Inhibitor | Quercetagetin  

Compound name Brutto MW CAS PubChem CID Action Reference Reference
Quercetagetin   C15H10O8 318.30 90-18-6 5281680 PIM1 Holder S. (2007) Mol. Cancer Ther. 6 163

Screening Results Chart

Screening Results Tables

Screen Conc: 1.00µM
Kinase % Activity Remaining Standard Deviation
AMPK 73 6
ASK1 118 0
Aurora A 95 11
Aurora B 62 4
BRSK1 82 1
BRSK2 71 10
BTK 61 2
CAMK1 49 1
CAMKK beta 72 0
CDK2-Cyclin A 89 12
CHK1 92 12
CHK2 48 12
CK1 delta 90 0
CK2 46 3
CLK2 58 9
CSK 125 12
DAPK1 95 11
DYRK1A 71 11
DYRK2 45 2
DYRK3 59 3
EF2K 110 8
EPH-A2 94 14
EPH-A4 117 3
EPH-B1 85 8
EPH-B2 69 4
EPH-B3 93 5
EPH-B4 90 13
ERK1 101 2
ERK2 107 8
ERK8 89 0
FGF-R1 27 1
GCK 93 1
GSK3 beta 94 5
HER4 109 4
HIPK1 93 5
HIPK2 62 7
HIPK3 88 10
IGF-1R 96 3
IKK beta 100 6
IKK epsilon 69 4
IR 86 0
IRAK4 80 3
IRR 76 4
JAK2 91 5
JNK1 93 1
JNK2 106 7
JNK3 107 2
Lck 102 15
LKB1 95 12
MAPKAP-K2 94 1
MAPKAP-K3 92 3
MARK1 40 0
MARK2 86 2
MARK3 51 1
MARK4 34 1
MEKK1 67 4
MELK 53 3
MINK1 56 4
MKK1 84 0
MKK2 94 1
MKK6 102 7
MLK1 100 5
MLK3 62 1
MNK1 61 2
MNK2 63 7
MSK1 88 1
MST2 58 2
MST4 87 2
NEK2a 86 3
NEK6 99 8
NUAK1 33 7
p38 alpha MAPK 100 4
p38 beta MAPK 101 7
p38 delta MAPK 96 7
p38 gamma MAPK 107 2
PAK2 96 7
PAK4 50 3
PAK5 67 0
PAK6 58 2
PDK1 104 0
PHK 98 2
PIM1 37 6
PIM2 74 1
PIM3 34 1
PKA 109 7
PKB alpha 106 9
PKB beta 21 7
PKC alpha 99 7
PKC zeta 62 0
PKD1 69 3
PLK1 107 11
PRAK 87 1
PRK2 106 7
RIPK2 83 10
ROCK 2 95 4
RSK1 51 0
RSK2 22 0
S6K1 104 3
SGK1 87 3
SmMLCK 87 0
Src 38 0
SRPK1 55 10
SYK 89 6
TAK1 94 10
TAO1 94 11
TBK1 54 4
TrkA 92 9
TTK 75 0
VEGFR1 27 4
YES1 42 1
Screen Conc: 10.00µM
Kinase % Activity Remaining Standard Deviation
AMPK
9
 3
Aurora A 28 2
Aurora B
8
 1
BRSK1
7
 0
BRSK2 13 1
BTK 32 2
CAMK1 19 3
CAMKK beta 61 5
CDK2-Cyclin A 32 0
CHK1 32 1
CHK2
5
 1
CK1 delta 29 1
CK2
7
 0
CSK 74 0
DYRK1A
3
 0
DYRK2
1
 0
DYRK3
2
 0
EF2K 109 1
EPH-A2 73 6
EPH-A4 74 6
EPH-B3 61 6
EPH-B4 56 11
ERK1 54 4
ERK2 105 1
ERK8 65 1
FGF-R1 14 0
GCK 23 1
GSK3 beta 19 1
HER4 44 2
HIPK1 11 1
HIPK2 19 0
HIPK3 55 0
IGF-1R 43 2
IKK beta 16 5
IKK epsilon 21 1
IR 62 3
IRAK4 46 0
IRR 21 1
JAK2 13 7
JNK1 93 3
JNK2 100 9
JNK3 89 1
Lck 95 9
LKB1 55 6
MAPKAP-K2 53 14
MAPKAP-K3 14 0
MARK1 11 0
MARK2 26 3
MARK3
6
 1
MARK4 20 0
MEKK1 74 6
MELK
9
 1
MINK1
10
 0
MKK1 24 4
MLK1 24 0
MLK3 16 0
MNK1 12 4
MNK2 26 5
MSK1 38 0
MST2
9
 0
MST4 58 5
NEK2a 13 1
NEK6 21 1
NUAK1 12 0
p38 alpha MAPK 119 6
p38 beta MAPK 90 0
p38 delta MAPK 97 8
p38 gamma MAPK 88 6
PAK2 98 2
PAK4 38 6
PAK5 55 6
PAK6 60 12
PDK1 83 13
PHK
2
 0
PIM1
7
 0
PIM2 11 0
PIM3
0
 0
PKA 79 2
PKB alpha 99 10
PKB beta
1
 0
PKC alpha 80 13
PKC zeta 20 0
PKD1 15 6
PLK1 23 4
PRAK
1
 0
PRK2 102 1
RIPK2
7
 0
ROCK 2 56 3
RSK1 15 0
RSK2 12 1
S6K1 14 0
SGK1 24 2
SmMLCK 23 0
Src 25 2
SRPK1
3
 0
SYK 93 8
TAK1
5
 2
TBK1 64 10
TrkA 29 2
TTK 36 6
VEGFR1
7
 0
YES1
9
 0