Compound name | Brutto | MW | CAS | PubChem CID | Action | Reference | Reference |
---|---|---|---|---|---|---|---|
KU 55933 | C21H17NO3S2 | 395.49 | 587871-26-9 | 5278396 | ATM kinase | Hickson (2004) Cancer Res. 64 9152 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
AMPK | 111 | 9 |
Aurora A | 116 | 3 |
Aurora B | 94 | 7 |
BRSK1 | 99 | 10 |
BRSK2 | 117 | 3 |
BTK | 91 | 9 |
CAMK1 | 103 | 3 |
CAMKK beta | 128 | 16 |
CDK2-Cyclin A | 105 | 15 |
CHK1 | 92 | 1 |
CHK2 | 120 | 10 |
CK1 delta | 133 | 7 |
CK2 | 103 | 1 |
CSK | 142 | 12 |
DYRK1A | 98 | 0 |
DYRK2 | 93 | 2 |
DYRK3 | 61 | 2 |
EF2K | 99 | 12 |
EPH-A2 | 127 | 9 |
EPH-A4 | 114 | 1 |
EPH-B3 | 100 | 1 |
EPH-B4 | 125 | 5 |
ERK1 | 123 | 12 |
ERK2 | 109 | 8 |
ERK8 | 106 | 2 |
FGF-R1 | 121 | 2 |
GCK | 72 | 3 |
GSK3 beta | 108 | 12 |
HER4 | 118 | 1 |
HIPK1 | 118 | 9 |
HIPK2 | 108 | 5 |
HIPK3 | 119 | 20 |
IGF-1R | 101 | 2 |
IKK beta | 90 | 9 |
IKK epsilon | 81 | 2 |
IR | 107 | 3 |
IRAK4 | 66 | 7 |
IRR | 102 | 11 |
JAK2 | 117 | 6 |
JNK1 | 112 | 13 |
JNK2 | 113 | 5 |
JNK3 | 119 | 15 |
Lck | 109 | 4 |
LKB1 | 95 | 10 |
MAPKAP-K2 | 131 | 26 |
MAPKAP-K3 | 123 | 2 |
MARK1 | 87 | 14 |
MARK2 | 116 | 9 |
MARK3 | 82 | 7 |
MARK4 | 111 | 7 |
MEKK1 | 99 | 0 |
MELK | 81 | 4 |
MINK1 | 77 | 3 |
MKK1 | 90 | 9 |
MLK1 | 80 | 8 |
MLK3 | 56 | 6 |
MNK1 | 144 | 42 |
MNK2 | 146 | 29 |
MSK1 | 97 | 18 |
MST2 | 93 | 6 |
MST4 | 137 | 9 |
NEK2a | 101 | 6 |
NEK6 | 114 | 1 |
NUAK1 | 89 | 11 |
p38 alpha MAPK | 98 | 4 |
p38 beta MAPK | 108 | 7 |
p38 delta MAPK | 100 | 22 |
p38 gamma MAPK | 111 | 0 |
PAK2 | 124 | 4 |
PAK4 | 110 | 2 |
PAK5 | 129 | 2 |
PAK6 | 104 | 7 |
PDK1 | 134 | 3 |
PHK | 78 | 4 |
PIM1 | 106 | 4 |
PIM2 | 91 | 21 |
PIM3 | 101 | 2 |
PKA | 101 | 0 |
PKB alpha | 100 | 2 |
PKB beta | 107 | 14 |
PKC alpha | 119 | 10 |
PKC zeta | 112 | 3 |
PKD1 | 105 | 10 |
PLK1 | 120 | 3 |
PRAK | 126 | 18 |
PRK2 | 83 | 10 |
RIPK2 | 105 | 4 |
ROCK 2 | 111 | 5 |
RSK1 | 98 | 7 |
RSK2 | 112 | 5 |
S6K1 | 112 | 6 |
SGK1 | 116 | 9 |
SmMLCK | 116 | 7 |
Src | 98 | 1 |
SRPK1 | 107 | 6 |
SYK | 119 | 28 |
TAK1 | 109 | 8 |
TBK1 | 109 | 12 |
TrkA | 104 | 39 |
TTK | 117 | 8 |
VEGFR1 | 122 | 25 |
YES1 | 108 | 7 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
AMPK | 97 | 7 |
Aurora A | 121 | 1 |
Aurora B | 97 | 2 |
BRSK1 | 100 | 8 |
BRSK2 | 110 | 10 |
BTK | 86 | 5 |
CAMK1 | 92 | 1 |
CAMKK beta | 100 | 30 |
CDK2-Cyclin A | 102 | 3 |
CHK1 | 66 | 5 |
CHK2 | 87 | 5 |
CK1 delta | 93 | 5 |
CK2 | 94 | 2 |
CSK | 101 | 10 |
DYRK1A | 77 | 1 |
DYRK2 | 71 | 7 |
DYRK3 | 83 | 33 |
EF2K | 81 | 21 |
EPH-A2 | 82 | 18 |
EPH-A4 | 109 | 3 |
EPH-B3 | 86 | 4 |
EPH-B4 | 83 | 3 |
ERK1 | 105 | 4 |
ERK2 | 84 | 0 |
ERK8 | 101 | 2 |
FGF-R1 | 105 | 5 |
GCK | 62 | 1 |
GSK3 beta | 78 | 5 |
HER4 | 99 | 1 |
HIPK1 | 93 | 1 |
HIPK2 | 90 | 2 |
HIPK3 | 92 | 10 |
IGF-1R | 94 | 10 |
IKK beta | 65 | 2 |
IKK epsilon | 50 | 3 |
IR | 107 | 6 |
IRAK4 | 58 | 0 |
IRR | 78 | 10 |
JAK2 | 85 | 10 |
JNK1 | 96 | 4 |
JNK2 | 86 | 1 |
JNK3 | 91 | 2 |
Lck | 65 | 34 |
LKB1 | 94 | 6 |
MAPKAP-K2 | 112 | 5 |
MAPKAP-K3 | 86 | 3 |
MARK1 | 74 | 6 |
MARK2 | 91 | 0 |
MARK3 | 65 | 14 |
MARK4 | 77 | 3 |
MEKK1 | 67 | 19 |
MELK | 73 | 3 |
MINK1 | 69 | 7 |
MKK1 | 62 | 9 |
MLK1 | 66 | 10 |
MLK3 | 38 | 5 |
MNK1 | 113 | 8 |
MNK2 | 76 | 13 |
MSK1 | 70 | 8 |
MST2 | 66 | 8 |
MST4 | 111 | 16 |
NEK2a | 74 | 10 |
NEK6 | 78 | 11 |
NUAK1 | 89 | 1 |
p38 alpha MAPK | 67 | 10 |
p38 beta MAPK | 90 | 1 |
p38 delta MAPK | 83 | 20 |
p38 gamma MAPK | 91 | 2 |
PAK2 | 89 | 1 |
PAK4 | 90 | 13 |
PAK5 | 96 | 3 |
PAK6 | 82 | 12 |
PDK1 | 114 | 5 |
PHK | 61 | 0 |
PIM1 | 88 | 4 |
PIM2 | 82 | 2 |
PIM3 | 51 | 6 |
PKA | 90 | 10 |
PKB alpha | 65 | 5 |
PKB beta | 90 | 5 |
PKC alpha | 102 | 10 |
PKC zeta | 99 | 11 |
PKD1 | 88 | 12 |
PLK1 | 95 | 21 |
PRAK | 90 | 7 |
PRK2 | 73 | 1 |
RIPK2 | 96 | 1 |
ROCK 2 | 81 | 10 |
RSK1 | 78 | 2 |
RSK2 | 94 | 4 |
S6K1 | 91 | 4 |
SGK1 | 80 | 11 |
SmMLCK | 93 | 10 |
Src | 93 | 2 |
SRPK1 | 78 | 0 |
SYK | 108 | 23 |
TAK1 | 80 | 0 |
TBK1 | 90 | 8 |
TrkA | 78 | 12 |
TTK | 106 | 5 |
VEGFR1 | 92 | 15 |
YES1 | 103 | 11 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
AMPK | 96 | 5 |
ASK1 | 92 | 13 |
Aurora A | 109 | 3 |
Aurora B | 115 | 4 |
BRSK1 | 104 | 3 |
BRSK2 | 113 | 3 |
BTK | 97 | 3 |
CAMK1 | 103 | 5 |
CAMKK beta | 94 | 3 |
CDK2-Cyclin A | 98 | 8 |
CHK1 | 98 | 14 |
CHK2 | 123 | 10 |
CK1 delta | 112 | 4 |
CK2 | 101 | 10 |
CLK2 | 88 | 10 |
CSK | 93 | 1 |
DAPK1 | 81 | 8 |
DYRK1A | 66 | 3 |
DYRK2 | 93 | 1 |
DYRK3 | 84 | 3 |
EF2K | 66 | 5 |
EPH-A2 | 104 | 1 |
EPH-A4 | 101 | 8 |
EPH-B1 | 100 | 6 |
EPH-B2 | 107 | 1 |
EPH-B3 | 100 | 6 |
EPH-B4 | 106 | 2 |
ERK1 | 96 | 4 |
ERK2 | 100 | 8 |
ERK8 | 84 | 6 |
FGF-R1 | 97 | 12 |
GCK | 100 | 5 |
GSK3 beta | 66 | 2 |
HER4 | 83 | 7 |
HIPK1 | 97 | 6 |
HIPK2 | 83 | 4 |
HIPK3 | 109 | 7 |
IGF-1R | 74 | 3 |
IKK beta | 94 | 14 |
IKK epsilon | 88 | 1 |
IR | 100 | 4 |
IRAK4 | 73 | 7 |
IRR | 87 | 3 |
JAK2 | 89 | 3 |
JNK1 | 106 | 0 |
JNK2 | 103 | 5 |
JNK3 | 87 | 10 |
Lck | 109 | 2 |
LKB1 | 95 | 4 |
MAPKAP-K2 | 97 | 4 |
MAPKAP-K3 | 99 | 2 |
MARK1 | 99 | 6 |
MARK2 | 101 | 14 |
MARK3 | 107 | 3 |
MARK4 | 99 | 11 |
MEKK1 | 109 | 9 |
MELK | 87 | 6 |
MINK1 | 94 | 7 |
MKK1 | 81 | 7 |
MKK2 | 94 | 5 |
MKK6 | 104 | 3 |
MLK1 | 97 | 4 |
MLK3 | 99 | 5 |
MNK1 | 104 | 7 |
MNK2 | 88 | 7 |
MSK1 | 94 | 7 |
MST2 | 82 | 2 |
MST4 | 102 | 2 |
NEK2a | 105 | 7 |
NEK6 | 104 | 1 |
NUAK1 | 88 | 1 |
p38 alpha MAPK | 113 | 0 |
p38 beta MAPK | 96 | 8 |
p38 delta MAPK | 87 | 7 |
p38 gamma MAPK | 102 | 6 |
PAK2 | 91 | 12 |
PAK4 | 96 | 9 |
PAK5 | 100 | 1 |
PAK6 | 108 | 5 |
PDK1 | 88 | 3 |
PHK | 91 | 9 |
PIM1 | 56 | 12 |
PIM2 | 84 | 7 |
PIM3 | 31 | 1 |
PKA | 105 | 1 |
PKB alpha | 92 | 3 |
PKB beta | 90 | 14 |
PKC alpha | 104 | 2 |
PKC zeta | 104 | 8 |
PKD1 | 89 | 1 |
PLK1 | 89 | 7 |
PRAK | 85 | 2 |
PRK2 | 101 | 4 |
RIPK2 | 99 | 1 |
ROCK 2 | 96 | 4 |
RSK1 | 101 | 5 |
RSK2 | 101 | 7 |
S6K1 | 98 | 1 |
SGK1 | 103 | 7 |
SmMLCK | 96 | 3 |
Src | 99 | 5 |
SRPK1 | 106 | 12 |
SYK | 97 | 0 |
TAK1 | 113 | 1 |
TAO1 | 94 | 5 |
TBK1 | 105 | 12 |
TrkA | 95 | 3 |
TTK | 74 | 2 |
VEGFR1 | 96 | 8 |
YES1 | 96 | 8 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
AMPK | 88 | 8 |
ASK1 | 76 | 5 |
Aurora A | 94 | 8 |
Aurora B | 81 | 3 |
BRSK1 | 115 | 1 |
BRSK2 | 91 | 13 |
BTK | 62 | 1 |
CAMK1 | 64 | 6 |
CAMKK beta | 72 | 12 |
CDK2-Cyclin A | 61 | 8 |
CHK1 | 104 | 11 |
CHK2 | 97 | 9 |
CK1 delta | 97 | 11 |
CK2 | 92 | 3 |
CLK2 | 65 | 10 |
CSK | 90 | 3 |
DAPK1 | 84 | 3 |
DYRK1A | 19 | 1 |
DYRK2 | 86 | 9 |
DYRK3 | 78 | 4 |
EF2K | 43 | 3 |
EPH-A2 | 98 | 3 |
EPH-A4 | 95 | 11 |
EPH-B1 | 110 | 0 |
EPH-B2 | 108 | 3 |
EPH-B3 | 103 | 4 |
EPH-B4 | 129 | 5 |
ERK1 | 109 | 7 |
ERK2 | 101 | 0 |
ERK8 | 28 | 2 |
FGF-R1 | 94 | 10 |
GCK | 80 | 4 |
GSK3 beta | 26 | 0 |
HER4 | 91 | 1 |
HIPK1 | 82 | 3 |
HIPK2 | 52 | 8 |
HIPK3 | 78 | 0 |
IGF-1R | 63 | 11 |
IKK beta | 90 | 5 |
IKK epsilon | 84 | 1 |
IR | 102 | 13 |
IRAK4 | 79 | 10 |
IRR | 60 | 5 |
JAK2 | 95 | 1 |
JNK1 | 98 | 1 |
JNK2 | 94 | 0 |
JNK3 | 115 | 2 |
Lck | 94 | 11 |
LKB1 | 88 | 1 |
MAPKAP-K2 | 97 | 13 |
MAPKAP-K3 | 93 | 10 |
MARK1 | 104 | 12 |
MARK2 | 94 | 3 |
MARK3 | 82 | 2 |
MARK4 | 100 | 4 |
MEKK1 | 94 | 12 |
MELK | 82 | 7 |
MINK1 | 81 | 11 |
MKK1 | 59 | 2 |
MKK2 | 95 | 2 |
MKK6 | 118 | 13 |
MLK1 | 88 | 3 |
MLK3 | 90 | 7 |
MNK1 | 115 | 2 |
MNK2 | 89 | 3 |
MSK1 | 78 | 5 |
MST2 | 83 | 3 |
MST4 | 63 | 3 |
NEK2a | 85 | 6 |
NEK6 | 107 | 14 |
NUAK1 | 76 | 2 |
p38 alpha MAPK | 95 | 1 |
p38 beta MAPK | 120 | 3 |
p38 delta MAPK | 104 | 7 |
p38 gamma MAPK | 85 | 14 |
PAK2 | 90 | 1 |
PAK4 | 97 | 1 |
PAK5 | 67 | 11 |
PAK6 | 79 | 2 |
PDK1 | 92 | 4 |
PHK | 88 | 7 |
PIM1 | 13 | 0 |
PIM2 | 35 | 4 |
PIM3 | 19 | 0 |
PKA | 89 | 1 |
PKB alpha | 100 | 1 |
PKB beta | 61 | 8 |
PKC alpha | 73 | 2 |
PKC zeta | 87 | 11 |
PKD1 | 58 | 8 |
PLK1 | 78 | 1 |
PRAK | 43 | 0 |
PRK2 | 94 | 9 |
RIPK2 | 97 | 2 |
ROCK 2 | 83 | 2 |
RSK1 | 78 | 5 |
RSK2 | 84 | 13 |
S6K1 | 86 | 1 |
SGK1 | 106 | 1 |
SmMLCK | 51 | 2 |
Src | 110 | 15 |
SRPK1 | 98 | 7 |
SYK | 94 | 11 |
TAK1 | 63 | 4 |
TAO1 | 90 | 3 |
TBK1 | 78 | 2 |
TrkA | 97 | 2 |
TTK | 74 | 0 |
VEGFR1 | 80 | 6 |
YES1 | 112 | 9 |