Compound name | Brutto | MW | CAS | PubChem CID | Action | Reference | Reference |
---|---|---|---|---|---|---|---|
GSK2334470 | C25H34N8O | 462.59 | 1227911-45-6 | 46215815 | PDK1 | Najafov A. (2011) Biochem. J. 433 357-69 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
AMPK | 107 | 2 |
Aurora A | 112 | 7 |
Aurora B | 105 | 6 |
BRSK1 | 110 | 17 |
BRSK2 | 114 | 2 |
BTK | 126 | 9 |
CAMK1 | 108 | 3 |
CAMKK beta | 112 | 9 |
CDK2-Cyclin A | 104 | 3 |
CHK1 | 111 | 11 |
CHK2 | 129 | 25 |
CK1 delta | 100 | 1 |
CK2 | 103 | 0 |
CSK | 103 | 7 |
DYRK1A | 102 | 2 |
DYRK2 | 100 | 3 |
DYRK3 | 100 | 19 |
EF2K | 108 | 2 |
EPH-A2 | 110 | 4 |
EPH-B3 | 106 | 11 |
ERK1 | 93 | 5 |
ERK2 | 117 | 8 |
ERK8 | 106 | 12 |
FGF-R1 | 119 | 3 |
GCK | 109 | 3 |
GSK3 beta | 108 | 4 |
HER4 | 106 | 10 |
HIPK1 | 102 | 3 |
HIPK2 | 119 | 1 |
HIPK3 | 111 | 2 |
IGF-1R | 126 | 35 |
IKK beta | 105 | 3 |
IKK epsilon | 114 | 9 |
IR | 101 | 8 |
IRAK4 | 109 | 0 |
IRR | 111 | 4 |
JNK1 | 92 | 3 |
JNK2 | 117 | 6 |
JNK3 | 106 | 7 |
Lck | 112 | 18 |
LKB1 | 104 | 8 |
MAPKAP-K2 | 104 | 2 |
MAPKAP-K3 | 112 | 18 |
MARK2 | 113 | 1 |
MARK3 | 113 | 5 |
MARK4 | 106 | 7 |
MELK | 115 | 12 |
MINK1 | 121 | 4 |
MKK1 | 86 | 17 |
MLK1 | 110 | 1 |
MLK3 | 100 | 5 |
MNK1 | 106 | 14 |
MNK2 | 91 | 2 |
MSK1 | 102 | 0 |
MST2 | 116 | 4 |
MST4 | 112 | 7 |
NEK2a | 118 | 15 |
NEK6 | 98 | 6 |
NUAK1 | 120 | 19 |
p38 alpha MAPK | 105 | 5 |
p38 beta MAPK | 113 | 6 |
p38 delta MAPK | 106 | 2 |
p38 gamma MAPK | 109 | 6 |
PAK2 | 105 | 8 |
PAK4 | 108 | 1 |
PAK5 | 97 | 2 |
PAK6 | 108 | 7 |
PDK1 | 62 | 8 |
PHK | 106 | 8 |
PIM1 | 99 | 1 |
PIM2 | 97 | 7 |
PIM3 | 105 | 4 |
PKA | 103 | 13 |
PKB alpha | 179 | 71 |
PKB beta | 125 | 11 |
PKC alpha | 104 | 4 |
PKC zeta | 113 | 0 |
PKD1 | 99 | 5 |
PLK1 | 95 | 5 |
PRAK | 81 | 2 |
PRK2 | 90 | 10 |
RIPK2 | 110 | 1 |
ROCK 2 | 96 | 4 |
RSK1 | 123 | 12 |
RSK2 | 96 | 20 |
S6K1 | 111 | 4 |
SGK1 | 96 | 1 |
SmMLCK | 116 | 6 |
Src | 101 | 5 |
SRPK1 | 106 | 5 |
SYK | 109 | 14 |
TBK1 | 110 | 6 |
TTK | 90 | 1 |
VEGFR1 | 98 | 6 |
YES1 | 122 | 1 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
AMPK | 111 | 7 |
Aurora A | 115 | 4 |
Aurora B | 106 | 2 |
BRSK1 | 95 | 6 |
BRSK2 | 110 | 0 |
BTK | 121 | 15 |
CAMK1 | 112 | 3 |
CAMKK beta | 123 | 11 |
CDK2-Cyclin A | 101 | 11 |
CHK1 | 106 | 5 |
CHK2 | 121 | 5 |
CK1 delta | 108 | 6 |
CK2 | 104 | 12 |
CSK | 104 | 5 |
DYRK1A | 107 | 9 |
DYRK2 | 108 | 5 |
DYRK3 | 103 | 5 |
EF2K | 100 | 3 |
EPH-A2 | 118 | 12 |
EPH-B3 | 107 | 8 |
ERK1 | 106 | 12 |
ERK2 | 111 | 10 |
ERK8 | 117 | 7 |
FGF-R1 | 119 | 1 |
GCK | 116 | 14 |
GSK3 beta | 111 | 6 |
HER4 | 107 | 5 |
HIPK1 | 105 | 2 |
HIPK2 | 124 | 17 |
HIPK3 | 105 | 7 |
IGF-1R | 115 | 5 |
IKK beta | 112 | 7 |
IKK epsilon | 97 | 2 |
IR | 103 | 4 |
IRAK4 | 112 | 5 |
IRR | 111 | 8 |
JNK1 | 108 | 5 |
JNK2 | 126 | 19 |
JNK3 | 106 | 8 |
Lck | 107 | 3 |
LKB1 | 124 | 8 |
MAPKAP-K2 | 111 | 13 |
MAPKAP-K3 | 112 | 11 |
MARK2 | 114 | 0 |
MARK3 | 109 | 7 |
MARK4 | 114 | 6 |
MELK | 77 | 1 |
MINK1 | 110 | 8 |
MKK1 | 101 | 12 |
MLK1 | 111 | 1 |
MLK3 | 110 | 2 |
MNK1 | 108 | 5 |
MNK2 | 100 | 28 |
MSK1 | 100 | 2 |
MST2 | 128 | 11 |
MST4 | 108 | 14 |
NEK2a | 118 | 11 |
NEK6 | 101 | 6 |
NUAK1 | 105 | 3 |
p38 alpha MAPK | 109 | 8 |
p38 beta MAPK | 129 | 18 |
p38 delta MAPK | 113 | 12 |
p38 gamma MAPK | 110 | 5 |
PAK2 | 119 | 2 |
PAK4 | 117 | 16 |
PAK5 | 101 | 11 |
PAK6 | 120 | 17 |
PDK1 | 12 | 5 |
PHK | 108 | 3 |
PIM1 | 100 | 3 |
PIM2 | 100 | 28 |
PIM3 | 112 | 14 |
PKA | 111 | 15 |
PKB alpha | 117 | 22 |
PKB beta | 118 | 14 |
PKC alpha | 105 | 13 |
PKC zeta | 105 | 10 |
PKD1 | 116 | 0 |
PLK1 | 113 | 2 |
PRAK | 92 | 7 |
PRK2 | 102 | 12 |
RIPK2 | 114 | 15 |
ROCK 2 | 92 | 4 |
RSK1 | 113 | 3 |
RSK2 | 97 | 6 |
S6K1 | 106 | 16 |
SGK1 | 96 | 4 |
SmMLCK | 113 | 4 |
Src | 105 | 1 |
SRPK1 | 120 | 9 |
SYK | 105 | 4 |
TBK1 | 115 | 11 |
TTK | 98 | 10 |
VEGFR1 | 108 | 1 |
YES1 | 119 | 14 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
ABL | 116 | 7 |
AMPK | 91 | 1 |
ASK1 | 106 | 12 |
Aurora A | 98 | 3 |
Aurora B | 72 | 1 |
BRK | 127 | 9 |
BRSK1 | 53 | 1 |
BRSK2 | 62 | 3 |
BTK | 97 | 2 |
CAMK1 | 89 | 6 |
CAMKK beta | 99 | 9 |
CDK2-Cyclin A | 103 | 3 |
CDK9-Cyclin T1 | 92 | 8 |
CHK1 | 96 | 12 |
CHK2 | 96 | 14 |
CK1 delta | 96 | 3 |
CK1 gamma 2 | 101 | 10 |
CK2 | 91 | 3 |
CLK2 | 98 | 1 |
CSK | 100 | 12 |
DAPK1 | 35 | 3 |
DDR2 | 107 | 11 |
DYRK1A | 92 | 6 |
DYRK2 | 97 | 4 |
DYRK3 | 94 | 0 |
EF2K | 105 | 1 |
EIF2AK3 | 100 | 9 |
EPH-A2 | 100 | 3 |
EPH-A4 | 86 | 5 |
EPH-B1 | 111 | 7 |
EPH-B2 | 119 | 14 |
EPH-B3 | 120 | 0 |
EPH-B4 | 119 | 15 |
ERK1 | 103 | 13 |
ERK2 | 107 | 11 |
ERK8 | 99 | 4 |
FGF-R1 | 105 | 2 |
GCK | 97 | 6 |
GSK3 beta | 106 | 10 |
HER4 | 106 | 9 |
HIPK1 | 94 | 10 |
HIPK2 | 95 | 5 |
HIPK3 | 99 | 7 |
IGF-1R | 98 | 2 |
IKK beta | 118 | 0 |
IKK epsilon | 91 | 5 |
IR | 101 | 11 |
IRAK1 | 105 | 3 |
IRAK4 | 92 | 6 |
IRR | 117 | 5 |
JAK2 | 108 | 7 |
JNK1 | 94 | 5 |
JNK2 | 104 | 1 |
JNK3 | 87 | 6 |
Lck | 97 | 5 |
LKB1 | 110 | 3 |
MAPKAP-K2 | 86 | 12 |
MAPKAP-K3 | 91 | 0 |
MARK1 | 99 | 2 |
MARK2 | 96 | 4 |
MARK3 | 88 | 12 |
MARK4 | 99 | 7 |
MEKK1 | 87 | 2 |
MELK | 31 | 1 |
MINK1 | 89 | 1 |
MKK1 | 85 | 6 |
MKK2 | 114 | 7 |
MKK6 | 87 | 5 |
MLK1 | 93 | 2 |
MLK3 | 80 | 5 |
MNK1 | 111 | 9 |
MNK2 | 80 | 6 |
MPSK1 | 105 | 12 |
MSK1 | 95 | 1 |
MST2 | 91 | 2 |
MST3 | 110 | 6 |
MST4 | 102 | 15 |
NEK2a | 94 | 2 |
NEK6 | 84 | 13 |
NUAK1 | 47 | 7 |
OSR1 | 112 | 15 |
p38 alpha MAPK | 100 | 6 |
p38 beta MAPK | 105 | 5 |
p38 delta MAPK | 93 | 4 |
p38 gamma MAPK | 99 | 4 |
PAK2 | 102 | 7 |
PAK4 | 100 | 2 |
PAK5 | 97 | 7 |
PAK6 | 99 | 13 |
PDK1 |
2
|
0 |
PHK | 101 | 3 |
PIM1 | 112 | 8 |
PIM2 | 97 | 5 |
PIM3 | 94 | 15 |
PKA | 102 | 10 |
PKB alpha | 98 | 14 |
PKB beta | 107 | 2 |
PKC alpha | 98 | 10 |
PKC gamma | 100 | 23 |
PKC zeta | 74 | 14 |
PKD1 | 106 | 7 |
PLK1 | 97 | 12 |
PRAK | 110 | 14 |
PRK2 | 118 | 6 |
RIPK2 | 116 | 1 |
ROCK 2 | 67 | 1 |
RSK1 | 86 | 12 |
RSK2 | 79 | 3 |
S6K1 | 108 | 9 |
SGK1 | 81 | 5 |
SIK2 | 106 | 0 |
SIK3 | 76 | 2 |
SmMLCK | 99 | 15 |
Src | 95 | 2 |
SRPK1 | 104 | 13 |
STK33 | 89 | 0 |
SYK | 104 | 7 |
TAK1 | 99 | 7 |
TAO1 | 86 | 3 |
TBK1 | 89 | 3 |
TESK1 | 91 | 1 |
TIE2 | 105 | 8 |
TLK1 | 101 | 6 |
TrkA | 94 | 7 |
TSSK1 | 88 | 0 |
TTBK1 | 112 | 7 |
TTK | 84 | 9 |
VEGFR1 | 89 | 6 |
WNK1 | 109 | 4 |
YES1 | 106 | 6 |
ZAP70 | 98 | 0 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
ABL | 100 | 11 |
AMPK | 44 | 9 |
ASK1 | 99 | 10 |
Aurora A | 89 | 5 |
Aurora B | 29 | 12 |
BRK | 116 | 1 |
BRSK1 | 11 | 1 |
BRSK2 | 15 | 2 |
BTK | 90 | 6 |
CAMK1 | 95 | 1 |
CAMKK beta | 91 | 1 |
CDK2-Cyclin A | 85 | 1 |
CDK9-Cyclin T1 | 100 | 15 |
CHK1 | 103 | 11 |
CHK2 | 51 | 1 |
CK1 delta | 88 | 2 |
CK1 gamma 2 | 97 | 1 |
CK2 | 111 | 3 |
CLK2 | 88 | 12 |
CSK | 93 | 4 |
DAPK1 | 12 | 1 |
DDR2 | 111 | 25 |
DYRK1A | 82 | 6 |
DYRK2 | 58 | 6 |
DYRK3 | 88 | 6 |
EF2K | 100 | 2 |
EIF2AK3 | 100 | 16 |
EPH-A2 | 84 | 3 |
EPH-A4 | 98 | 2 |
EPH-B1 | 118 | 4 |
EPH-B2 | 111 | 16 |
EPH-B3 | 103 | 3 |
EPH-B4 | 117 | 5 |
ERK1 | 108 | 1 |
ERK2 | 109 | 6 |
ERK8 | 83 | 1 |
FGF-R1 | 88 | 2 |
GCK | 86 | 7 |
GSK3 beta | 101 | 24 |
HER4 | 101 | 13 |
HIPK1 | 112 | 4 |
HIPK2 | 113 | 1 |
HIPK3 | 103 | 1 |
IGF-1R | 100 | 10 |
IKK beta | 103 | 5 |
IKK epsilon | 45 | 5 |
IR | 89 | 13 |
IRAK1 | 106 | 6 |
IRAK4 | 99 | 1 |
IRR | 101 | 21 |
JAK2 | 99 | 10 |
JNK1 | 108 | 4 |
JNK2 | 114 | 5 |
JNK3 | 97 | 4 |
Lck | 99 | 5 |
LKB1 | 103 | 4 |
MAPKAP-K2 | 84 | 2 |
MAPKAP-K3 | 68 | 2 |
MARK1 | 84 | 3 |
MARK2 | 102 | 7 |
MARK3 | 87 | 1 |
MARK4 | 103 | 7 |
MEKK1 | 104 | 1 |
MELK | 22 | 3 |
MINK1 | 74 | 0 |
MKK1 | 74 | 5 |
MKK2 | 94 | 2 |
MKK6 | 94 | 3 |
MLK1 | 78 | 1 |
MLK3 | 44 | 1 |
MNK1 | 92 | 3 |
MNK2 | 94 | 6 |
MPSK1 | 104 | 1 |
MSK1 | 66 | 10 |
MST2 | 84 | 2 |
MST3 | 110 | 16 |
MST4 | 102 | 9 |
NEK2a | 91 | 9 |
NEK6 | 79 | 1 |
NUAK1 |
9
|
2 |
OSR1 | 103 | 12 |
p38 alpha MAPK | 99 | 8 |
p38 beta MAPK | 109 | 5 |
p38 delta MAPK | 101 | 7 |
p38 gamma MAPK | 110 | 6 |
PAK2 | 77 | 3 |
PAK4 | 106 | 35 |
PAK5 | 99 | 1 |
PAK6 | 96 | 6 |
PDK1 | 15 | 0 |
PHK | 78 | 2 |
PIM1 | 93 | 4 |
PIM2 | 110 | 3 |
PIM3 | 73 | 7 |
PKA | 84 | 5 |
PKB alpha | 36 | 5 |
PKB beta | 56 | 2 |
PKC alpha | 96 | 4 |
PKC gamma | 87 | 17 |
PKC zeta | 23 | 6 |
PKD1 | 84 | 8 |
PLK1 | 94 | 22 |
PRAK | 95 | 5 |
PRK2 | 81 | 0 |
RIPK2 | 100 | 11 |
ROCK 2 | 27 | 2 |
RSK1 | 40 | 11 |
RSK2 | 28 | 2 |
S6K1 | 81 | 1 |
SGK1 | 37 | 1 |
SIK2 | 78 | 18 |
SIK3 | 58 | 7 |
SmMLCK | 62 | 3 |
Src | 99 | 6 |
SRPK1 | 90 | 5 |
STK33 | 43 | 5 |
SYK | 105 | 7 |
TAK1 | 79 | 0 |
TAO1 | 96 | 8 |
TBK1 | 81 | 2 |
TESK1 | 101 | 7 |
TIE2 | 76 | 13 |
TLK1 | 115 | 11 |
TrkA | 84 | 10 |
TSSK1 | 64 | 3 |
TTBK1 | 99 | 11 |
TTK | 61 | 0 |
VEGFR1 | 64 | 10 |
WNK1 | 104 | 6 |
YES1 | 98 | 5 |
ZAP70 | 127 | 30 |