Kinase Profiling Inhibitor Database

Inhibitor Structure Image Brutto MW Action Reference Reference 2 Patent Commercial Vendor Notes Results
SGK1-Sanofi-308-S C23H23FN6O4S 498.53 SGK1 WO2014140065 Download

Results as Barchart

View results as a bar chart
1µM

Results as Table

Screening Concentration: 1µM
Kinase % Activity Remaining Standard Deviation
MKK1 66 0
MKK2 77 6
MKK6 102 14
ERK1 119 2
ERK2 106 10
ERK5 94 5
JNK1 107 3
JNK2 92 16
JNK3 105 10
p38 alpha MAPK 86 7
p38 beta MAPK 104 0
p38 gamma MAPK 102 6
p38 delta MAPK 116 3
ERK8 50 13
RSK1 9 1
RSK2 36 3
PDK1 84 23
PKB alpha 91 6
PKB beta 44 9
SGK1 11 4
S6K1 1 0
PKA 98 6
ROCK 2 73 10
PRK2 71 11
PKC alpha 94 18
PKC gamma 89 6
PKC zeta 81 22
PKD1 58 3
STK33 46 27
MSK1 13 1
MNK1 96 13
MNK2 66 10
MAPKAP-K2 88 2
MAPKAP-K3 91 0
PRAK 100 1
CAMKK beta 102 1
CAMK1 30 16
SmMLCK 88 10
PHK 90 11
DAPK1 114 3
CHK1 103 1
CHK2 21 3
GSK3 beta 93 3
CDK2-Cyclin A 52 3
CDK9-Cyclin T1 71 0
PLK1 92 2
Aurora A 94 5
Aurora B 108 3
TLK1 87 11
LKB1 98 10
AMPK (hum) 72 3
MARK1 102 18
MARK2 76 3
MARK3 94 2
MARK4 98 9
BRSK1 121 14
BRSK2 77 13
MELK 22 4
NUAK1 70 1
SIK2 97 25
SIK3 87 28
TSSK1 92 4
CK1 gamma 2 104 13
CK1 delta 118 2
CK2 93 13
TTBK1 95 1
TTBK2 121 10
DYRK1A 99 1
DYRK2 96 17
DYRK3 99 0
NEK2a 83 22
NEK6 112 2
IKK beta 88 1
IKK epsilon 30 1
TBK1 86 2
PIM1 114 14
PIM2 97 8
PIM3 76 7
SRPK1 121 17
EF2K 115 13
EIF2AK3 86 0
HIPK1 71 3
HIPK2 40 4
HIPK3 58 0
CLK2 104 5
PAK2 95 10
PAK4 93 12
PAK5 105 3
PAK6 91 6
MST2 101 6
MST3 73 1
MST4 141 48
GCK 89 1
MAP4K3 38 2
MAP4K5 80 7
MINK1 91 6
MEKK1 98 7
MLK1 24 6
MLK3 29 1
TESK1 101 1
TAO1 88 0
ASK1 76 3
TAK1 80 4
IRAK1 107 9
IRAK4 100 1
RIPK2 103 19
OSR1 101 3
TTK 97 1
MPSK1 101 0
WNK1 98 2
ULK1 93 14
ULK2 99 8
TGFBR1 103 7
Src 132 3
Lck 106 6
CSK 101 3
YES1 77 22
ABL 75 1
BTK 74 6
JAK2 92 4
SYK 86 5
ZAP70 116 7
TIE2 59 0
BRK 83 20
EPH-A2 105 10
EPH-A4 73 18
EPH-B1 103 6
EPH-B2 84 4
EPH-B3 109 20
EPH-B4 113 2
FGF-R1 121 10
HER4 103 6
IGF-1R 92 7
IR 126 6
IRR 99 9
TrkA 79 7
DDR2 99 10
VEGFR1 126 10
PDGFRA 122 7
PINK 102 26

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