Kinase Profiling Inhibitor Database

Inhibitor Structure Image Brutto MW Action Reference Reference 2 Patent Commercial Vendor Notes Results
STOCK1S-50699 C29H31IN2S2 598.60 WNK Mori T. (2013) Biochem J. 1 455(3) 339-45 Molport Download

Results as Barchart

View results as a bar chart
1µM
10µM

Results as Table

Screening Concentration: 10µM
Kinase % Activity Remaining Standard Deviation
MKK1 94 8
MKK2 85 3
MKK6 112 9
ERK1 58 2
ERK2 69 8
ERK5 87 16
JNK1 87 7
JNK2 96 2
JNK3 103 8
p38 alpha MAPK 91 5
p38 beta MAPK 98 5
p38 gamma MAPK 90 1
p38 delta MAPK 87 4
ERK8 55 7
RSK1 47 18
RSK2 43 8
PDK1 116 4
PKB alpha 65 2
PKB beta 77 3
SGK1 51 2
S6K1 85 16
PKA 92 7
ROCK 2 89 1
PRK2 65 17
PKC alpha 88 23
PKC gamma 86 5
PKC zeta 110 1
PKD1 61 4
STK33 95 3
MSK1 67 3
MNK1 97 7
MNK2 105 16
MAPKAP-K2 98 3
MAPKAP-K3 84 8
PRAK 92 1
CAMKK beta 96 12
CAMK1 95 1
SmMLCK 99 28
PHK 104 0
DAPK1 115 14
CHK1 97 6
CHK2 88 8
GSK3 beta 116 1
CDK2-Cyclin A 99 20
CDK9-Cyclin T1 102 3
PLK1 114 21
Aurora A 108 6
Aurora B 41 10
TLK1 101 11
LKB1 105 27
AMPK (hum) 112 8
MARK1 89 14
MARK2 102 8
MARK3 83 20
MARK4 113 8
BRSK1 95 15
BRSK2 61 10
MELK 53 1
NUAK1 88 8
SIK2 83 10
SIK3 88 3
TSSK1 72 10
CK1 gamma 2 72 10
CK1 delta 32 12
CK2 82 2
TTBK1 104 0
TTBK2 100 5
DYRK1A 66 3
DYRK2 85 2
DYRK3 102 6
NEK2a 103 2
NEK6 91 2
IKK beta 78 3
IKK epsilon 60 6
TBK1 84 12
PIM1 73 4
PIM2 84 2
PIM3 84 7
SRPK1 95 16
EF2K 87 2
EIF2AK3 107 7
HIPK1 76 10
HIPK2 116 10
HIPK3 93 7
CLK2 90 1
PAK2 94 0
PAK4 108 0
PAK5 99 1
PAK6 102 1
MST2 69 11
MST3 110 7
MST4 85 14
GCK 100 10
MAP4K3 89 3
MAP4K5 103 2
MINK1 88 0
MEKK1 84 3
MLK1 87 4
MLK3 75 3
TESK1 112 10
TAO1 93 0
ASK1 101 3
TAK1 68 13
IRAK1 57 3
IRAK4 96 17
RIPK2 82 9
OSR1 112 2
TTK 64 17
MPSK1 79 7
WNK1 104 12
ULK1 83 5
ULK2 90 1
TGFBR1 108 1
Src 143 5
Lck 101 1
CSK 109 19
YES1 105 10
ABL 99 5
BTK 104 6
JAK2 125 13
SYK 64 1
ZAP70 112 11
TIE2 96 4
BRK 95 32
EPH-A2 103 1
EPH-A4 98 14
EPH-B1 93 11
EPH-B2 106 10
EPH-B3 98 16
EPH-B4 109 13
FGF-R1 77 4
HER4 110 12
IGF-1R 83 4
IR 90 17
IRR 72 5
TrkA 90 1
DDR2 110 9
VEGFR1 23 3
PDGFRA 123 16
PINK 103 21
Screening Concentration: 1µM
Kinase % Activity Remaining Standard Deviation
MKK1 96 14
MKK2 90 2
MKK6 95 6
ERK1 94 11
ERK2 84 11
ERK5 103 8
JNK1 97 12
JNK2 97 2
JNK3 105 1
p38 alpha MAPK 95 3
p38 beta MAPK 121 15
p38 gamma MAPK 94 5
p38 delta MAPK 104 2
ERK8 88 12
RSK1 85 5
RSK2 108 10
PDK1 93 14
PKB alpha 85 6
PKB beta 93 2
SGK1 110 14
S6K1 96 9
PKA 96 12
ROCK 2 90 2
PRK2 92 13
PKC alpha 80 1
PKC gamma 105 5
PKC zeta 92 3
PKD1 100 11
STK33 106 1
MSK1 100 2
MNK1 106 19
MNK2 99 12
MAPKAP-K2 106 10
MAPKAP-K3 95 1
PRAK 97 6
CAMKK beta 104 6
CAMK1 97 15
SmMLCK 95 25
PHK 103 4
DAPK1 103 0
CHK1 106 4
CHK2 99 12
GSK3 beta 103 10
CDK2-Cyclin A 104 14
CDK9-Cyclin T1 101 1
PLK1 102 0
Aurora A 99 1
Aurora B 87 22
TLK1 93 8
LKB1 103 10
AMPK (hum) 108 3
MARK1 100 14
MARK2 95 2
MARK3 100 7
MARK4 111 32
BRSK1 113 15
BRSK2 94 4
MELK 90 4
NUAK1 101 5
SIK2 108 22
SIK3 97 0
TSSK1 96 3
CK1 gamma 2 97 1
CK1 delta 86 7
CK2 107 0
TTBK1 102 9
TTBK2 90 5
DYRK1A 78 3
DYRK2 91 4
DYRK3 102 6
NEK2a 107 6
NEK6 99 15
IKK beta 98 10
IKK epsilon 96 8
TBK1 111 4
PIM1 94 10
PIM2 93 6
PIM3 82 8
SRPK1 93 3
EF2K 101 6
EIF2AK3 101 1
HIPK1 95 5
HIPK2 110 0
HIPK3 95 1
CLK2 89 1
PAK2 96 1
PAK4 103 1
PAK5 105 6
PAK6 100 0
MST2 71 6
MST3 110 8
MST4 75 16
GCK 107 6
MAP4K3 97 1
MAP4K5 103 3
MINK1 90 6
MEKK1 90 6
MLK1 95 4
MLK3 96 8
TESK1 104 3
TAO1 96 0
ASK1 107 10
TAK1 100 10
IRAK1 82 15
IRAK4 90 10
RIPK2 84 9
OSR1 112 5
TTK 87 18
MPSK1 101 5
WNK1 103 2
ULK1 108 8
ULK2 96 8
TGFBR1 111 1
Src 91 5
Lck 115 2
CSK 85 10
YES1 106 11
ABL 113 17
BTK 106 21
JAK2 110 1
SYK 92 2
ZAP70 112 1
TIE2 93 1
BRK 104 14
EPH-A2 116 6
EPH-A4 93 14
EPH-B1 125 24
EPH-B2 102 7
EPH-B3 93 13
EPH-B4 112 5
FGF-R1 96 1
HER4 121 8
IGF-1R 95 29
IR 114 1
IRR 105 18
TrkA 96 7
DDR2 102 1
VEGFR1 84 10
PDGFRA 102 2
PINK 101 1

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