Kinase Profiling Inhibitor Database

Inhibitor Structure Image Brutto MW Action Reference Reference 2 Patent Commercial Vendor Notes Results
Ischemin C15H17N3O4S 335.38 p53 CBP Jagat C. Borah (2011) Chemistry & Biology, 18 4 531-541 Download

Results as Barchart

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100µM

Results as Table

Screening Concentration: 100µM
Kinase % Activity Remaining Standard Deviation
MKK1 103 8
MKK2 109 3
MKK6 113 8
ERK1 98 8
ERK2 134 0
JNK1 113 0
JNK2 112 2
JNK3 100 9
p38 alpha MAPK 58 2
p38 beta MAPK 58 5
p38 gamma MAPK 108 3
p38 delta MAPK 109 8
ERK8 65 8
RSK1 99 2
RSK2 80 1
PDK1 90 1
PKB alpha 108 10
PKB beta 37 7
SGK1 52 5
S6K1 102 1
PKA 90 2
ROCK 2 105 0
PRK2 126 6
PKC alpha 81 4
PKC gamma 55 9
PKC zeta 97 6
PKD1 55 11
STK33 107 14
MSK1 84 8
MNK1 99 5
MNK2 100 3
MAPKAP-K2 107 8
MAPKAP-K3 62 7
PRAK 70 8
CAMKK beta 99 2
CAMK1 45 1
SmMLCK 97 7
PHK 86 4
DAPK1 82 3
CHK1 196 6
CHK2 100 1
GSK3 beta 31 3
CDK2-Cyclin A 94 8
PLK1 79 8
Aurora A 32 5
Aurora B 93 3
TLK1 108 0
LKB1 126 1
AMPK 71 2
MARK1 99 1
MARK2 98 2
MARK3 96 9
MARK4 81 7
BRSK1 76 1
BRSK2 46 5
MELK 87 9
NUAK1 44 7
TSSK1 107 2
CK1 delta 108 24
CK2 51 0
TTBK1 94 13
DYRK1A 113 7
DYRK2 78 1
DYRK3 65 4
NEK2a 118 6
NEK6 146 63
IKK beta 97 12
IKK epsilon 94 1
TBK1 94 1
PIM1 62 2
PIM2 58 0
PIM3 45 7
SRPK1 59 4
EF2K 92 7
EIF2AK3 94 1
HIPK1 94 6
HIPK2 42 14
HIPK3 74 8
CLK2 101 28
PAK2 100 4
PAK4 70 6
PAK5 87 9
PAK6 96 12
MST2 81 6
MST4 67 0
GCK 80 0
MINK1 62 7
MEKK1 88 16
MLK1 58 12
MLK3 83 7
TESK1 73 2
TAO1 109 3
ASK1 151 9
TAK1 31 5
IRAK1 104 3
IRAK4 108 20
RIPK2 46 4
OSR1 97 4
TTK 90 4
MPSK1 111 5
Src 40 2
Lck 112 1
CSK 132 11
YES1 52 8
ABL 92 1
BTK 102 8
JAK2 71 4
SYK 103 8
ZAP70 103 3
TIE2 103 1
BRK 100 4
EPH-A2 89 6
EPH-A4 92 5
EPH-B1 97 7
EPH-B2 96 9
EPH-B3 48 3
EPH-B4 123 8
FGF-R1 59 6
HER4 99 7
IGF-1R 109 2
IR 141 8
IRR 103 13
TrkA 65 4
VEGFR1 62 0

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