Inhibitor | FMK (Caspase Inhibitor I)  

Compound name Brutto MW CAS PubChem CID Action Reference Reference
FMK (Caspase Inhibitor I)   C22H30FN3O7 467.50 187389-52-2 5737 Caspase Martin U. (2007) Apoptosis 12 525 Misaghi S. (2004) Chem. Biol. 11 1677

Screening Results Chart

Screening Results Tables

Screen Conc: 3.00µM
Kinase % Activity Remaining Standard Deviation
AMPK 79 4
Aurora B 59 3
Aurora C 75 6
BRSK2 53 6
CAMK1 77 9
CAMKK alpha 70 12
CAMKK beta 49 3
CDK2-Cyclin A 80 7
CHK1 88 4
CHK2 81 9
CK1 delta 63 6
CK2 92 10
CSK 55 7
DYRK1A 86 11
DYRK2 91 8
DYRK3 68 7
EF2K 97 8
ERK1 92 6
ERK2 79 5
ERK8 58 4
GSK3 beta 65 6
HIPK2 79 11
HIPK3 79 9
IKK beta 92 8
JNK1 81 3
JNK2 83 5
JNK3 89 4
Lck
10
1
MAPKAP-K2 94 10
MAPKAP-K3 92 6
MARK3 80 3
MELK 65 8
MKK1 80 8
MNK1 42 2
MNK2 65 6
MSK1 75 3
MST2 76 4
NEK2a 95 4
NEK6 90 4
NEK7 92 8
p38 alpha MAPK 72 2
p38 beta MAPK 85 4
p38 delta MAPK 103 9
p38 gamma MAPK 92 7
PAK4 91 1
PAK5 88 6
PAK6 93 5
PDK1 89 10
PHK 93 5
PIM1 61 6
PIM2 85 10
PIM3 56 6
PKA 85 7
PKB alpha 82 3
PKB beta 97 4
PKC alpha 85 7
PKC zeta 91 5
PKD1 83 4
PLK1 82 5
PRAK 97 5
PRK2 83 3
ROCK 2 86 7
RSK1 92 6
RSK2 74 2
S6K1 33 2
SGK1 107 8
SmMLCK 82 4
Src
10
1
SRPK1 85 1