Inhibitor | FMK (Caspase Inhibitor I)  

Compound name Brutto MW CAS PubChem CID Action Reference Reference
FMK (Caspase Inhibitor I)   C22H30FN3O7 467.50 187389-52-2 5737 Caspase Martin U. (2007) Apoptosis 12 525 Misaghi S. (2004) Chem. Biol. 11 1677

Screening Results Chart

Screening Results Tables

Screen Conc: 3.00µM
Kinase Sort ascending % Activity Remaining Standard Deviation
SRPK1 85 1
Src
10
1
SmMLCK 82 4
SGK1 107 8
S6K1 33 2
RSK2 74 2
RSK1 92 6
ROCK 2 86 7
PRK2 83 3
PRAK 97 5
PLK1 82 5
PKD1 83 4
PKC zeta 91 5
PKC alpha 85 7
PKB beta 97 4
PKB alpha 82 3
PKA 85 7
PIM3 56 6
PIM2 85 10
PIM1 61 6
PHK 93 5
PDK1 89 10
PAK6 93 5
PAK5 88 6
PAK4 91 1
p38 gamma MAPK 92 7
p38 delta MAPK 103 9
p38 beta MAPK 85 4
p38 alpha MAPK 72 2
NEK7 92 8
NEK6 90 4
NEK2a 95 4
MST2 76 4
MSK1 75 3
MNK2 65 6
MNK1 42 2
MKK1 80 8
MELK 65 8
MARK3 80 3
MAPKAP-K3 92 6
MAPKAP-K2 94 10
Lck
10
1
JNK3 89 4
JNK2 83 5
JNK1 81 3
IKK beta 92 8
HIPK3 79 9
HIPK2 79 11
GSK3 beta 65 6
ERK8 58 4
ERK2 79 5
ERK1 92 6
EF2K 97 8
DYRK3 68 7
DYRK2 91 8
DYRK1A 86 11
CSK 55 7
CK2 92 10
CK1 delta 63 6
CHK2 81 9
CHK1 88 4
CDK2-Cyclin A 80 7
CAMKK beta 49 3
CAMKK alpha 70 12
CAMK1 77 9
BRSK2 53 6
Aurora C 75 6
Aurora B 59 3
AMPK 79 4