Compound name | Brutto | MW | CAS | PubChem CID | Action | Reference | Reference |
---|---|---|---|---|---|---|---|
JNKIN7 | C28H27N7O2 | 493.56 | JNK | Zhang T. (2012) Chem Biol. 19(1) 140-54 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
ABL | 77 | 9 |
AMPK | 92 | 12 |
ASK1 | 96 | 9 |
Aurora A | 107 | 7 |
Aurora B | 74 | 1 |
BRK | 81 | 11 |
BRSK1 | 94 | 4 |
BRSK2 | 82 | 8 |
BTK | 86 | 22 |
CAMK1 | 87 | 12 |
CAMKK beta | 87 | 10 |
CDK2-Cyclin A | 85 | 0 |
CDK9-Cyclin T1 | 22 | 4 |
CHK1 | 74 | 17 |
CHK2 | 89 | 2 |
CK1 delta | 63 | 5 |
CK1 gamma 2 | 88 | 1 |
CK2 | 80 | 1 |
CLK2 | 49 | 2 |
CSK | 109 | 20 |
DAPK1 | 90 | 8 |
DDR2 | 89 | 7 |
DYRK1A | 97 | 2 |
DYRK2 | 82 | 20 |
DYRK3 | 81 | 9 |
EF2K | 97 | 5 |
EIF2AK3 | 90 | 2 |
EPH-A2 | 110 | 7 |
EPH-A4 | 92 | 5 |
EPH-B1 | 93 | 9 |
EPH-B2 | 101 | 9 |
EPH-B3 | 101 | 6 |
EPH-B4 | 105 | 2 |
ERK1 | 110 | 16 |
ERK2 | 99 | 16 |
ERK8 | 46 | 5 |
FGF-R1 | 94 | 19 |
GCK | 45 | 4 |
GSK3 beta | 88 | 8 |
HER4 | 108 | 32 |
HIPK1 | 86 | 11 |
HIPK2 | 85 | 10 |
HIPK3 | 113 | 0 |
IGF-1R | 75 | 22 |
IKK beta | 76 | 16 |
IKK epsilon | 97 | 4 |
IR | 81 | 1 |
IRAK1 | 26 | 14 |
IRAK4 | 86 | 12 |
IRR | 72 | 1 |
JAK2 | 85 | 10 |
JNK1 |
9
|
2 |
JNK2 | 81 | 8 |
JNK3 | 15 | 2 |
Lck | 95 | 0 |
LKB1 | 78 | 3 |
MAPKAP-K2 | 91 | 1 |
MAPKAP-K3 | 104 | 9 |
MARK1 | 91 | 9 |
MARK2 | 94 | 1 |
MARK3 | 101 | 5 |
MARK4 | 85 | 3 |
MEKK1 | 85 | 11 |
MELK | 71 | 0 |
MINK1 | 92 | 9 |
MKK1 | 98 | 6 |
MKK2 | 87 | 19 |
MKK6 | 97 | 13 |
MLK1 | 72 | 0 |
MLK3 | 79 | 1 |
MNK1 | 84 | 16 |
MNK2 | 92 | 5 |
MPSK1 | 108 | 3 |
MSK1 | 88 | 9 |
MST2 | 83 | 10 |
MST3 | 94 | 3 |
MST4 | 98 | 2 |
NEK2a | 93 | 1 |
NEK6 | 88 | 12 |
NUAK1 | 35 | 1 |
OSR1 | 99 | 2 |
p38 alpha MAPK | 98 | 0 |
p38 beta MAPK | 96 | 5 |
p38 delta MAPK | 106 | 7 |
p38 gamma MAPK | 90 | 10 |
PAK2 | 102 | 2 |
PAK4 | 84 | 8 |
PAK5 | 89 | 1 |
PAK6 | 87 | 4 |
PDK1 | 89 | 14 |
PHK | 94 | 10 |
PIM1 | 97 | 3 |
PIM2 | 96 | 8 |
PIM3 | 97 | 6 |
PKA | 97 | 5 |
PKB alpha | 92 | 5 |
PKB beta | 93 | 13 |
PKC alpha | 89 | 4 |
PKC gamma | 96 | 4 |
PKC zeta | 112 | 3 |
PKD1 | 105 | 37 |
PLK1 | 91 | 9 |
PRAK | 96 | 17 |
PRK2 | 99 | 0 |
RIPK2 | 74 | 21 |
ROCK 2 | 89 | 10 |
RSK1 | 95 | 21 |
RSK2 | 80 | 11 |
S6K1 | 88 | 2 |
SGK1 | 105 | 20 |
SIK2 | 78 | 1 |
SIK3 | 81 | 4 |
SmMLCK | 96 | 6 |
Src | 93 | 9 |
SRPK1 | 105 | 16 |
STK33 | 92 | 8 |
SYK | 89 | 17 |
TAK1 | 67 | 4 |
TAO1 | 96 | 1 |
TBK1 | 77 | 5 |
TESK1 | 90 | 16 |
TIE2 | 94 | 5 |
TLK1 | 99 | 7 |
TrkA | 96 | 24 |
TSSK1 | 88 | 3 |
TTBK1 | 88 | 13 |
TTK | 83 | 6 |
ULK1 | 37 | 1 |
ULK2 | 50 | 5 |
VEGFR1 | 59 | 4 |
WNK1 | 103 | 17 |
YES1 | 80 | 17 |
ZAP70 | 82 | 1 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
ABL | 85 | 12 |
AMPK | 87 | 4 |
ASK1 | 100 | 1 |
Aurora A | 97 | 3 |
Aurora B | 73 | 1 |
BRK | 81 | 16 |
BRSK1 | 86 | 6 |
BRSK2 | 76 | 6 |
BTK | 85 | 14 |
CAMK1 | 92 | 4 |
CAMKK beta | 35 | 4 |
CDK2-Cyclin A | 72 | 2 |
CDK9-Cyclin T1 | 42 | 2 |
CHK1 | 88 | 2 |
CHK2 | 73 | 1 |
CK1 delta | 33 | 0 |
CK1 gamma 2 | 88 | 4 |
CK2 | 81 | 10 |
CLK2 | 18 | 5 |
CSK | 103 | 7 |
DAPK1 | 83 | 2 |
DDR2 | 108 | 9 |
DYRK1A | 85 | 6 |
DYRK2 | 56 | 2 |
DYRK3 | 79 | 6 |
EF2K | 101 | 1 |
EIF2AK3 | 99 | 9 |
EPH-A2 | 125 | 17 |
EPH-A4 | 105 | 2 |
EPH-B1 | 86 | 19 |
EPH-B2 | 103 | 10 |
EPH-B3 | 118 | 20 |
EPH-B4 | 109 | 6 |
ERK1 | 109 | 9 |
ERK2 | 114 | 17 |
ERK8 | 20 | 8 |
FGF-R1 | 95 | 14 |
GCK | 20 | 1 |
GSK3 beta | 56 | 1 |
HER4 | 106 | 7 |
HIPK1 | 78 | 10 |
HIPK2 | 46 | 4 |
HIPK3 | 101 | 22 |
IGF-1R | 102 | 8 |
IKK beta | 63 | 2 |
IKK epsilon | 98 | 8 |
IR | 77 | 24 |
IRAK1 |
5
|
0 |
IRAK4 | 88 | 6 |
IRR | 64 | 6 |
JAK2 | 77 | 8 |
JNK1 |
4
|
1 |
JNK2 | 19 | 9 |
JNK3 | 16 | 0 |
Lck | 101 | 1 |
LKB1 | 91 | 18 |
MAPKAP-K2 | 106 | 11 |
MAPKAP-K3 | 101 | 4 |
MARK1 | 80 | 1 |
MARK2 | 85 | 2 |
MARK3 | 76 | 2 |
MARK4 | 83 | 16 |
MEKK1 | 100 | 8 |
MELK | 48 | 1 |
MINK1 | 69 | 2 |
MKK1 | 113 | 9 |
MKK2 | 102 | 13 |
MKK6 | 91 | 0 |
MLK1 | 39 | 0 |
MLK3 | 59 | 8 |
MNK1 | 95 | 23 |
MNK2 | 84 | 21 |
MPSK1 | 103 | 8 |
MSK1 | 91 | 6 |
MST2 | 64 | 6 |
MST3 | 93 | 15 |
MST4 | 104 | 1 |
NEK2a | 105 | 21 |
NEK6 | 96 | 0 |
NUAK1 | 82 | 10 |
OSR1 | 105 | 7 |
p38 alpha MAPK | 113 | 3 |
p38 beta MAPK | 82 | 6 |
p38 delta MAPK | 100 | 4 |
p38 gamma MAPK | 103 | 0 |
PAK2 | 93 | 1 |
PAK4 | 66 | 6 |
PAK5 | 91 | 8 |
PAK6 | 103 | 8 |
PDK1 | 98 | 4 |
PHK | 83 | 0 |
PIM1 | 114 | 6 |
PIM2 | 102 | 8 |
PIM3 | 84 | 6 |
PKA | 108 | 15 |
PKB alpha | 104 | 5 |
PKB beta | 106 | 18 |
PKC alpha | 97 | 8 |
PKC gamma | 101 | 5 |
PKC zeta | 103 | 4 |
PKD1 | 82 | 9 |
PLK1 | 106 | 1 |
PRAK | 85 | 8 |
PRK2 | 92 | 3 |
RIPK2 | 42 | 1 |
ROCK 2 | 71 | 2 |
RSK1 | 77 | 31 |
RSK2 | 80 | 4 |
S6K1 | 112 | 4 |
SGK1 | 105 | 9 |
SIK2 | 67 | 7 |
SIK3 | 64 | 12 |
SmMLCK | 85 | 1 |
Src | 72 | 10 |
SRPK1 | 104 | 4 |
STK33 | 91 | 12 |
SYK | 72 | 5 |
TAK1 | 39 | 1 |
TAO1 | 95 | 20 |
TBK1 | 79 | 11 |
TESK1 | 98 | 10 |
TIE2 | 84 | 15 |
TLK1 | 98 | 8 |
TrkA | 82 | 11 |
TSSK1 | 101 | 7 |
TTBK1 | 79 | 8 |
TTK | 77 | 3 |
ULK1 | 63 | 13 |
ULK2 | 69 | 7 |
VEGFR1 | 32 | 2 |
WNK1 | 117 | 8 |
YES1 | 58 | 4 |
ZAP70 | 123 | 1 |