Compound name | Brutto | MW | CAS | PubChem CID | Action | Reference | Reference |
---|---|---|---|---|---|---|---|
Genistein | C15H10O5 | 270.20 | 446-72-0 | 5280961 | Tyrosine-kinases | Constantinou A. and Huberman E. (1995) Proc. Soc. Exp. Biol. Med. 208 109 | Wei H. (1995) Proc. Soc. Exp. Biol. Med. 208 124 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
AMPK | 84 | 11 |
Aurora B | 48 | 5 |
CAMK1 | 77 | 3 |
CDK2-Cyclin A | 96 | 3 |
CHK1 | 83 | 17 |
CHK2 | 67 | 2 |
CK1 delta | 51 | 0 |
CK2 | 91 | 0 |
CSK | 92 | 16 |
DYRK1A | 53 | 8 |
EF2K | 94 | 2 |
ERK2 | 103 | 3 |
ERK8 | 53 | 5 |
GSK3 beta | 57 | 7 |
IKK beta | 78 | 9 |
JNK1 | 80 | 8 |
JNK2 | 77 | 3 |
Lck | 73 | 2 |
MAPKAP-K2 | 89 | 6 |
MAPKAP-K3 | 93 | 8 |
MARK3 | 93 | 8 |
MKK1 | 68 | 3 |
MNK1 | 57 | 2 |
MNK2 | 51 | 1 |
MSK1 | 97 | 2 |
MST2 | 80 | 0 |
NEK2a | 74 | 0 |
NEK6 | 98 | 1 |
NEK7 | 85 | 7 |
p38 alpha MAPK | 83 | 19 |
p38 beta MAPK | 90 | 4 |
p38 delta MAPK | 81 | 20 |
p38 gamma MAPK | 104 | 13 |
PDK1 | 90 | 23 |
PHK | 106 | 10 |
PIM2 | 38 | 4 |
PKA | 81 | 16 |
PKB alpha | 105 | 3 |
PKB beta | 96 | 0 |
PKC alpha | 81 | 3 |
PKD1 | 91 | 9 |
PLK1 | 99 | 14 |
PRAK | 76 | 0 |
PRK2 | 74 | 4 |
ROCK 2 | 77 | 1 |
RSK1 | 105 | 15 |
RSK2 | 98 | 0 |
S6K1 | 74 | 11 |
SGK1 | 65 | 7 |
SmMLCK | 75 | 12 |
Src | 94 | 2 |
SRPK1 | 92 | 10 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
AMPK | 97 | 1 |
ASK1 | 93 | 9 |
Aurora A | 110 | 2 |
Aurora B | 90 | 12 |
BRSK1 | 100 | 6 |
BRSK2 | 117 | 9 |
BTK | 88 | 9 |
CAMK1 | 93 | 6 |
CAMKK beta | 94 | 8 |
CDK2-Cyclin A | 101 | 2 |
CHK1 | 95 | 13 |
CHK2 | 83 | 4 |
CK1 delta | 90 | 7 |
CK2 | 95 | 9 |
CLK2 | 71 | 9 |
CSK | 96 | 4 |
DAPK1 | 77 | 2 |
DYRK1A | 54 | 2 |
DYRK2 | 78 | 5 |
DYRK3 | 58 | 3 |
EF2K | 87 | 8 |
EPH-A2 | 85 | 7 |
EPH-A4 | 91 | 0 |
EPH-B1 | 86 | 12 |
EPH-B2 | 109 | 9 |
EPH-B3 | 101 | 6 |
EPH-B4 | 107 | 13 |
ERK1 | 109 | 7 |
ERK2 | 106 | 6 |
ERK8 | 95 | 7 |
FGF-R1 | 96 | 4 |
GCK | 48 | 1 |
GSK3 beta | 90 | 0 |
HER4 | 86 | 2 |
HIPK1 | 93 | 4 |
HIPK2 | 79 | 12 |
HIPK3 | 102 | 3 |
IGF-1R | 96 | 3 |
IKK beta | 102 | 8 |
IKK epsilon | 106 | 5 |
IR | 95 | 9 |
IRAK4 | 86 | 9 |
IRR | 58 | 2 |
JAK2 | 84 | 9 |
JNK1 | 103 | 10 |
JNK2 | 98 | 5 |
JNK3 | 92 | 6 |
Lck | 104 | 2 |
LKB1 | 96 | 2 |
MAPKAP-K2 | 108 | 5 |
MAPKAP-K3 | 87 | 1 |
MARK1 | 106 | 0 |
MARK2 | 103 | 6 |
MARK3 | 108 | 7 |
MARK4 | 99 | 4 |
MEKK1 | 98 | 1 |
MELK | 88 | 9 |
MINK1 | 109 | 9 |
MKK1 | 86 | 14 |
MKK2 | 102 | 7 |
MKK6 | 98 | 14 |
MLK1 | 114 | 9 |
MLK3 | 95 | 3 |
MNK1 | 88 | 1 |
MNK2 | 61 | 5 |
MSK1 | 87 | 11 |
MST2 | 81 | 2 |
MST4 | 96 | 4 |
NEK2a | 115 | 5 |
NEK6 | 93 | 2 |
NUAK1 | 104 | 2 |
p38 alpha MAPK | 117 | 13 |
p38 beta MAPK | 101 | 11 |
p38 delta MAPK | 100 | 2 |
p38 gamma MAPK | 95 | 3 |
PAK2 | 99 | 7 |
PAK4 | 78 | 4 |
PAK5 | 97 | 3 |
PAK6 | 83 | 9 |
PDK1 | 87 | 3 |
PHK | 106 | 6 |
PIM1 | 54 | 0 |
PIM2 | 90 | 9 |
PIM3 | 40 | 0 |
PKA | 103 | 10 |
PKB alpha | 104 | 7 |
PKB beta | 83 | 6 |
PKC alpha | 81 | 3 |
PKC zeta | 99 | 6 |
PKD1 | 98 | 7 |
PLK1 | 101 | 10 |
PRAK | 89 | 6 |
PRK2 | 105 | 13 |
RIPK2 | 48 | 5 |
ROCK 2 | 95 | 1 |
RSK1 | 97 | 3 |
RSK2 | 103 | 14 |
S6K1 | 84 | 8 |
SGK1 | 100 | 3 |
SmMLCK | 77 | 1 |
Src | 92 | 9 |
SRPK1 | 102 | 8 |
SYK | 124 | 9 |
TAK1 | 96 | 5 |
TAO1 | 93 | 3 |
TBK1 | 99 | 3 |
TrkA | 105 | 4 |
TTK | 107 | 5 |
VEGFR1 | 70 | 15 |
YES1 | 105 | 13 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
AMPK | 92 | 12 |
ASK1 | 96 | 4 |
Aurora A | 79 | 14 |
Aurora B | 61 | 1 |
BRSK1 | 83 | 9 |
BRSK2 | 81 | 5 |
BTK | 80 | 5 |
CAMK1 | 95 | 11 |
CAMKK beta | 89 | 1 |
CDK2-Cyclin A | 78 | 3 |
CHK1 | 94 | 15 |
CHK2 | 82 | 9 |
CK1 delta | 44 | 2 |
CK2 | 80 | 8 |
CLK2 | 39 | 0 |
CSK | 91 | 1 |
DAPK1 | 57 | 10 |
DYRK1A | 32 | 3 |
DYRK2 | 46 | 0 |
DYRK3 | 24 | 3 |
EF2K | 88 | 2 |
EPH-A2 | 96 | 4 |
EPH-A4 | 90 | 12 |
EPH-B1 | 97 | 7 |
EPH-B2 | 105 | 9 |
EPH-B3 | 105 | 0 |
EPH-B4 | 99 | 7 |
ERK1 | 92 | 3 |
ERK2 | 103 | 8 |
ERK8 | 67 | 14 |
FGF-R1 | 85 | 8 |
GCK | 21 | 3 |
GSK3 beta | 50 | 4 |
HER4 | 84 | 10 |
HIPK1 | 94 | 2 |
HIPK2 | 57 | 3 |
HIPK3 | 86 | 3 |
IGF-1R | 61 | 3 |
IKK beta | 92 | 2 |
IKK epsilon | 75 | 1 |
IR | 97 | 8 |
IRAK4 | 89 | 0 |
IRR | 43 | 2 |
JAK2 | 50 | 1 |
JNK1 | 88 | 1 |
JNK2 | 94 | 5 |
JNK3 | 78 | 10 |
Lck | 84 | 0 |
LKB1 | 89 | 3 |
MAPKAP-K2 | 100 | 5 |
MAPKAP-K3 | 94 | 6 |
MARK1 | 96 | 6 |
MARK2 | 92 | 10 |
MARK3 | 104 | 1 |
MARK4 | 107 | 7 |
MEKK1 | 89 | 9 |
MELK | 76 | 4 |
MINK1 | 74 | 4 |
MKK1 | 93 | 4 |
MKK2 | 92 | 15 |
MKK6 | 99 | 7 |
MLK1 | 98 | 5 |
MLK3 | 64 | 6 |
MNK1 | 63 | 3 |
MNK2 | 91 | 3 |
MSK1 | 76 | 3 |
MST2 | 91 | 2 |
MST4 | 94 | 2 |
NEK2a | 106 | 8 |
NEK6 | 98 | 7 |
NUAK1 | 77 | 9 |
p38 alpha MAPK | 97 | 1 |
p38 beta MAPK | 109 | 9 |
p38 delta MAPK | 94 | 3 |
p38 gamma MAPK | 98 | 10 |
PAK2 | 91 | 0 |
PAK4 | 97 | 5 |
PAK5 | 96 | 11 |
PAK6 | 100 | 4 |
PDK1 | 104 | 10 |
PHK | 102 | 11 |
PIM1 | 25 | 0 |
PIM2 | 48 | 0 |
PIM3 | 23 | 1 |
PKA | 98 | 1 |
PKB alpha | 107 | 7 |
PKB beta | 76 | 2 |
PKC alpha | 83 | 4 |
PKC zeta | 91 | 8 |
PKD1 | 91 | 5 |
PLK1 | 102 | 2 |
PRAK | 93 | 8 |
PRK2 | 83 | 13 |
RIPK2 | 21 | 5 |
ROCK 2 | 85 | 2 |
RSK1 | 82 | 4 |
RSK2 | 91 | 12 |
S6K1 | 67 | 2 |
SGK1 | 82 | 3 |
SmMLCK | 51 | 6 |
Src | 75 | 6 |
SRPK1 | 87 | 11 |
SYK | 110 | 1 |
TAK1 | 97 | 2 |
TAO1 | 85 | 3 |
TBK1 | 90 | 7 |
TrkA | 99 | 2 |
TTK | 78 | 5 |
VEGFR1 | 62 | 2 |
YES1 | 74 | 4 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
AMPK | 58 | 2 |
Aurora B | 13 | 2 |
CAMK1 | 61 | 1 |
CDK2-Cyclin A | 83 | 3 |
CHK1 | 73 | 6 |
CHK2 | 47 | 4 |
CK1 delta |
6
|
4 |
CK2 | 43 | 10 |
CSK | 70 | 3 |
DYRK1A | 11 | 0 |
EF2K | 87 | 0 |
ERK2 | 101 | 8 |
ERK8 | 19 | 0 |
GSK3 beta | 20 | 0 |
IKK beta | 64 | 2 |
JNK1 | 68 | 5 |
JNK2 | 73 | 8 |
Lck | 40 | 1 |
MAPKAP-K2 | 80 | 0 |
MAPKAP-K3 | 85 | 0 |
MARK3 | 86 | 1 |
MKK1 | 56 | 12 |
MNK1 | 22 | 0 |
MNK2 | 14 | 5 |
MSK1 | 41 | 4 |
MST2 | 73 | 10 |
NEK2a | 81 | 13 |
NEK6 | 71 | 4 |
NEK7 | 64 | 0 |
p38 alpha MAPK | 114 | 7 |
p38 beta MAPK | 82 | 1 |
p38 delta MAPK | 91 | 4 |
p38 gamma MAPK | 82 | 4 |
PDK1 | 80 | 3 |
PHK | 79 | 5 |
PIM2 |
8
|
0 |
PKA | 71 | 7 |
PKB alpha | 96 | 5 |
PKB beta | 73 | 1 |
PKC alpha | 59 | 0 |
PKD1 | 73 | 2 |
PLK1 | 85 | 8 |
PRAK | 73 | 6 |
PRK2 | 39 | 4 |
ROCK 2 | 62 | 3 |
RSK1 | 53 | 1 |
RSK2 | 54 | 11 |
S6K1 | 44 | 1 |
SGK1 | 25 | 2 |
SmMLCK | 19 | 2 |
Src | 48 | 2 |
SRPK1 | 82 | 4 |