Compound name | Brutto | MW | CAS | PubChem CID | Action | Reference | Reference |
---|---|---|---|---|---|---|---|
BAY 61-3606 | C20H18N6O3 · xHCl · yH2O | 390.40 | 732983-37-8 | 10200390 | Syk | Yamamoto N. (2003) J. Pharmacol. Exp. Ther. 306 1174-1181 |
Kinase | % Activity Remaining Sort descending | Standard Deviation |
---|---|---|
NUAK1 |
1
|
0 |
GCK |
5
|
1 |
IGF-1R |
6
|
1 |
CLK2 | 12 | 2 |
IR | 13 | 1 |
TAK1 | 14 | 0 |
ROCK 2 | 14 | 1 |
GSK3 beta | 16 | 2 |
CDK9-Cyclin T1 | 21 | 9 |
PRK2 | 21 | 3 |
MLK3 | 22 | 4 |
CDK2-Cyclin A | 23 | 1 |
HIPK2 | 24 | 8 |
DYRK3 | 24 | 4 |
IRR | 25 | 4 |
MAP4K3 | 29 | 4 |
RIPK2 | 29 | 1 |
PKD1 | 29 | 6 |
IRAK1 | 31 | 3 |
SYK | 32 | 1 |
MLK1 | 33 | 3 |
DYRK2 | 36 | 2 |
PDGFRA | 38 | 5 |
ERK8 | 39 | 7 |
CAMKK beta | 43 | 3 |
MARK3 | 44 | 2 |
PIM3 | 45 | 2 |
BTK | 46 | 1 |
PKC alpha | 46 | 1 |
Aurora B | 48 | 1 |
VEGFR1 | 50 | 9 |
YES1 | 51 | 15 |
MAP4K5 | 52 | 0 |
MKK6 | 55 | 2 |
IKK beta | 55 | 2 |
MST2 | 55 | 3 |
MNK2 | 56 | 1 |
HIPK1 | 56 | 6 |
DYRK1A | 58 | 1 |
JAK2 | 58 | 7 |
LKB1 | 59 | 0 |
AMPK (hum) | 59 | 35 |
MINK1 | 59 | 4 |
IKK epsilon | 60 | 9 |
JNK3 | 62 | 5 |
Src | 63 | 6 |
ERK2 | 65 | 7 |
STK33 | 66 | 2 |
ERK5 | 67 | 4 |
FGF-R1 | 67 | 15 |
IRAK4 | 68 | 8 |
ULK1 | 68 | 5 |
PIM1 | 69 | 1 |
TAO1 | 69 | 5 |
MARK2 | 69 | 10 |
ERK1 | 71 | 12 |
TTK | 71 | 1 |
PAK5 | 71 | 3 |
MELK | 71 | 6 |
SIK2 | 72 | 2 |
BRK | 73 | 14 |
MNK1 | 73 | 0 |
HIPK3 | 73 | 4 |
DAPK1 | 74 | 1 |
MARK4 | 74 | 12 |
CK1 delta | 75 | 2 |
S6K1 | 75 | 7 |
JNK2 | 75 | 9 |
PAK4 | 75 | 12 |
EPH-A2 | 76 | 5 |
Lck | 76 | 1 |
ASK1 | 77 | 0 |
MST4 | 78 | 16 |
EPH-A4 | 78 | 1 |
BRSK2 | 78 | 12 |
TBK1 | 78 | 8 |
SIK3 | 79 | 2 |
PKB beta | 79 | 15 |
MST3 | 79 | 1 |
PHK | 80 | 4 |
PAK6 | 80 | 9 |
MSK1 | 81 | 4 |
PIM2 | 81 | 10 |
RSK1 | 82 | 7 |
SRPK1 | 82 | 3 |
MAPKAP-K3 | 82 | 5 |
EIF2AK3 | 82 | 1 |
NEK2a | 82 | 7 |
NEK6 | 82 | 10 |
MEKK1 | 82 | 2 |
ZAP70 | 82 | 5 |
MKK2 | 83 | 18 |
CHK2 | 83 | 5 |
TESK1 | 84 | 2 |
HER4 | 84 | 4 |
p38 beta MAPK | 84 | 11 |
p38 gamma MAPK | 84 | 13 |
p38 delta MAPK | 85 | 3 |
PKC zeta | 85 | 7 |
PLK1 | 86 | 12 |
EPH-B1 | 86 | 2 |
EPH-B2 | 86 | 3 |
BRSK1 | 86 | 2 |
TTBK1 | 87 | 10 |
CSK | 88 | 9 |
TSSK1 | 88 | 14 |
OSR1 | 89 | 11 |
SGK1 | 89 | 6 |
MARK1 | 89 | 5 |
EF2K | 90 | 3 |
ABL | 91 | 9 |
ULK2 | 91 | 14 |
MKK1 | 92 | 10 |
TrkA | 92 | 47 |
DDR2 | 92 | 9 |
CK1 gamma 2 | 93 | 11 |
TLK1 | 93 | 4 |
CK2 | 93 | 9 |
EPH-B4 | 93 | 2 |
PDK1 | 94 | 17 |
SmMLCK | 94 | 16 |
JNK1 | 94 | 3 |
TGFBR1 | 94 | 2 |
WNK1 | 96 | 7 |
TTBK2 | 98 | 2 |
PKA | 99 | 12 |
EPH-B3 | 99 | 8 |
CAMK1 | 100 | 11 |
AMPK | 101 | 2 |
PAK2 | 102 | 6 |
PRAK | 103 | 18 |
MPSK1 | 103 | 13 |
PKC gamma | 103 | 12 |
PKB alpha | 106 | 12 |
p38 alpha MAPK | 107 | 10 |
CHK1 | 108 | 12 |
RSK2 | 113 | 12 |
TIE2 | 113 | 2 |
Aurora A | 114 | 17 |
MAPKAP-K2 | 146 | 51 |
Kinase | % Activity Remaining Sort descending | Standard Deviation |
---|---|---|
GCK |
4
|
1 |
IGF-1R |
10
|
4 |
CLK2 | 14 | 1 |
GSK3 beta | 15 | 5 |
IR | 16 | 1 |
TAK1 | 16 | 1 |
ROCK 2 | 18 | 0 |
MLK3 | 20 | 1 |
DYRK3 | 24 | 2 |
CDK2-Cyclin A | 25 | 3 |
HIPK2 | 25 | 1 |
NUAK1 | 26 | 1 |
CDK9-Cyclin T1 | 26 | 7 |
PKD1 | 27 | 1 |
IRR | 29 | 2 |
IRAK1 | 31 | 0 |
RIPK2 | 32 | 0 |
PRK2 | 32 | 3 |
MAP4K3 | 34 | 4 |
SYK | 36 | 2 |
MLK1 | 36 | 2 |
CAMKK beta | 37 | 8 |
PDGFRA | 40 | 1 |
Aurora B | 40 | 3 |
DYRK2 | 40 | 0 |
MARK3 | 49 | 7 |
MST2 | 50 | 8 |
LKB1 | 50 | 5 |
IKK epsilon | 51 | 1 |
DYRK1A | 51 | 0 |
Src | 54 | 12 |
ERK8 | 55 | 23 |
PKC alpha | 56 | 1 |
IKK beta | 56 | 4 |
MAP4K5 | 56 | 5 |
MARK2 | 56 | 5 |
PIM1 | 59 | 9 |
BTK | 59 | 1 |
MKK6 | 62 | 3 |
HIPK1 | 62 | 12 |
MELK | 63 | 13 |
YES1 | 63 | 15 |
MARK4 | 64 | 3 |
TSSK1 | 65 | 17 |
ERK5 | 67 | 1 |
CHK2 | 68 | 3 |
ERK2 | 68 | 7 |
JAK2 | 69 | 7 |
ERK1 | 69 | 7 |
MNK2 | 69 | 11 |
FGF-R1 | 69 | 11 |
PIM3 | 70 | 41 |
VEGFR1 | 71 | 15 |
p38 beta MAPK | 71 | 2 |
EF2K | 71 | 1 |
HIPK3 | 71 | 2 |
CK1 delta | 72 | 4 |
JNK2 | 72 | 11 |
JNK3 | 73 | 11 |
ULK1 | 73 | 1 |
PAK5 | 74 | 2 |
TTK | 74 | 10 |
MSK1 | 74 | 5 |
Lck | 74 | 8 |
PAK4 | 74 | 7 |
MST3 | 75 | 10 |
STK33 | 75 | 5 |
SIK2 | 75 | 2 |
S6K1 | 75 | 4 |
TESK1 | 75 | 7 |
TAO1 | 75 | 2 |
PKC zeta | 76 | 5 |
p38 gamma MAPK | 76 | 8 |
BRSK2 | 77 | 10 |
DAPK1 | 77 | 9 |
IRAK4 | 78 | 9 |
EPH-B1 | 78 | 2 |
MINK1 | 78 | 7 |
ZAP70 | 79 | 7 |
PLK1 | 79 | 9 |
NEK2a | 79 | 7 |
TrkA | 80 | 30 |
MKK2 | 80 | 6 |
TLK1 | 80 | 12 |
SRPK1 | 81 | 1 |
MKK1 | 82 | 6 |
PAK6 | 82 | 3 |
ASK1 | 82 | 7 |
MST4 | 83 | 5 |
PIM2 | 83 | 9 |
MNK1 | 83 | 4 |
PKA | 84 | 2 |
PHK | 84 | 12 |
TBK1 | 85 | 13 |
JNK1 | 85 | 3 |
CSK | 85 | 8 |
p38 delta MAPK | 87 | 0 |
EPH-B2 | 87 | 1 |
AMPK | 87 | 3 |
EPH-A4 | 88 | 10 |
MEKK1 | 88 | 10 |
BRSK1 | 89 | 11 |
BRK | 89 | 1 |
EPH-B3 | 89 | 1 |
EPH-B4 | 89 | 8 |
AMPK (hum) | 89 | 12 |
MARK1 | 89 | 2 |
PAK2 | 89 | 1 |
SIK3 | 90 | 4 |
CHK1 | 91 | 18 |
PKB alpha | 92 | 6 |
CK1 gamma 2 | 92 | 4 |
DDR2 | 93 | 1 |
OSR1 | 93 | 13 |
TTBK1 | 93 | 19 |
PDK1 | 94 | 3 |
WNK1 | 95 | 9 |
MAPKAP-K3 | 95 | 21 |
EIF2AK3 | 95 | 2 |
EPH-A2 | 96 | 15 |
ULK2 | 96 | 4 |
CK2 | 96 | 9 |
MPSK1 | 98 | 24 |
TGFBR1 | 98 | 7 |
TTBK2 | 98 | 10 |
NEK6 | 99 | 17 |
PKC gamma | 99 | 4 |
MAPKAP-K2 | 99 | 4 |
SGK1 | 100 | 1 |
ABL | 100 | 6 |
PRAK | 101 | 7 |
CAMK1 | 101 | 3 |
RSK1 | 102 | 21 |
p38 alpha MAPK | 103 | 10 |
HER4 | 103 | 2 |
TIE2 | 105 | 0 |
PKB beta | 106 | 19 |
Aurora A | 110 | 12 |
SmMLCK | 111 | 10 |
RSK2 | 117 | 3 |