Kinase Profiling Inhibitor Database

Inhibitor Structure Image Brutto MW Action Reference Reference 2 Patent Commercial Vendor Notes Results
Chloroquine C18H26ClN3 319.87214 Anti Malarial Download

Results as Barchart

View results as a bar chart
10µM
1µM

Results as Table

Screening Concentration: 10µM
Kinase % Activity Remainingsort descending Standard Deviation
IKK beta 76 4
TIE2 81 8
PHK 83 26
PRAK 84 7
DYRK2 89 0
PIM1 90 6
LKB1 90 7
PAK4 91 9
CK1 delta 92 5
BRSK1 93 22
S6K1 94 1
DAPK1 94 7
p38 alpha MAPK 95 13
TBK1 96 11
PIM3 96 2
MARK1 96 9
EPH-B4 97 21
MARK3 97 14
PAK5 97 9
MST3 98 5
PKB alpha 98 1
CDK2-Cyclin A 99 8
IRAK1 99 2
TrkA 99 15
IKK epsilon 100 22
EPH-A2 100 9
EPH-A4 100 8
MKK1 100 17
EPH-B2 100 11
CSK 100 5
YES1 100 7
JNK1 100 9
IR 100 11
MSK1 101 3
ERK2 101 3
HIPK3 101 11
ABL 101 10
MARK4 101 5
NEK2a 101 31
ZAP70 102 2
PKA 102 8
NEK6 102 0
p38 delta MAPK 103 1
TLK1 103 7
SmMLCK 103 20
ASK1 103 5
PRK2 103 3
PKC alpha 103 10
MELK 104 10
BRK 104 6
ERK8 104 5
ULK2 104 2
CAMKK beta 104 14
MLK3 104 4
CAMK1 104 5
TSSK1 105 6
MAPKAP-K3 105 18
Src 105 2
AMPK (hum) 105 4
TAO1 105 11
p38 beta MAPK 106 10
MST4 106 2
DYRK3 106 8
IRR 106 27
CHK1 106 10
MST2 107 3
EIF2AK3 107 12
HIPK1 107 9
DYRK1A 107 8
JNK2 107 13
BRSK2 108 19
p38 gamma MAPK 108 9
MPSK1 108 15
ULK1 108 11
MEKK1 108 5
ERK1 108 7
MARK2 108 6
NUAK1 109 5
PINK 109 23
MAPKAP-K2 109 1
EPH-B3 109 3
MLK1 109 1
SGK1 109 14
Lck 109 16
ERK5 109 12
CLK2 109 5
VEGFR1 110 15
OSR1 110 13
PDGFRA 110 6
TTK 110 1
PKC gamma 111 1
PAK6 111 4
SYK 111 1
PIM2 111 26
RSK1 111 5
Aurora A 111 27
SRPK1 111 1
AMPK 111 19
FGF-R1 111 8
IRAK4 112 3
CK1 gamma 2 112 5
PDK1 112 0
MINK1 112 17
TTBK2 112 0
IGF-1R 112 25
SIK2 114 8
MAP4K3 114 16
ROCK 2 114 1
RIPK2 115 2
GCK 115 9
MNK1 115 0
MKK2 115 21
GSK3 beta 116 3
MAP4K5 116 11
TAK1 116 1
JNK3 116 10
DDR2 117 5
RSK2 117 2
PKB beta 117 37
TGFBR1 118 18
TESK1 118 15
PAK2 118 7
CHK2 119 28
WNK1 119 3
CK2 119 3
HER4 119 23
JAK2 119 17
PKC zeta 121 6
STK33 121 24
CDK9-Cyclin T1 121 12
PLK1 121 2
MNK2 123 5
EF2K 124 5
TTBK1 124 2
BTK 124 8
SIK3 125 7
EPH-B1 125 27
Aurora B 126 2
HIPK2 128 4
PKD1 129 44
MKK6 130 15
Screening Concentration: 1µM
Kinase % Activity Remainingsort descending Standard Deviation
PHK 76 4
NEK2a 79 5
IKK epsilon 79 2
PKC alpha 81 24
TIE2 84 1
YES1 85 4
MST3 85 19
BRK 88 8
TSSK1 89 8
PRAK 89 18
PKB beta 90 1
HIPK3 91 11
EPH-A4 92 9
MNK2 92 24
MAPKAP-K2 92 13
ZAP70 92 3
MINK1 94 5
BRSK1 94 7
MNK1 95 33
ULK2 95 37
CK1 delta 96 2
ERK8 97 6
MKK2 97 16
TBK1 97 15
PKA 98 1
IRR 98 8
CHK1 98 3
CDK9-Cyclin T1 99 28
PIM1 99 3
CK2 99 8
PIM3 100 1
ERK5 100 2
BRSK2 100 24
PIM2 101 19
JNK1 101 3
ASK1 101 15
PAK5 101 11
MST4 102 3
TLK1 102 8
EPH-B2 102 7
EPH-B3 102 7
CAMK1 102 5
MARK2 102 20
S6K1 103 12
CSK 103 7
p38 alpha MAPK 103 12
IKK beta 103 9
PDGFRA 103 7
DYRK2 104 0
VEGFR1 104 8
p38 delta MAPK 105 16
MPSK1 105 1
WNK1 105 5
TrkA 105 2
MAP4K5 106 13
AMPK (hum) 106 4
ERK2 106 8
MSK1 107 8
PKB alpha 107 12
SmMLCK 107 16
TTK 108 2
Aurora A 108 7
MKK1 108 24
TTBK2 108 1
ABL 108 6
DDR2 108 3
MELK 108 15
OSR1 108 12
PINK 109 9
CK1 gamma 2 109 0
MLK3 109 7
Lck 109 15
PAK4 109 3
IRAK4 109 7
ERK1 110 3
DAPK1 110 15
NEK6 110 4
MEKK1 111 11
AMPK 111 17
TTBK1 111 3
CLK2 111 1
IR 111 6
PRK2 111 16
PAK6 111 2
DYRK1A 112 2
MARK3 112 1
PKC gamma 112 1
GCK 113 3
RSK1 113 4
RSK2 113 1
MAPKAP-K3 113 6
EIF2AK3 113 7
CAMKK beta 113 16
DYRK3 113 14
IRAK1 113 7
p38 gamma MAPK 113 1
SRPK1 114 20
LKB1 114 10
TAO1 114 6
MARK4 114 4
JAK2 114 8
CDK2-Cyclin A 114 19
PLK1 115 23
HIPK1 115 13
MLK1 115 9
EPH-B4 115 6
SGK1 115 2
HER4 115 22
TAK1 115 1
FGF-R1 116 20
EPH-B1 117 17
HIPK2 117 4
TESK1 117 18
BTK 117 26
SYK 117 7
RIPK2 117 9
STK33 118 15
MARK1 118 2
EPH-A2 119 11
Aurora B 119 8
PAK2 119 12
p38 beta MAPK 119 25
PDK1 120 6
JNK2 120 6
JNK3 120 16
MST2 120 2
SIK2 121 1
SIK3 121 14
ULK1 121 4
MAP4K3 122 22
MKK6 122 22
TGFBR1 123 13
ROCK 2 123 3
NUAK1 123 22
IGF-1R 126 30
PKC zeta 126 19
EF2K 127 15
Src 127 13
GSK3 beta 127 12
CHK2 128 24
PKD1 133 19

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