Inhibitor | ER-27319  

Screen Conc: 10.00µM

Kinase	% Activity Remaining Sort descending	Standard Deviation
PIM3	43	9
ERK8	54	9
IRR	65	10
PIM1	67	1
CK2	69	5
IR	73	2
MNK1	78	12
MELK	78	4
RSK1	78	6
PKD1	80	17
PKC zeta	81	0
FGF-R1	83	9
CHK2	83	8
BRSK2	85	0
PAK4	85	5
EPH-B3	85	4
DYRK1A	85	12
ERK1	85	12
p38 beta MAPK	85	7
Lck	86	3
PDK1	87	0
DYRK3	87	2
PKC alpha	88	12
BTK	88	11
PHK	89	0
MKK1	89	2
MST4	89	9
SYK	89	4
MNK2	90	0
SGK1	90	3
CDK2-Cyclin A	90	11
Aurora B	90	1
Src	92	7
SmMLCK	92	6
p38 delta MAPK	93	7
MAPKAP-K2	93	8
IGF-1R	93	2
ROCK 2	94	5
PIM2	95	0
SRPK1	95	4
VEGFR1	95	4
PRAK	96	2
IKK epsilon	96	1
IKK beta	96	6
PRK2	96	0
JNK2	96	11
AMPK	96	3
MARK3	96	5
HIPK2	97	20
CAMKK beta	97	0
DYRK2	97	9
CHK1	97	6
EPH-A2	97	2
TBK1	98	11
CAMK1	98	5
RSK2	99	1
PAK6	99	8
JNK1	99	2
PAK5	100	7
CSK	100	10
NEK6	100	0
ERK2	100	4
YES1	100	3
PKB alpha	101	1
MST2	101	1
p38 gamma MAPK	101	5
CK1 delta	107	8
GSK3 beta	107	1
S6K1	109	8
PKA	109	8
p38 alpha MAPK	111	9
MSK1	112	0
PLK1	113	7
PKB beta	117	3
NEK2a	120	12
EF2K	120	1

Screen Conc: 1.00µM

Kinase	% Activity Remaining Sort descending	Standard Deviation
IR	76	4
MELK	77	2
FGF-R1	79	5
IRR	80	3
p38 beta MAPK	81	10
PIM3	82	1
PKC zeta	83	12
YES1	84	5
NEK6	84	4
BTK	85	7
PAK5	85	2
MNK1	85	12
EPH-B3	86	13
TBK1	88	0
MAPKAP-K2	88	9
SGK1	89	10
BRSK2	89	9
PAK4	89	7
p38 delta MAPK	89	11
ERK8	91	9
CDK2-Cyclin A	91	2
MKK1	92	11
CK2	93	5
Src	93	2
DYRK3	93	5
CHK2	93	14
ERK2	95	7
PKD1	95	10
CHK1	95	9
PKA	96	17
PIM2	96	2
PRAK	96	5
DYRK1A	97	2
JNK2	97	10
CSK	97	5
JNK1	98	0
p38 gamma MAPK	98	7
PIM1	98	0
HIPK2	99	7
PAK6	99	0
DYRK2	99	3
EPH-A2	99	4
MST4	99	8
SYK	99	8
PDK1	100	5
CAMKK beta	100	0
ERK1	100	3
IKK beta	100	10
IGF-1R	101	19
CAMK1	101	4
RSK1	101	1
Aurora B	102	1
MNK2	102	10
MST2	103	2
PLK1	105	6
VEGFR1	105	6
MARK3	105	13
SmMLCK	105	8
Lck	106	8
PHK	106	11
GSK3 beta	106	0
ROCK 2	107	13
IKK epsilon	107	13
PKB alpha	108	12
p38 alpha MAPK	110	0
SRPK1	111	0
AMPK	113	8
PRK2	113	2
RSK2	113	4
PKC alpha	118	27
MSK1	118	0
NEK2a	120	1
CK1 delta	121	1
EF2K	122	0
PKB beta	123	0
S6K1	130	8