Inhibitor | FMK (Caspase Inhibitor I)  

Compound name Brutto MW CAS PubChem CID Action Reference Reference
FMK (Caspase Inhibitor I)   C22H30FN3O7 467.50 187389-52-2 5737 Caspase Martin U. (2007) Apoptosis 12 525 Misaghi S. (2004) Chem. Biol. 11 1677

Screening Results Chart

Screening Results Tables

Screen Conc: 3.00µM
Kinase % Activity Remaining Sort ascending Standard Deviation
SGK1 107 8
p38 delta MAPK 103 9
EF2K 97 8
PRAK 97 5
PKB beta 97 4
NEK2a 95 4
MAPKAP-K2 94 10
PHK 93 5
PAK6 93 5
p38 gamma MAPK 92 7
RSK1 92 6
MAPKAP-K3 92 6
CK2 92 10
NEK7 92 8
IKK beta 92 8
ERK1 92 6
PKC zeta 91 5
PAK4 91 1
DYRK2 91 8
NEK6 90 4
JNK3 89 4
PDK1 89 10
CHK1 88 4
PAK5 88 6
ROCK 2 86 7
DYRK1A 86 11
PKA 85 7
PIM2 85 10
SRPK1 85 1
PKC alpha 85 7
p38 beta MAPK 85 4
JNK2 83 5
PRK2 83 3
PKD1 83 4
PLK1 82 5
PKB alpha 82 3
SmMLCK 82 4
JNK1 81 3
CHK2 81 9
CDK2-Cyclin A 80 7
MARK3 80 3
MKK1 80 8
ERK2 79 5
HIPK2 79 11
HIPK3 79 9
AMPK 79 4
CAMK1 77 9
MST2 76 4
MSK1 75 3
Aurora C 75 6
RSK2 74 2
p38 alpha MAPK 72 2
CAMKK alpha 70 12
DYRK3 68 7
GSK3 beta 65 6
MNK2 65 6
MELK 65 8
CK1 delta 63 6
PIM1 61 6
Aurora B 59 3
ERK8 58 4
PIM3 56 6
CSK 55 7
BRSK2 53 6
CAMKK beta 49 3
MNK1 42 2
S6K1 33 2
Src
10
1
Lck
10
1