Kinase Profiling Inhibitor Database

Inhibitor Structure Image Brutto MW Action Reference Reference 2 Patent Commercial Vendor Notes Results
2-Aminopurine C5H5N5 135.1267 PKR Sigma Download

Results as Barchart

View results as a bar chart
100µM

Results as Table

Screening Concentration: 100µM
Kinase % Activity Remainingsort ascending Standard Deviation
PIM1 122 0
FGF-R1 109 18
EPH-B1 108 7
TLK1 108 7
IR 106 8
EPH-B3 105 36
HIPK1 104 15
PKC alpha 104 27
SYK 102 8
PIM2 102 7
ZAP70 101 4
TGFBR1 101 2
PAK2 100 10
PKB alpha 99 5
p38 delta MAPK 97 6
SRPK1 96 1
EPH-B2 95 10
YES1 94 6
PKA 93 7
HIPK3 92 2
MKK6 91 6
CSK 91 17
EPH-B4 90 10
PINK 90 11
GSK3 beta 89 12
MPSK1 89 4
CK2 89 5
EIF2AK3 89 0
NEK6 88 10
EF2K 88 3
CAMKK beta 87 1
WNK1 87 2
S6K1 85 15
CAMK1 85 5
p38 alpha MAPK 85 4
TIE2 85 1
PKC gamma 84 6
MSK1 84 4
EPH-A4 84 4
PKB beta 83 7
ABL 83 7
JNK2 83 8
JNK3 83 6
p38 beta MAPK 83 0
EPH-A2 83 1
PAK6 82 5
DDR2 82 11
TTK 82 1
LKB1 82 9
JNK1 81 6
BRSK2 81 3
CDK2-Cyclin A 81 2
MST3 81 2
RSK1 81 2
TTBK1 80 12
AMPK (hum) 80 11
OSR1 80 7
Lck 79 3
BRSK1 79 8
PDGFRA 79 3
ERK8 79 10
RSK2 79 8
ERK1 78 8
ERK2 78 0
PKC zeta 78 3
MEKK1 78 0
DAPK1 77 7
HIPK2 76 2
PHK 76 2
IRAK4 76 7
PLK1 76 1
PIM3 76 4
PRAK 75 0
SmMLCK 75 2
IGF-1R 75 23
p38 gamma MAPK 75 0
MNK2 75 2
TTBK2 74 6
MARK4 74 5
AMPK 73 6
Src 73 1
PRK2 73 8
IRR 73 5
TrkA 73 13
TBK1 73 4
HER4 72 0
DYRK3 72 5
CDK9-Cyclin T1 72 9
MST4 72 3
MAPKAP-K3 70 3
MARK2 69 2
ULK2 69 0
DYRK2 68 6
MARK1 67 0
ERK5 67 1
BTK 67 3
STK33 67 6
MNK1 67 7
MAP4K5 67 3
PDK1 67 1
TAO1 66 3
IRAK1 65 10
PKD1 65 7
DYRK1A 64 3
ROCK 2 64 2
PAK5 64 0
Aurora A 64 3
SGK1 63 1
MELK 63 2
MST2 63 1
MINK1 63 3
MKK2 63 2
IKK epsilon 62 5
MARK3 61 5
TESK1 60 4
NEK2a 60 14
CHK1 57 9
ULK1 57 2
SIK3 56 2
MKK1 56 5
IKK beta 55 4
TAK1 54 2
MAP4K3 50 6
BRK 47 5
ASK1 44 3
PAK4 44 5
TSSK1 44 8
RIPK2 43 1
SIK2 43 2
MAPKAP-K2 40 3
CLK2 37 4
NUAK1 33 0
JAK2 30 0
MLK1 29 6
VEGFR1 29 3
CK1 delta 24 4
Aurora B 23 2
CHK2 21 0
GCK 20 0
MLK3 18 5
CK1 gamma 2 16 1

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