 5 |
NEK6 | 87 | 2 |
NEK7 | 95 | 3 |
p38 alpha MAPK | 75 | 4 |
p38 beta MAPK | 108 | 10 |
p38 delta MAPK | 72 | 9 |
p38 gamma MAPK | 65 | 2 |
PAK4 | 67 | 5 |
PAK5 | 75 | 3 |
PAK6 | 100 | 3 |
PDK1 | 56 | 11 |
PHK | 23 | 7 |
PIM1 |
4
|
0 |
PIM2 | 27 | 8 |
PIM3 |
2
|
0 |
PKA | 91 | 2 |
PKB alpha | 63 | 11 |
PKB beta | 76 | 11 |
PKC alpha | 58 | 3 |
PKC zeta | 99 | 4 |
PKD1 | 51 | 0 |
PLK1 | 78 | 9 |
PRAK | 56 | 5 |
PRK2 | 21 | 6 |
ROCK 2 | 21 | 7 |
RSK1 | 15 | 1 |
RSK2 | 18 | 0 |
S6K1 | 15 | 1 |
SGK1 | 23 | 1 |
SmMLCK | 15 | 5 |
Src | 47 | 2 |
SRPK1 | 93 | 5 |