Inhibitor | A-83-01  

Screen Conc: 1.00µM

Kinase	% Activity Remaining Sort descending	Standard Deviation
VEGFR1	8	1
RIPK2	9	3
MINK1	13	2
p38 alpha MAPK	16	1
PKD1	32	9
FGF-R1	37	2
CK1 delta	46	5
p38 beta MAPK	61	7
Lck	62	3
GCK	68	7
YES1	70	5
Src	75	1
GSK3 beta	79	4
TAK1	81	9
AMPK	82	4
HER4	82	15
SRPK1	84	1
NUAK1	84	4
MLK1	86	2
MARK4	87	2
p38 gamma MAPK	88	8
PDK1	88	0
SmMLCK	89	1
JNK2	90	7
DAPK1	90	2
PRK2	91	3
MNK2	91	2
NEK2a	92	3
EPH-A2	92	14
BRSK2	92	14
DYRK3	93	4
PAK4	93	4
CSK	93	1
MNK1	93	1
ERK8	93	4
JAK2	93	4
EPH-B4	93	19
IR	94	6
p38 delta MAPK	94	4
PIM2	94	3
ERK2	94	2
HIPK2	95	12
DYRK2	95	7
RSK1	95	2
EPH-B2	95	5
BRSK1	95	7
PKB beta	96	5
MAPKAP-K3	97	4
PIM1	97	4
TTK	98	6
CLK2	98	0
MARK3	98	7
EPH-A4	98	3
MKK1	98	1
HIPK1	98	11
JNK3	99	7
HIPK3	99	1
TrkA	99	11
LKB1	99	11
MST4	99	1
PRAK	99	16
PKA	99	5
IRAK4	99	5
PKC zeta	100	3
NEK6	100	5
IKK beta	100	12
MST2	100	6
ERK1	100	5
EF2K	100	3
PAK2	101	12
MSK1	101	0
JNK1	101	4
PKC alpha	102	7
CDK2-Cyclin A	102	11
Aurora B	102	1
PAK5	102	4
IGF-1R	103	11
IRR	103	3
SGK1	103	14
CK2	104	11
DYRK1A	104	1
BTK	104	5
CAMKK beta	104	2
EPH-B3	104	0
ROCK 2	104	2
S6K1	105	13
MELK	105	3
CHK1	105	3
PLK1	106	7
IKK epsilon	106	0
SYK	106	2
TBK1	106	1
PKB alpha	106	9
Aurora A	107	3
CAMK1	107	13
MLK3	107	4
MAPKAP-K2	108	2
RSK2	109	8
CHK2	110	6
MARK2	110	9
MEKK1	111	0
PHK	112	4
PAK6	113	19
MARK1	113	7
PIM3	117	11

Screen Conc: 0.10µM

Kinase	% Activity Remaining Sort descending	Standard Deviation
RIPK2	26	6
VEGFR1	27	0
p38 alpha MAPK	56	1
FGF-R1	64	3
MINK1	66	2
PKD1	80	1
MNK2	81	5
p38 beta MAPK	89	15
PAK4	89	6
CK1 delta	90	8
PIM3	91	4
p38 delta MAPK	91	20
EPH-B4	93	2
CDK2-Cyclin A	93	4
DAPK1	94	3
MST4	95	2
MLK1	96	7
ROCK 2	96	2
NUAK1	96	10
HIPK1	96	4
PIM2	97	4
IGF-1R	97	5
PKC alpha	97	5
CSK	97	2
GCK	98	3
MARK4	98	2
IRR	98	5
PKC zeta	98	0
Aurora B	98	5
AMPK	99	3
TAK1	99	9
GSK3 beta	99	1
PLK1	99	11
CAMKK beta	100	10
PHK	100	11
DYRK2	100	0
MARK3	101	4
SRPK1	101	7
IRAK4	101	3
LKB1	101	5
TBK1	102	7
PKB alpha	102	5
EF2K	102	4
CK2	102	0
Src	102	1
p38 gamma MAPK	102	13
DYRK3	102	8
PDK1	103	8
CAMK1	103	18
MNK1	103	1
SmMLCK	104	8
MLK3	104	2
ERK2	104	11
HER4	104	1
HIPK2	104	8
EPH-A2	105	5
PIM1	105	3
ERK1	105	15
JNK2	105	6
PRK2	105	12
HIPK3	105	8
Lck	105	7
CLK2	106	10
YES1	106	4
IKK beta	107	1
MST2	107	0
JAK2	107	18
MAPKAP-K3	107	3
MARK1	107	3
SGK1	107	1
CHK1	107	10
PAK5	107	2
NEK6	107	3
EPH-A4	108	1
PKB beta	108	3
S6K1	108	2
IR	108	7
ERK8	108	16
SYK	109	10
PKA	109	2
DYRK1A	109	11
NEK2a	109	8
RSK1	110	6
BRSK1	110	12
MSK1	110	6
BTK	110	5
MKK1	111	20
MELK	111	2
JNK1	111	3
PAK2	111	17
PAK6	111	12
IKK epsilon	112	5
EPH-B3	112	6
PRAK	113	7
EPH-B2	113	2
TTK	113	0
CHK2	115	10
MAPKAP-K2	117	3
BRSK2	117	6
TrkA	118	2
JNK3	119	3
Aurora A	120	7
MARK2	121	8
RSK2	126	3
MEKK1	130	15