Inhibitor | Lenalidomide (Revlimid)  

Screen Conc: 1.00µM

Kinase	% Activity Remaining	Standard Deviation
ABL	96	14
AMPK	98	1
AMPK (hum)	106	0
ASK1	102	12
Aurora A	113	18
Aurora B	83	5
BRK	101	26
BRSK1	84	5
BRSK2	98	5
BTK	104	12
CAMK1	103	2
CAMKK beta	92	7
CDK2-Cyclin A	96	7
CDK9-Cyclin T1	106	52
CHK1	94	3
CHK2	96	12
CK1 delta	102	2
CK1 gamma 2	99	7
CK2	106	5
CLK2	104	12
CSK	87	7
DAPK1	95	12
DDR2	102	17
DYRK1A	107	1
DYRK2	101	9
DYRK3	104	8
EF2K	94	7
EIF2AK3	86	8
EPH-A2	106	35
EPH-A4	110	9
EPH-B1	115	7
EPH-B2	107	15
EPH-B3	98	21
EPH-B4	91	7
ERK1	90	10
ERK2	104	27
ERK5	98	9
ERK8	92	9
FGF-R1	110	21
GCK	103	15
GSK3 beta	104	20
HER4	105	36
HIPK1	92	7
HIPK2	107	3
HIPK3	108	35
IGF-1R	106	14
IKK beta	100	7
IKK epsilon	119	1
IR	103	29
IRAK1	96	0
IRAK4	107	4
IRR	102	14
JAK2	103	3
JNK1	99	11
JNK2	100	16
JNK3	90	0
Lck	100	6
LKB1	116	2
MAP4K3	100	9
MAP4K5	109	2
MAPKAP-K2	79	13
MAPKAP-K3	94	5
MARK1	98	6
MARK2	99	0
MARK3	91	11
MARK4	86	22
MEKK1	101	15
MELK	94	3
MINK1	111	6
MKK1	90	7
MKK2	83	2
MKK6	93	2
MLK1	99	3
MLK3	92	17
MNK1	116	7
MNK2	80	2
MPSK1	98	5
MSK1	91	9
MST2	102	7
MST3	82	10
MST4	106	3
NEK2a	97	18
NEK6	105	13
NUAK1	99	5
OSR1	91	2
p38 alpha MAPK	105	4
p38 beta MAPK	96	6
p38 delta MAPK	109	11
p38 gamma MAPK	109	8
PAK2	101	6
PAK4	102	0
PAK5	86	7
PAK6	102	12
PDGFRA	85	4
PDK1	91	21
PHK	101	2
PIM1	93	7
PIM2	98	9
PIM3	101	9
PKA	101	16
PKB alpha	88	3
PKB beta	85	9
PKC alpha	107	1
PKC gamma	108	4
PKC zeta	100	16
PKD1	103	7
PLK1	104	8
PRAK	86	12
PRK2	93	8
RIPK2	97	2
ROCK 2	90	8
RSK1	98	1
RSK2	93	2
S6K1	94	10
SGK1	91	10
SIK2	83	9
SIK3	91	7
SmMLCK	94	9
Src	105	17
SRPK1	104	5
STK33	128	18
SYK	108	25
TAK1	99	5
TAO1	106	7
TBK1	95	6
TESK1	77	6
TGFBR1	105	19
TIE2	85	23
TLK1	95	9
TrkA	116	22
TSSK1	89	17
TTBK1	106	18
TTBK2	93	25
TTK	104	5
ULK1	104	2
ULK2	106	12
VEGFR1	100	1
WNK1	104	5
YES1	102	14
ZAP70	110	18

Screen Conc: 10.00µM

Kinase	% Activity Remaining	Standard Deviation
ABL	101	10
AMPK	92	5
AMPK (hum)	102	3
ASK1	101	3
Aurora A	100	16
Aurora B	105	9
BRK	114	7
BRSK1	94	10
BRSK2	105	7
BTK	107	12
CAMK1	91	12
CAMKK beta	84	8
CDK2-Cyclin A	87	2
CDK9-Cyclin T1	119	21
CHK1	82	4
CHK2	93	6
CK1 delta	97	4
CK1 gamma 2	90	1
CK2	93	7
CLK2	98	2
CSK	97	3
DAPK1	104	12
DDR2	102	4
DYRK1A	99	11
DYRK2	103	14
DYRK3	99	2
EF2K	82	5
EIF2AK3	101	2
EPH-A2	96	11
EPH-A4	124	6
EPH-B1	126	12
EPH-B2	113	18
EPH-B3	102	16
EPH-B4	99	15
ERK1	94	5
ERK2	101	25
ERK5	107	19
ERK8	98	3
FGF-R1	109	6
GCK	114	0
GSK3 beta	92	15
HER4	106	6
HIPK1	101	10
HIPK2	103	16
HIPK3	119	27
IGF-1R	106	8
IKK beta	106	4
IKK epsilon	99	2
IR	107	11
IRAK1	101	19
IRAK4	110	10
IRR	109	8
JAK2	93	7
JNK1	106	9
JNK2	102	9
JNK3	95	7
Lck	99	1
LKB1	112	7
MAP4K3	110	12
MAP4K5	115	6
MAPKAP-K2	92	16
MAPKAP-K3	86	2
MARK1	100	0
MARK2	104	17
MARK3	94	0
MARK4	90	19
MEKK1	97	5
MELK	90	2
MINK1	118	2
MKK1	92	1
MKK2	81	10
MKK6	100	19
MLK1	99	2
MLK3	98	9
MNK1	111	10
MNK2	89	1
MPSK1	100	3
MSK1	94	24
MST2	101	1
MST3	84	9
MST4	112	12
NEK2a	96	15
NEK6	96	8
NUAK1	90	22
OSR1	112	4
p38 alpha MAPK	103	9
p38 beta MAPK	106	3
p38 delta MAPK	123	6
p38 gamma MAPK	108	10
PAK2	103	11
PAK4	107	8
PAK5	77	15
PAK6	104	3
PDGFRA	82	2
PDK1	89	7
PHK	103	3
PIM1	87	1
PIM2	99	21
PIM3	103	12
PKA	84	3
PKB alpha	91	12
PKB beta	94	7
PKC alpha	100	7
PKC gamma	112	6
PKC zeta	108	15
PKD1	114	18
PLK1	96	16
PRAK	87	10
PRK2	88	8
RIPK2	106	0
ROCK 2	88	5
RSK1	97	4
RSK2	101	8
S6K1	93	0
SGK1	96	23
SIK2	91	0
SIK3	94	10
SmMLCK	94	6
Src	114	8
SRPK1	104	8
STK33	119	11
SYK	114	17
TAK1	104	9
TAO1	96	0
TBK1	102	7
TESK1	77	4
TGFBR1	115	5
TIE2	90	39
TLK1	106	13
TrkA	141	7
TSSK1	100	14
TTBK1	118	14
TTBK2	101	8
TTK	118	14
ULK1	103	3
ULK2	105	0
VEGFR1	110	12
WNK1	106	3
YES1	102	11
ZAP70	116	3