Compound name | Brutto | MW | CAS | PubChem CID | Action | Reference | Reference |
---|---|---|---|---|---|---|---|
KU55933 | C21H17NO3S2 | 395.49 | 587871-26-9 | 5278396 | ATM | Li Y. (2010) Mol. Cancer Ther. 2010 Jan. 9(1) 113-25 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
ABL | 101 | 5 |
AMPK (hum) | 65 | 8 |
ASK1 | 108 | 17 |
Aurora A | 99 | 10 |
Aurora B | 64 | 14 |
BRK | 91 | 3 |
BRSK1 | 85 | 1 |
BRSK2 | 104 | 4 |
BTK | 90 | 2 |
CAMK1 | 90 | 4 |
CAMKK beta | 82 | 6 |
CDK2-Cyclin A | 84 | 7 |
CDK9-Cyclin T1 | 88 | 2 |
CHK1 | 74 | 0 |
CHK2 | 97 | 0 |
CK1 delta | 81 | 2 |
CK1 gamma 2 | 93 | 6 |
CK2 | 96 | 1 |
CLK2 | 93 | 1 |
CSK | 112 | 17 |
DAPK1 | 98 | 2 |
DDR2 | 89 | 3 |
DYRK1A | 76 | 6 |
DYRK2 | 89 | 1 |
DYRK3 | 100 | 2 |
EF2K | 97 | 13 |
EIF2AK3 | 98 | 1 |
EPH-A2 | 104 | 12 |
EPH-A4 | 88 | 12 |
EPH-B1 | 98 | 4 |
EPH-B2 | 85 | 1 |
EPH-B3 | 91 | 5 |
EPH-B4 | 97 | 17 |
ERK1 | 94 | 3 |
ERK2 | 78 | 2 |
ERK5 | 88 | 1 |
ERK8 | 75 | 2 |
FGF-R1 | 91 | 14 |
GCK | 85 | 16 |
GSK3 beta | 94 | 4 |
HER4 | 96 | 6 |
HIPK1 | 79 | 7 |
HIPK2 | 84 | 11 |
HIPK3 | 82 | 4 |
IGF-1R | 79 | 6 |
IKK beta | 102 | 4 |
IKK epsilon | 73 | 6 |
IR | 77 | 12 |
IRAK1 | 87 | 7 |
IRAK4 | 80 | 1 |
IRR | 98 | 7 |
JAK2 | 83 | 12 |
JNK1 | 83 | 0 |
JNK2 | 86 | 0 |
JNK3 | 108 | 25 |
Lck | 86 | 4 |
LKB1 | 82 | 9 |
MAP4K3 | 82 | 5 |
MAP4K5 | 73 | 6 |
MAPKAP-K2 | 91 | 2 |
MAPKAP-K3 | 91 | 6 |
MARK1 | 69 | 3 |
MARK2 | 76 | 3 |
MARK3 | 62 | 10 |
MARK4 | 84 | 3 |
MEKK1 | 90 | 13 |
MELK | 67 | 2 |
MINK1 | 71 | 4 |
MKK1 | 71 | 15 |
MKK2 | 70 | 2 |
MKK6 | 78 | 1 |
MLK1 | 81 | 11 |
MLK3 | 68 | 2 |
MNK1 | 99 | 4 |
MNK2 | 94 | 2 |
MPSK1 | 90 | 2 |
MSK1 | 97 | 8 |
MST2 | 64 | 5 |
MST3 | 68 | 8 |
MST4 | 79 | 0 |
NEK2a | 100 | 1 |
NEK6 | 80 | 8 |
NUAK1 | 99 | 10 |
OSR1 | 89 | 5 |
p38 alpha MAPK | 87 | 2 |
p38 beta MAPK | 75 | 6 |
p38 delta MAPK | 76 | 4 |
p38 gamma MAPK | 67 | 14 |
PAK2 | 86 | 3 |
PAK4 | 119 | 17 |
PAK5 | 83 | 2 |
PAK6 | 88 | 6 |
PDGFRA | 106 | 31 |
PDK1 | 93 | 8 |
PHK | 110 | 21 |
PIM1 | 93 | 3 |
PIM2 | 108 | 14 |
PIM3 | 103 | 9 |
PINK | 81 | 6 |
PKA | 93 | 2 |
PKB alpha | 73 | 2 |
PKB beta | 87 | 5 |
PKC alpha | 89 | 11 |
PKC gamma | 95 | 4 |
PKC zeta | 98 | 1 |
PKD1 | 95 | 4 |
PLK1 | 87 | 13 |
PRAK | 94 | 6 |
PRK2 | 74 | 6 |
RIPK2 | 70 | 2 |
ROCK 2 | 82 | 5 |
RSK1 | 88 | 3 |
RSK2 | 74 | 6 |
S6K1 | 82 | 10 |
SGK1 | 94 | 2 |
SIK2 | 67 | 3 |
SIK3 | 72 | 5 |
SmMLCK | 84 | 1 |
Src | 85 | 15 |
SRPK1 | 87 | 8 |
STK33 | 95 | 5 |
SYK | 89 | 1 |
TAK1 | 68 | 4 |
TAO1 | 79 | 9 |
TBK1 | 92 | 13 |
TESK1 | 85 | 2 |
TGFBR1 | 75 | 1 |
TIE2 | 85 | 16 |
TLK1 | 88 | 1 |
TrkA | 94 | 2 |
TSSK1 | 72 | 2 |
TTBK1 | 87 | 2 |
TTBK2 | 94 | 9 |
TTK | 86 | 4 |
ULK1 | 69 | 3 |
ULK2 | 84 | 5 |
VEGFR1 | 78 | 8 |
WNK1 | 88 | 6 |
YES1 | 85 | 5 |
ZAP70 | 95 | 5 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
ABL | 101 | 6 |
AMPK (hum) | 100 | 7 |
ASK1 | 100 | 17 |
Aurora A | 95 | 7 |
Aurora B | 69 | 6 |
BRK | 81 | 3 |
BRSK1 | 94 | 10 |
BRSK2 | 94 | 10 |
BTK | 84 | 6 |
CAMK1 | 91 | 3 |
CAMKK beta | 93 | 6 |
CDK2-Cyclin A | 94 | 9 |
CDK9-Cyclin T1 | 88 | 8 |
CHK1 | 82 | 10 |
CHK2 | 101 | 8 |
CK1 delta | 79 | 1 |
CK1 gamma 2 | 62 | 3 |
CK2 | 99 | 1 |
CLK2 | 94 | 13 |
CSK | 119 | 29 |
DAPK1 | 107 | 22 |
DDR2 | 95 | 3 |
DYRK1A | 57 | 0 |
DYRK2 | 96 | 4 |
DYRK3 | 108 | 11 |
EF2K | 90 | 2 |
EIF2AK3 | 99 | 6 |
EPH-A2 | 107 | 10 |
EPH-A4 | 101 | 12 |
EPH-B1 | 102 | 1 |
EPH-B2 | 88 | 2 |
EPH-B3 | 86 | 9 |
EPH-B4 | 98 | 9 |
ERK1 | 99 | 12 |
ERK2 | 88 | 1 |
ERK5 | 79 | 13 |
ERK8 | 63 | 2 |
FGF-R1 | 85 | 10 |
GCK | 74 | 15 |
GSK3 beta | 93 | 3 |
HER4 | 92 | 3 |
HIPK1 | 78 | 2 |
HIPK2 | 90 | 9 |
HIPK3 | 86 | 4 |
IGF-1R | 84 | 2 |
IKK beta | 102 | 8 |
IKK epsilon | 77 | 3 |
IR | 91 | 21 |
IRAK1 | 95 | 8 |
IRAK4 | 80 | 1 |
IRR | 107 | 5 |
JAK2 | 96 | 6 |
JNK1 | 94 | 14 |
JNK2 | 86 | 14 |
JNK3 | 104 | 5 |
Lck | 87 | 2 |
LKB1 | 79 | 3 |
MAP4K3 | 83 | 14 |
MAP4K5 | 74 | 3 |
MAPKAP-K2 | 95 | 2 |
MAPKAP-K3 | 98 | 2 |
MARK1 | 86 | 4 |
MARK2 | 92 | 9 |
MARK3 | 68 | 10 |
MARK4 | 94 | 10 |
MEKK1 | 95 | 9 |
MELK | 89 | 12 |
MINK1 | 77 | 1 |
MKK1 | 90 | 7 |
MKK2 | 77 | 17 |
MKK6 | 75 | 9 |
MLK1 | 78 | 10 |
MLK3 | 79 | 13 |
MNK1 | 83 | 4 |
MNK2 | 102 | 4 |
MPSK1 | 101 | 7 |
MSK1 | 98 | 8 |
MST2 | 69 | 2 |
MST3 | 63 | 6 |
MST4 | 76 | 4 |
NEK2a | 101 | 16 |
NEK6 | 87 | 4 |
NUAK1 | 99 | 9 |
OSR1 | 99 | 2 |
p38 alpha MAPK | 92 | 10 |
p38 beta MAPK | 87 | 18 |
p38 delta MAPK | 83 | 1 |
p38 gamma MAPK | 77 | 8 |
PAK2 | 93 | 8 |
PAK4 | 100 | 24 |
PAK5 | 87 | 4 |
PAK6 | 97 | 8 |
PDGFRA | 102 | 13 |
PDK1 | 93 | 10 |
PHK | 103 | 12 |
PIM1 | 86 | 5 |
PIM2 | 97 | 3 |
PIM3 | 73 | 0 |
PINK | 78 | 4 |
PKA | 94 | 0 |
PKB alpha | 86 | 1 |
PKB beta | 89 | 3 |
PKC alpha | 103 | 11 |
PKC gamma | 103 | 9 |
PKC zeta | 96 | 3 |
PKD1 | 88 | 2 |
PLK1 | 89 | 10 |
PRAK | 94 | 2 |
PRK2 | 85 | 0 |
RIPK2 | 63 | 2 |
ROCK 2 | 86 | 3 |
RSK1 | 92 | 1 |
RSK2 | 79 | 8 |
S6K1 | 85 | 2 |
SGK1 | 96 | 6 |
SIK2 | 83 | 2 |
SIK3 | 76 | 4 |
SmMLCK | 82 | 8 |
Src | 85 | 0 |
SRPK1 | 84 | 8 |
STK33 | 87 | 6 |
SYK | 93 | 2 |
TAK1 | 83 | 3 |
TAO1 | 79 | 4 |
TBK1 | 81 | 0 |
TESK1 | 82 | 1 |
TGFBR1 | 80 | 9 |
TIE2 | 88 | 9 |
TLK1 | 98 | 5 |
TrkA | 90 | 9 |
TSSK1 | 90 | 8 |
TTBK1 | 86 | 2 |
TTBK2 | 80 | 13 |
TTK | 89 | 3 |
ULK1 | 74 | 10 |
ULK2 | 99 | 13 |
VEGFR1 | 83 | 9 |
WNK1 | 93 | 9 |
YES1 | 93 | 3 |
ZAP70 | 92 | 3 |