Inhibitor | AZD8055  

Screen Conc: 1.00µM

Kinase	% Activity Remaining Sort descending	Standard Deviation
MARK3	53	72
VEGFR1	76	5
PKB beta	80	10
SRPK1	81	7
BTK	83	10
DYRK1A	83	14
CAMK1	84	5
JNK2	84	3
RSK2	84	7
EPH-B3	85	5
PAK6	86	7
GSK3 beta	87	12
p38 alpha MAPK	87	0
PAK5	87	1
Lck	88	6
CHK2	88	7
PKC zeta	88	2
RSK1	88	16
ERK1	89	21
PKA	89	8
p38 beta MAPK	89	11
p38 delta MAPK	89	20
CAMKK beta	90	5
IKK beta	91	12
PRK2	91	15
MSK1	91	7
PRAK	91	16
SmMLCK	92	10
EPH-A2	92	11
ERK2	92	17
PKB alpha	93	8
PHK	94	15
IRR	94	12
BRSK2	94	16
IR	94	21
PIM3	95	9
YES1	95	4
CK1 delta	96	6
MAPKAP-K2	96	3
PDK1	98	10
PIM2	98	10
DYRK3	99	9
PIM1	99	4
SYK	99	9
JNK1	99	6
PLK1	99	2
MELK	99	27
NEK2a	100	7
AMPK	100	10
EF2K	100	25
CSK	101	14
CHK1	101	15
MST4	101	10
PKC alpha	101	5
CDK2-Cyclin A	102	7
MNK1	102	14
ERK8	102	14
MNK2	102	3
DYRK2	103	15
MKK1	104	6
S6K1	105	13
p38 gamma MAPK	105	0
HIPK2	105	13
Src	105	13
MST2	106	10
IKK epsilon	107	0
IGF-1R	107	2
PAK4	108	17
SGK1	110	10
CK2	113	2
TBK1	116	9
FGF-R1	122	2
PKD1	124	3
ROCK 2	128	31
NEK6	130	41

Screen Conc: 0.10µM

Kinase	% Activity Remaining Sort descending	Standard Deviation
CAMK1	76	0
VEGFR1	80	7
ERK2	80	1
PAK6	80	1
p38 alpha MAPK	80	2
PKA	81	3
RSK2	81	3
JNK2	82	8
Lck	82	4
IR	83	9
DYRK1A	84	11
SRPK1	84	9
PKB beta	84	10
NEK6	86	13
MNK2	86	4
BRSK2	87	15
MST4	87	9
BTK	89	1
EPH-B3	89	14
RSK1	90	4
CHK1	90	3
ERK1	91	11
MELK	91	18
DYRK3	91	5
MSK1	91	14
EF2K	91	16
CK1 delta	92	11
IRR	92	1
CSK	93	5
IKK beta	93	1
EPH-A2	93	2
PRAK	93	0
SmMLCK	93	2
PHK	93	6
PAK5	94	10
JNK1	94	5
p38 gamma MAPK	94	15
p38 delta MAPK	94	15
GSK3 beta	94	13
PKB alpha	94	3
PKC zeta	95	4
NEK2a	96	11
SYK	96	2
PKC alpha	97	2
PIM3	97	4
MAPKAP-K2	98	6
PDK1	98	7
CAMKK beta	98	13
PLK1	98	12
AMPK	98	4
MST2	98	2
PIM1	99	16
CDK2-Cyclin A	100	1
CHK2	102	12
PRK2	102	11
Src	102	8
PIM2	103	13
TBK1	104	8
MARK3	104	6
YES1	105	5
ROCK 2	106	5
p38 beta MAPK	106	5
S6K1	106	6
DYRK2	107	2
PAK4	108	9
PKD1	111	7
ERK8	111	7
CK2	112	12
MKK1	112	16
HIPK2	118	9
IKK epsilon	118	0
SGK1	118	13
FGF-R1	129	4
IGF-1R	131	3
MNK1	132	20