| Compound name | Brutto | MW | CAS | PubChem CID | Action | Reference | Reference |
|---|---|---|---|---|---|---|---|
| D 4476 | C23H18N4O3 | 398.41 | 301836-43-1 | 6419753 | CK1 | Liverton N.J. (1999) J. Med. Chem 42 2180-2190 |
| Kinase | % Activity Remaining | Standard Deviation |
|---|---|---|
| AMPK | 98 | 0 |
| Aurora B | 75 | 5 |
| Aurora C | 81 | 4 |
| BRSK2 | 89 | 5 |
| BTK | 71 | 5 |
| CAMK1 | 88 | 2 |
| CAMKK alpha | 89 | 1 |
| CAMKK beta | 100 | 2 |
| CDK2-Cyclin A | 112 | 8 |
| CHK1 | 83 | 8 |
| CHK2 | 92 | 5 |
| CK1 delta |
3
|
0 |
| CK2 | 82 | 5 |
| CSK | 81 | 5 |
| DYRK1A | 86 | 6 |
| DYRK2 | 93 | 3 |
| DYRK3 | 76 | 1 |
| EF2K | 100 | 1 |
| EPH-A2 | 97 | 12 |
| EPH-B3 | 115 | 8 |
| ERK1 | 101 | 3 |
| ERK2 | 85 | 1 |
| ERK8 | 79 | 4 |
| FGF-R1 | 69 | 2 |
| GSK3 beta | 88 | 5 |
| HIPK2 | 80 | 4 |
| HIPK3 | 96 | 2 |
| IGF-1R | 77 | 0 |
| IKK beta | 63 | 3 |
| IKK epsilon | 88 | 4 |
| IR | 108 | 9 |
| IRR | 55 | 1 |
| JNK1 | 86 | 4 |
| JNK2 | 76 | 6 |
| JNK3 | 81 | 0 |
| Lck | 82 | 5 |
| MAPKAP-K2 | 99 | 4 |
| MAPKAP-K3 | 98 | 2 |
| MARK3 | 82 | 4 |
| MELK | 83 | 1 |
| MKK1 | 93 | 2 |
| MNK1 | 81 | 1 |
| MNK2 | 88 | 4 |
| MSK1 | 90 | 7 |
| MST2 | 96 | 2 |
| MST4 | 83 | 0 |
| NEK2a | 89 | 6 |
| NEK6 | 78 | 1 |
| NEK7 | 99 | 6 |
| p38 alpha MAPK | 38 | 1 |
| p38 beta MAPK | 55 | 2 |
| p38 delta MAPK | 88 | 2 |
| p38 gamma MAPK | 87 | 0 |
| PAK4 | 105 | 1 |
| PAK5 | 100 | 1 |
| PAK6 | 103 | 4 |
| PDK1 | 84 | 1 |
| PHK | 88 | 3 |
| PIM1 | 93 | 7 |
| PIM2 | 90 | 4 |
| PIM3 | 82 | 4 |
| PKA | 85 | 5 |
| PKB alpha | 106 | 8 |
| PKB beta | 88 | 1 |
| PKC alpha | 94 | 5 |
| PKC zeta | 81 | 0 |
| PKD1 | 43 | 4 |
| PLK1 | 91 | 1 |
| PRAK | 77 | 2 |
| PRK2 | 107 | 4 |
| ROCK 2 | 104 | 1 |
| RSK1 | 81 | 1 |
| RSK2 | 81 | 1 |
| S6K1 | 76 | 5 |
| SGK1 | 73 | 1 |
| SmMLCK | 80 | 5 |
| Src | 82 | 0 |
| SRPK1 | 84 | 5 |
| SYK | 82 | 2 |
| TBK1 | 95 | 9 |
| VEGFR1 | 85 | 12 |
| YES1 | 81 | 2 |