Inhibitor | ML-9, Hydrochloride  

Compound name Brutto MW CAS PubChem CID Action Reference Reference
ML-9, Hydrochloride   C15H17ClN2O2S • HCl 361.30 105637-50-1 108047 MLCK Reig J.A. (1993) Neurochem. Res. 18 317 Nagatsu T. (1987) Biochem. Biophys. Res. Commun. 143 1045

Screening Results Chart

Screening Results Tables

Screen Conc: 100.00µM
Kinase % Activity Remaining Sort descending Standard Deviation
PRK2
1
1
BRSK2
2
5
ROCK 2
6
0
PIM1
7
0
PIM3
7
0
MSK1 11 3
RSK1 12 0
S6K1 13 1
CDK2-Cyclin A 13 1
CAMK1 17 3
RSK2 19 1
PKA 25 5
CK2 25 2
PKC alpha 27 0
MNK1 28 4
DYRK3 30 2
SmMLCK 31 0
AMPK 32 3
PRAK 37 6
MNK2 40 2
PIM2 43 6
HIPK2 43 1
PKB alpha 44 4
DYRK1A 46 5
PHK 47 6
PKD1 48 5
PKC zeta 50 5
ERK8 50 2
Aurora B 57 2
PKB beta 58 3
CK1 delta 58 3
SGK1 59 4
MELK 66 7
IKK beta 67 1
HIPK3 68 5
MAPKAP-K2 69 4
Aurora C 73 3
MST2 74 4
CAMKK beta 75 1
MKK1 75 3
CSK 78 2
DYRK2 79 6
MAPKAP-K3 79 2
Lck 81 1
PAK5 85 4
p38 beta MAPK 86 1
p38 gamma MAPK 87 4
PDK1 87 2
p38 delta MAPK 88 4
GSK3 beta 88 1
ERK1 91 1
ERK2 91 8
SRPK1 92 1
JNK2 92 4
JNK3 92 0
p38 alpha MAPK 92 6
PAK4 94 1
CHK1 94 2
NEK2a 94 3
PLK1 98 7
Src 100 1
NEK6 105 1
CAMKK alpha 108 1
PAK6 108 4
CHK2 108 5
JNK1 115 1
EF2K 122 1
NEK7 122 6
MARK3 130 1
Screen Conc: 10.00µM
Kinase % Activity Remaining Sort descending Standard Deviation
PRK2 15 0
ROCK 2 28 0
MSK1 30 1
S6K1 32 6
RSK1 43 8
CDK2-Cyclin A 57 2
MKK1 58 14
PKA 61 3
Aurora B 63 2
PIM2 63 0
p38 delta MAPK 65 13
MNK1 66 0
RSK2 67 6
IKK beta 71 1
PKC alpha 72 2
CAMK1 74 8
Lck 75 0
JNK3 76 1
PRAK 77 1
CHK2 77 5
CK2 78 4
CSK 80 8
p38 beta MAPK 80 4
GSK3 beta 80 5
MNK2 81 9
SGK1 82 11
MST2 82 0
Src 82 3
NEK2a 83 0
JNK1 84 9
ERK8 84 10
DYRK1A 84 16
PKD1 85 8
AMPK 85 14
MAPKAP-K2 85 4
CHK1 86 5
SRPK1 87 16
p38 alpha MAPK 88 3
EF2K 88 12
PKB alpha 89 5
p38 gamma MAPK 91 4
CK1 delta 91 3
NEK7 92 8
PKB beta 92 4
SmMLCK 95 40
PHK 95 5
PDK1 96 7
ERK2 96 7
MAPKAP-K3 97 6
PLK1 101 6
MARK3 103 5
NEK6 103 14