Inhibitor | FMK (Caspase Inhibitor I)  

Compound name Brutto MW CAS PubChem CID Action Reference Reference
FMK (Caspase Inhibitor I)   C22H30FN3O7 467.50 187389-52-2 5737 Caspase Martin U. (2007) Apoptosis 12 525 Misaghi S. (2004) Chem. Biol. 11 1677

Screening Results Chart

Screening Results Tables

Screen Conc: 3.00µM
Kinase % Activity Remaining Sort descending Standard Deviation
Src
10
1
Lck
10
1
S6K1 33 2
MNK1 42 2
CAMKK beta 49 3
BRSK2 53 6
CSK 55 7
PIM3 56 6
ERK8 58 4
Aurora B 59 3
PIM1 61 6
CK1 delta 63 6
MELK 65 8
GSK3 beta 65 6
MNK2 65 6
DYRK3 68 7
CAMKK alpha 70 12
p38 alpha MAPK 72 2
RSK2 74 2
MSK1 75 3
Aurora C 75 6
MST2 76 4
CAMK1 77 9
ERK2 79 5
HIPK2 79 11
HIPK3 79 9
AMPK 79 4
MARK3 80 3
MKK1 80 8
CDK2-Cyclin A 80 7
JNK1 81 3
CHK2 81 9
PKB alpha 82 3
SmMLCK 82 4
PLK1 82 5
JNK2 83 5
PRK2 83 3
PKD1 83 4
PKA 85 7
PIM2 85 10
SRPK1 85 1
PKC alpha 85 7
p38 beta MAPK 85 4
DYRK1A 86 11
ROCK 2 86 7
PAK5 88 6
CHK1 88 4
PDK1 89 10
JNK3 89 4
NEK6 90 4
DYRK2 91 8
PKC zeta 91 5
PAK4 91 1
RSK1 92 6
MAPKAP-K3 92 6
CK2 92 10
NEK7 92 8
IKK beta 92 8
ERK1 92 6
p38 gamma MAPK 92 7
PAK6 93 5
PHK 93 5
MAPKAP-K2 94 10
NEK2a 95 4
PRAK 97 5
PKB beta 97 4
EF2K 97 8
p38 delta MAPK 103 9
SGK1 107 8