Compound name | Brutto | MW | CAS | PubChem CID | Action | Reference | Reference |
---|---|---|---|---|---|---|---|
BI 2536 | C28H39N7O3 | 521.65 | 755038-02-9 | 11364421 | PLK1 | Steegmaier M. (2007) Current Biology 17 316-322 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
ABL | 104 | 4 |
AMPK | 95 | 6 |
ASK1 | 93 | 8 |
Aurora A | 100 | 2 |
Aurora B | 80 | 11 |
Aurora C | 116 | 3 |
BRK | 124 | 1 |
BRSK1 | 109 | 1 |
BRSK2 | 93 | 5 |
BTK | 85 | 8 |
CAMK1 | 99 | 6 |
CAMKK beta | 24 | 6 |
CDK2-Cyclin A | 90 | 2 |
CDK9-Cyclin T1 | 95 | 6 |
CHK1 | 105 | 12 |
CHK2 | 90 | 4 |
CK1 delta | 76 | 3 |
CK1 gamma 2 | 76 | 13 |
CK2 | 88 | 1 |
CLK2 | 64 | 10 |
CSK | 91 | 11 |
DAPK1 | 88 | 6 |
DDR2 | 100 | 2 |
DYRK1A | 102 | 4 |
DYRK2 | 97 | 4 |
DYRK3 | 94 | 9 |
EF2K | 89 | 8 |
EIF2AK3 | 64 | 3 |
EPH-A2 | 96 | 9 |
EPH-A4 | 115 | 1 |
EPH-B1 | 88 | 1 |
EPH-B2 | 110 | 7 |
EPH-B3 | 115 | 1 |
EPH-B4 | 106 | 9 |
ERK1 | 92 | 6 |
ERK2 | 94 | 8 |
ERK8 | 107 | 2 |
FGF-R1 | 108 | 6 |
GCK | 95 | 9 |
GSK3 beta | 84 | 1 |
HER4 | 107 | 8 |
HIPK1 | 104 | 4 |
HIPK2 | 93 | 3 |
HIPK3 | 97 | 9 |
IGF-1R | 73 | 6 |
IKK beta | 92 | 9 |
IKK epsilon | 91 | 4 |
IR | 79 | 6 |
IRAK1 | 99 | 3 |
IRAK4 | 88 | 5 |
IRR | 105 | 5 |
JAK2 | 106 | 11 |
JNK1 | 85 | 6 |
JNK2 | 94 | 1 |
JNK3 | 96 | 2 |
Lck | 108 | 8 |
LKB1 | 94 | 10 |
MAPKAP-K2 | 92 | 7 |
MAPKAP-K3 | 99 | 13 |
MARK1 | 90 | 6 |
MARK2 | 93 | 3 |
MARK3 | 82 | 1 |
MARK4 | 93 | 3 |
MEKK1 | 94 | 19 |
MELK | 78 | 6 |
MINK1 | 85 | 2 |
MKK1 | 95 | 8 |
MKK2 | 93 | 10 |
MKK6 | 99 | 11 |
MLK1 | 99 | 6 |
MLK3 | 89 | 6 |
MNK1 | 112 | 2 |
MNK2 | 93 | 9 |
MPSK1 | 96 | 9 |
MSK1 | 96 | 13 |
MST2 | 81 | 0 |
MST3 | 109 | 19 |
MST4 | 83 | 10 |
NEK2a | 90 | 10 |
NEK6 | 107 | 1 |
NUAK1 | 97 | 5 |
OSR1 | 104 | 7 |
p38 alpha MAPK | 102 | 6 |
p38 beta MAPK | 109 | 3 |
p38 delta MAPK | 99 | 1 |
p38 gamma MAPK | 99 | 6 |
PAK2 | 85 | 4 |
PAK4 | 86 | 1 |
PAK5 | 93 | 5 |
PAK6 | 98 | 12 |
PDK1 | 103 | 11 |
PHK | 89 | 2 |
PIM1 | 85 | 10 |
PIM2 | 97 | 1 |
PIM3 | 103 | 12 |
PKA | 98 | 7 |
PKB alpha | 103 | 4 |
PKB beta | 97 | 5 |
PKC alpha | 113 | 5 |
PKC gamma | 107 | 8 |
PKC zeta | 104 | 0 |
PKD1 | 90 | 12 |
PLK1 |
6
|
1 |
PRAK | 96 | 4 |
PRK2 | 94 | 2 |
RIPK2 | 98 | 12 |
ROCK 2 | 83 | 3 |
RSK1 | 95 | 1 |
RSK2 | 104 | 3 |
S6K1 | 94 | 14 |
SGK1 | 101 | 4 |
SIK2 | 83 | 9 |
SIK3 | 88 | 4 |
SmMLCK | 69 | 0 |
Src | 93 | 5 |
SRPK1 | 92 | 10 |
STK33 | 97 | 9 |
SYK | 80 | 11 |
TAK1 | 83 | 0 |
TAO1 | 92 | 1 |
TBK1 | 106 | 1 |
TESK1 | 91 | 6 |
TIE2 | 98 | 4 |
TLK1 | 100 | 1 |
TrkA | 110 | 14 |
TSSK1 | 87 | 5 |
TTBK1 | 95 | 5 |
TTK | 93 | 1 |
VEGFR1 | 103 | 1 |
WNK1 | 98 | 7 |
YES1 | 109 | 0 |
ZAP70 | 92 | 1 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
ABL | 97 | 9 |
AMPK | 97 | 7 |
ASK1 | 120 | 12 |
Aurora A | 119 | 11 |
Aurora B | 73 | 1 |
BRK | 118 | 5 |
BRSK1 | 102 | 10 |
BRSK2 | 92 | 2 |
BTK | 102 | 6 |
CAMK1 | 89 | 3 |
CAMKK beta | 16 | 4 |
CDK2-Cyclin A | 103 | 2 |
CDK9-Cyclin T1 | 84 | 1 |
CHK1 | 98 | 9 |
CHK2 | 58 | 4 |
CK1 delta | 88 | 10 |
CK1 gamma 2 | 89 | 3 |
CK2 | 99 | 4 |
CLK2 | 21 | 1 |
CSK | 101 | 2 |
DAPK1 | 60 | 2 |
DDR2 | 104 | 2 |
DYRK1A | 89 | 8 |
DYRK2 | 92 | 6 |
DYRK3 | 94 | 4 |
EF2K | 100 | 2 |
EIF2AK3 | 24 | 0 |
EPH-A2 | 88 | 7 |
EPH-A4 | 91 | 3 |
EPH-B1 | 100 | 1 |
EPH-B2 | 140 | 21 |
EPH-B3 | 114 | 2 |
EPH-B4 | 102 | 4 |
ERK1 | 103 | 3 |
ERK2 | 94 | 3 |
ERK8 | 109 | 15 |
FGF-R1 | 115 | 2 |
GCK | 92 | 2 |
GSK3 beta | 90 | 4 |
HER4 | 105 | 8 |
HIPK1 | 109 | 0 |
HIPK2 | 94 | 5 |
HIPK3 | 100 | 7 |
IGF-1R | 86 | 7 |
IKK beta | 92 | 4 |
IKK epsilon | 99 | 2 |
IR | 61 | 4 |
IRAK1 | 96 | 5 |
IRAK4 | 79 | 2 |
IRR | 85 | 7 |
JAK2 | 92 | 3 |
JNK1 | 93 | 1 |
JNK2 | 93 | 10 |
JNK3 | 90 | 0 |
Lck | 88 | 6 |
LKB1 | 85 | 2 |
MAPKAP-K2 | 90 | 2 |
MAPKAP-K3 | 98 | 8 |
MARK1 | 98 | 2 |
MARK2 | 93 | 5 |
MARK3 | 92 | 1 |
MARK4 | 83 | 9 |
MEKK1 | 90 | 5 |
MELK | 48 | 1 |
MINK1 | 77 | 1 |
MKK1 | 99 | 13 |
MKK2 | 104 | 0 |
MKK6 | 83 | 1 |
MLK1 | 94 | 2 |
MLK3 | 86 | 5 |
MNK1 | 112 | 2 |
MNK2 | 92 | 7 |
MPSK1 | 93 | 10 |
MSK1 | 105 | 1 |
MST2 | 91 | 1 |
MST3 | 93 | 15 |
MST4 | 88 | 8 |
NEK2a | 62 | 1 |
NEK6 | 85 | 10 |
NUAK1 | 75 | 1 |
OSR1 | 73 | 2 |
p38 alpha MAPK | 94 | 12 |
p38 beta MAPK | 106 | 12 |
p38 delta MAPK | 100 | 15 |
p38 gamma MAPK | 104 | 3 |
PAK2 | 92 | 8 |
PAK4 | 95 | 2 |
PAK5 | 90 | 0 |
PAK6 | 94 | 13 |
PDK1 | 104 | 10 |
PHK | 80 | 3 |
PIM1 | 102 | 4 |
PIM2 | 105 | 11 |
PIM3 | 98 | 2 |
PKA | 101 | 3 |
PKB alpha | 106 | 4 |
PKB beta | 90 | 6 |
PKC alpha | 117 | 10 |
PKC gamma | 106 | 4 |
PKC zeta | 109 | 8 |
PKD1 | 48 | 2 |
PLK1 |
6
|
1 |
PRAK | 97 | 15 |
PRK2 | 85 | 7 |
RIPK2 | 99 | 8 |
ROCK 2 | 89 | 4 |
RSK1 | 73 | 6 |
RSK2 | 69 | 4 |
S6K1 | 106 | 4 |
SGK1 | 108 | 5 |
SIK2 | 111 | 7 |
SIK3 | 82 | 5 |
SmMLCK | 23 | 0 |
Src | 79 | 5 |
SRPK1 | 77 | 11 |
STK33 | 78 | 18 |
SYK | 63 | 7 |
TAK1 | 80 | 3 |
TAO1 | 97 | 10 |
TBK1 | 82 | 2 |
TESK1 | 99 | 7 |
TIE2 | 93 | 11 |
TLK1 | 115 | 1 |
TrkA | 92 | 16 |
TSSK1 | 78 | 3 |
TTBK1 | 105 | 4 |
TTK | 96 | 3 |
VEGFR1 | 99 | 3 |
WNK1 | 100 | 4 |
YES1 | 109 | 7 |
ZAP70 | 94 | 0 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
AMPK | 86 | 3 |
Aurora B | 89 | 1 |
BRSK2 | 95 | 6 |
BTK | 93 | 8 |
CAMK1 | 47 | 1 |
CAMKK beta | 14 | 1 |
CDK2-Cyclin A | 75 | 7 |
CHK1 | 77 | 1 |
CHK2 | 26 | 3 |
CK1 delta | 27 | 0 |
CK2 | 78 | 3 |
CSK | 95 | 7 |
DYRK1A | 54 | 0 |
DYRK2 | 73 | 11 |
DYRK3 | 95 | 2 |
EF2K | 73 | 3 |
EPH-A2 | 76 | 7 |
EPH-B3 | 82 | 5 |
ERK1 | 74 | 2 |
ERK2 | 92 | 11 |
ERK8 | 115 | 6 |
FGF-R1 | 81 | 5 |
GCK | 67 | 4 |
GSK3 beta | 101 | 14 |
HER4 | 77 | 1 |
HIPK2 | 36 | 1 |
IGF-1R | 19 | 2 |
IKK beta | 76 | 3 |
IKK epsilon | 94 | 5 |
IR | 66 | 1 |
IRAK4 | 44 | 3 |
IRR | 70 | 0 |
JNK1 | 84 | 5 |
JNK2 | 84 | 1 |
Lck | 39 | 4 |
LKB1 | 83 | 7 |
MAPKAP-K2 | 74 | 4 |
MARK3 | 106 | 4 |
MELK |
9
|
2 |
MINK1 | 55 | 3 |
MKK1 | 72 | 6 |
MLK1 | 80 | 16 |
MLK3 | 97 | 5 |
MNK1 | 91 | 9 |
MNK2 | 98 | 11 |
MSK1 | 85 | 0 |
MST2 | 102 | 5 |
MST4 | 100 | 5 |
NEK2a |
4
|
2 |
NEK6 | 43 | 3 |
NUAK1 | 116 | 10 |
p38 alpha MAPK | 90 | 1 |
p38 beta MAPK | 84 | 4 |
p38 delta MAPK | 96 | 4 |
p38 gamma MAPK | 101 | 13 |
PAK4 | 113 | 3 |
PAK5 | 95 | 7 |
PAK6 | 79 | 5 |
PDK1 | 91 | 6 |
PHK | 29 | 3 |
PIM1 | 92 | 4 |
PIM2 | 128 | 4 |
PIM3 | 74 | 1 |
PKA | 81 | 0 |
PKB alpha | 81 | 1 |
PKB beta | 85 | 2 |
PKC alpha | 83 | 2 |
PKC zeta | 95 | 12 |
PKD1 |
10
|
1 |
PLK1 |
7
|
1 |
PRAK | 93 | 4 |
PRK2 | 95 | 4 |
ROCK 2 | 89 | 3 |
RSK1 | 30 | 4 |
RSK2 | 27 | 5 |
S6K1 | 77 | 10 |
SGK1 | 84 | 3 |
SmMLCK | 14 | 3 |
Src | 80 | 1 |
SRPK1 | 66 | 1 |
SYK | 54 | 4 |
TBK1 | 90 | 1 |
TTK | 66 | 21 |
VEGFR1 | 114 | 1 |
YES1 | 68 | 7 |