Inhibitor | AG879 (Tyrphostin)  

Screen Conc: 10.00µM

Kinase	% Activity Remaining Sort descending	Standard Deviation
MELK	8	4
PLK1	13	2
PKB beta	15	9
HIPK2	21	2
PIM1	25	3
PRAK	27	2
PHK	28	1
PIM3	34	8
ERK8	37	0
GSK3 beta	39	4
CDK2-Cyclin A	40	0
CAMKK beta	44	12
IRR	45	4
BTK	46	8
VEGFR1	50	3
SmMLCK	52	5
PIM2	53	5
MST2	54	1
EPH-B3	55	1
PAK4	56	2
DYRK1A	56	3
FGF-R1	59	0
DYRK3	60	1
SRPK1	61	12
RSK2	61	4
IKK epsilon	63	9
S6K1	64	14
BRSK2	66	4
PKC zeta	67	2
Src	67	0
JNK2	70	9
AMPK	70	2
MST4	72	14
MNK2	76	9
PKC alpha	78	6
RSK1	79	1
PKD1	80	3
PAK6	80	1
p38 alpha MAPK	81	9
NEK2a	82	18
MKK1	83	13
YES1	85	1
p38 beta MAPK	86	8
IGF-1R	86	4
p38 delta MAPK	86	11
JNK1	87	16
ERK2	87	1
MSK1	88	3
CAMK1	88	7
CSK	89	6
MARK3	90	7
EF2K	90	8
ERK1	90	8
p38 gamma MAPK	92	3
CK1 delta	92	6
CHK1	92	19
PKA	93	10
PKB alpha	94	4
ROCK 2	94	0
PDK1	96	5
CHK2	96	14
TBK1	97	1
MNK1	99	8
MAPKAP-K2	99	2
NEK6	101	16
DYRK2	102	31
IKK beta	105	13
Lck	107	13
SGK1	107	13
EPH-A2	113	11
PRK2	114	16
CK2	118	5
SYK	138	2
IR	139	52
PAK5	519	649

Screen Conc: 0.10µM

Kinase	% Activity Remaining Sort descending	Standard Deviation
BTK	55	4
RSK2	67	2
MELK	76	1
IKK epsilon	78	8
AMPK	78	0
CAMKK beta	78	22
MSK1	82	3
MST4	83	0
PKB beta	84	3
MNK2	84	0
DYRK1A	84	1
SmMLCK	85	20
NEK2a	85	17
PKA	85	3
CAMK1	85	9
CHK1	86	1
SRPK1	86	0
PKC zeta	86	7
PAK6	86	1
BRSK2	87	9
IRR	88	0
ERK1	88	16
p38 beta MAPK	89	6
JNK2	90	10
TBK1	90	6
ERK2	91	2
S6K1	92	4
MARK3	92	6
VEGFR1	92	3
CSK	92	15
PHK	93	19
p38 delta MAPK	93	11
EPH-A2	94	12
MKK1	95	1
GSK3 beta	95	7
CK1 delta	95	0
Src	95	11
ERK8	96	2
EPH-B3	96	10
PIM2	98	1
PIM3	98	19
IGF-1R	98	16
p38 gamma MAPK	98	7
DYRK3	98	11
JNK1	99	9
PKD1	99	12
RSK1	99	9
Lck	99	8
NEK6	100	24
PDK1	100	0
PRK2	101	30
PKC alpha	101	10
MNK1	101	4
PIM1	102	22
PRAK	102	2
PKB alpha	103	1
PLK1	105	9
p38 alpha MAPK	105	7
EF2K	105	4
PAK4	105	11
MAPKAP-K2	108	11
IKK beta	109	10
CHK2	109	23
CDK2-Cyclin A	110	1
DYRK2	110	8
YES1	111	13
ROCK 2	113	10
MST2	113	8
HIPK2	118	15
IR	118	7
FGF-R1	120	17
CK2	123	8
SGK1	124	15
SYK	173	70
PAK5	585	715