Inhibitor | EGCG (Epigallocatechin Gallate)  

Compound name Brutto MW CAS PubChem CID Action Reference Reference
EGCG (Epigallocatechin Gallate)   C22H18O11 458.40 989-51-5 65064 PKC Dell'Aica I. (2004) EMBO Rep. 5 418-422 Tachibana H. (2004) Nat. Struct. Mol. Biol. 11 380

Screening Results Chart

Screening Results Tables

Screen Conc: 10.00µM
Kinase % Activity Remaining Standard Deviation
AMPK 66 2
Aurora B 12 3
BRSK2 23 1
BTK 18 0
CAMK1 19 8
CAMKK beta 65 2
CDK2-Cyclin A 88 4
CHK1 72 3
CHK2 61 1
CK1 delta 90 9
CK2 89 17
CSK 88 10
DYRK1A
6
0
DYRK2
0
1
DYRK3
5
0
EF2K 86 2
EPH-A2 76 0
EPH-B3
1
0
ERK1 17 1
ERK2 72 4
ERK8 20 0
FGF-R1
6
0
GSK3 beta 70 6
HIPK2 15 0
IGF-1R 19 4
IKK beta 21 3
IKK epsilon 27 4
IR 70 5
IRR 28 1
JNK1 106 8
JNK2 84 2
Lck 90 3
MAPKAP-K2 22 1
MARK3
6
1
MELK 53 1
MKK1 58 24
MNK1 71 10
MNK2 73 7
MSK1 40 4
MST2 37 0
MST4 24 1
NEK2a
5
1
NEK6 56 4
p38 alpha MAPK 80 8
p38 beta MAPK 96 20
p38 delta MAPK 102 17
p38 gamma MAPK 98 15
PAK4 22 1
PAK5 35 1
PAK6
8
4
PDK1 73 0
PHK 75 6
PIM1 15 2
PIM2 47 0
PIM3 17 0
PKA 87 1
PKB alpha 75 20
PKB beta
1
0
PKC alpha 81 3
PKC zeta
2
1
PKD1 16 1
PLK1
7
2
PRAK
5
2
PRK2 82 3
ROCK 2 74 5
RSK1 46 2
RSK2
6
6
S6K1 37 1
SGK1 58 2
SmMLCK 51 2
Src 21 0
SRPK1
5
3
SYK 67 8
TBK1 65 4
VEGFR1 20 1
YES1 12 3