InhibitorScreening ConcentrationKinase% Activity RemainingStandard Deviation
Merck 7 (PDK1)0.10µMMKK110016
Merck 7 (PDK1)0.10µMMKK212113
Merck 7 (PDK1)0.10µMMKK6946
Merck 7 (PDK1)0.10µMERK1935
Merck 7 (PDK1)0.10µMERK21021
Merck 7 (PDK1)0.10µMJNK110010
Merck 7 (PDK1)0.10µMJNK2939
Merck 7 (PDK1)0.10µMJNK31014
Merck 7 (PDK1)0.10µMp38 alpha MAPK1147
Merck 7 (PDK1)0.10µMp38 beta MAPK1001
Merck 7 (PDK1)0.10µMp38 gamma MAPK981
Merck 7 (PDK1)0.10µMp38 delta MAPK9112
Merck 7 (PDK1)0.10µMERK8921
Merck 7 (PDK1)0.10µMRSK19517
Merck 7 (PDK1)0.10µMRSK21025
Merck 7 (PDK1)0.10µMPDK19010
Merck 7 (PDK1)0.10µMPKB alpha 964
Merck 7 (PDK1)0.10µMPKB beta 984
Merck 7 (PDK1)0.10µMSGK11062
Merck 7 (PDK1)0.10µMS6K11031
Merck 7 (PDK1)0.10µMPKA1051
Merck 7 (PDK1)0.10µMROCK 21058
Merck 7 (PDK1)0.10µMPRK21083
Merck 7 (PDK1)0.10µMPKC alpha 995
Merck 7 (PDK1)0.10µMPKC gamma 910
Merck 7 (PDK1)0.10µMPKC zeta 1045
Merck 7 (PDK1)0.10µMPKD19010
Merck 7 (PDK1)0.10µMSTK339213
Merck 7 (PDK1)0.10µMMSK11015
Merck 7 (PDK1)0.10µMMNK11068
Merck 7 (PDK1)0.10µMMNK211711
Merck 7 (PDK1)0.10µMMAPKAP-K2 999
Merck 7 (PDK1)0.10µMMAPKAP-K31161
Merck 7 (PDK1)0.10µMPRAK10811
Merck 7 (PDK1)0.10µMCAMKK beta 11930
Merck 7 (PDK1)0.10µMCAMK1959
Merck 7 (PDK1)0.10µMSmMLCK972
Merck 7 (PDK1)0.10µMPHK1004
Merck 7 (PDK1)0.10µMDAPK110618
Merck 7 (PDK1)0.10µMCHK1964
Merck 7 (PDK1)0.10µMCHK210210
Merck 7 (PDK1)0.10µMGSK3 beta 978
Merck 7 (PDK1)0.10µMCDK2-Cyclin A901
Merck 7 (PDK1)0.10µMPLK111814
Merck 7 (PDK1)0.10µMAurora A1106
Merck 7 (PDK1)0.10µMAurora B10516
Merck 7 (PDK1)0.10µMTLK1972
Merck 7 (PDK1)0.10µMLKB11023
Merck 7 (PDK1)0.10µMAMPK979
Merck 7 (PDK1)0.10µMMARK111120
Merck 7 (PDK1)0.10µMMARK21055
Merck 7 (PDK1)0.10µMMARK39912
Merck 7 (PDK1)0.10µMMARK41503
Merck 7 (PDK1)0.10µMBRSK11181
Merck 7 (PDK1)0.10µMBRSK211818
Merck 7 (PDK1)0.10µMMELK9717
Merck 7 (PDK1)0.10µMNUAK111512
Merck 7 (PDK1)0.10µMTSSK1934
Merck 7 (PDK1)0.10µMCK1 delta 1039
Merck 7 (PDK1)0.10µMCK21111
Merck 7 (PDK1)0.10µMTTBK110110
Merck 7 (PDK1)0.10µMDYRK1A1134
Merck 7 (PDK1)0.10µMDYRK21101
Merck 7 (PDK1)0.10µMDYRK31099
Merck 7 (PDK1)0.10µMNEK2a1073
Merck 7 (PDK1)0.10µMNEK61042
Merck 7 (PDK1)0.10µMIKK beta 1020
Merck 7 (PDK1)0.10µMIKK epsilon 10311
Merck 7 (PDK1)0.10µMTBK110916
Merck 7 (PDK1)0.10µMPIM11014
Merck 7 (PDK1)0.10µMPIM21076
Merck 7 (PDK1)0.10µMPIM31034
Merck 7 (PDK1)0.10µMSRPK11071
Merck 7 (PDK1)0.10µMEF2K9511
Merck 7 (PDK1)0.10µMEIF2AK31079
Merck 7 (PDK1)0.10µMHIPK1994
Merck 7 (PDK1)0.10µMHIPK29211
Merck 7 (PDK1)0.10µMHIPK3990
Merck 7 (PDK1)0.10µMCLK21066
Merck 7 (PDK1)0.10µMPAK211311
Merck 7 (PDK1)0.10µMPAK410214
Merck 7 (PDK1)0.10µMPAK51045
Merck 7 (PDK1)0.10µMPAK61022
Merck 7 (PDK1)0.10µMMST21027
Merck 7 (PDK1)0.10µMMST41012
Merck 7 (PDK1)0.10µMGCK1027
Merck 7 (PDK1)0.10µMMINK1921
Merck 7 (PDK1)0.10µMMEKK111012
Merck 7 (PDK1)0.10µMMLK111916
Merck 7 (PDK1)0.10µMMLK310416
Merck 7 (PDK1)0.10µMTESK19811
Merck 7 (PDK1)0.10µMTAO11116
Merck 7 (PDK1)0.10µMASK11106
Merck 7 (PDK1)0.10µMTAK1978
Merck 7 (PDK1)0.10µMIRAK11178
Merck 7 (PDK1)0.10µMIRAK41107
Merck 7 (PDK1)0.10µMRIPK21022
Merck 7 (PDK1)0.10µMOSR1975
Merck 7 (PDK1)0.10µMTTK990
Merck 7 (PDK1)0.10µMMPSK11019
Merck 7 (PDK1)0.10µMSrc10313
Merck 7 (PDK1)0.10µMLck1099
Merck 7 (PDK1)0.10µMCSK10913
Merck 7 (PDK1)0.10µMYES110412
Merck 7 (PDK1)0.10µMABL1060
Merck 7 (PDK1)0.10µMBTK1091
Merck 7 (PDK1)0.10µMJAK2981
Merck 7 (PDK1)0.10µMSYK9910
Merck 7 (PDK1)0.10µMZAP701021
Merck 7 (PDK1)0.10µMTIE21044
Merck 7 (PDK1)0.10µMBRK12015
Merck 7 (PDK1)0.10µMEPH-A29429
Merck 7 (PDK1)0.10µMEPH-A4952
Merck 7 (PDK1)0.10µMEPH-B1870
Merck 7 (PDK1)0.10µMEPH-B21182
Merck 7 (PDK1)0.10µMEPH-B31141
Merck 7 (PDK1)0.10µMEPH-B49524
Merck 7 (PDK1)0.10µMFGF-R1965
Merck 7 (PDK1)0.10µMHER41027
Merck 7 (PDK1)0.10µMIGF-1R1054
Merck 7 (PDK1)0.10µMIR994
Merck 7 (PDK1)0.10µMIRR1014
Merck 7 (PDK1)0.10µMTrkA1132
Merck 7 (PDK1)0.10µMVEGFR11062
Merck 7 (PDK1)1.00µMMKK111132
Merck 7 (PDK1)1.00µMMKK21244
Merck 7 (PDK1)1.00µMMKK6896
Merck 7 (PDK1)1.00µMERK11016
Merck 7 (PDK1)1.00µMERK21007
Merck 7 (PDK1)1.00µMJNK110820
Merck 7 (PDK1)1.00µMJNK2976
Merck 7 (PDK1)1.00µMJNK3904
Merck 7 (PDK1)1.00µMp38 alpha MAPK1217
Merck 7 (PDK1)1.00µMp38 beta MAPK11018
Merck 7 (PDK1)1.00µMp38 gamma MAPK1100
Merck 7 (PDK1)1.00µMp38 delta MAPK974
Merck 7 (PDK1)1.00µMERK8898
Merck 7 (PDK1)1.00µMRSK1933
Merck 7 (PDK1)1.00µMRSK2988
Merck 7 (PDK1)1.00µMPDK13810
Merck 7 (PDK1)1.00µMPKB alpha 971
Merck 7 (PDK1)1.00µMPKB beta 9610
Merck 7 (PDK1)1.00µMSGK11022
Merck 7 (PDK1)1.00µMS6K19710
Merck 7 (PDK1)1.00µMPKA1127
Merck 7 (PDK1)1.00µMROCK 21127
Merck 7 (PDK1)1.00µMPRK211314
Merck 7 (PDK1)1.00µMPKC alpha 9111
Merck 7 (PDK1)1.00µMPKC gamma 10311
Merck 7 (PDK1)1.00µMPKC zeta 10613
Merck 7 (PDK1)1.00µMPKD18014
Merck 7 (PDK1)1.00µMSTK3310711
Merck 7 (PDK1)1.00µMMSK11048
Merck 7 (PDK1)1.00µMMNK1991
Merck 7 (PDK1)1.00µMMNK212341
Merck 7 (PDK1)1.00µMMAPKAP-K2 10114
Merck 7 (PDK1)1.00µMMAPKAP-K31097
Merck 7 (PDK1)1.00µMPRAK1004
Merck 7 (PDK1)1.00µMCAMKK beta 1048
Merck 7 (PDK1)1.00µMCAMK1921
Merck 7 (PDK1)1.00µMSmMLCK9714
Merck 7 (PDK1)1.00µMPHK11719
Merck 7 (PDK1)1.00µMDAPK11134
Merck 7 (PDK1)1.00µMCHK1940
Merck 7 (PDK1)1.00µMCHK21067
Merck 7 (PDK1)1.00µMGSK3 beta 9616
Merck 7 (PDK1)1.00µMCDK2-Cyclin A916
Merck 7 (PDK1)1.00µMPLK11079
Merck 7 (PDK1)1.00µMAurora A1101
Merck 7 (PDK1)1.00µMAurora B1049
Merck 7 (PDK1)1.00µMTLK110318
Merck 7 (PDK1)1.00µMLKB110011
Merck 7 (PDK1)1.00µMAMPK997
Merck 7 (PDK1)1.00µMMARK110820
Merck 7 (PDK1)1.00µMMARK210210
Merck 7 (PDK1)1.00µMMARK39311
Merck 7 (PDK1)1.00µMMARK41433
Merck 7 (PDK1)1.00µMBRSK110213
Merck 7 (PDK1)1.00µMBRSK2904
Merck 7 (PDK1)1.00µMMELK1109
Merck 7 (PDK1)1.00µMNUAK11077
Merck 7 (PDK1)1.00µMTSSK11036
Merck 7 (PDK1)1.00µMCK1 delta 1108
Merck 7 (PDK1)1.00µMCK210312
Merck 7 (PDK1)1.00µMTTBK11104
Merck 7 (PDK1)1.00µMDYRK1A978
Merck 7 (PDK1)1.00µMDYRK21015
Merck 7 (PDK1)1.00µMDYRK31092
Merck 7 (PDK1)1.00µMNEK2a978
Merck 7 (PDK1)1.00µMNEK61006
Merck 7 (PDK1)1.00µMIKK beta 997
Merck 7 (PDK1)1.00µMIKK epsilon 1097
Merck 7 (PDK1)1.00µMTBK113213
Merck 7 (PDK1)1.00µMPIM11052
Merck 7 (PDK1)1.00µMPIM21055
Merck 7 (PDK1)1.00µMPIM310811
Merck 7 (PDK1)1.00µMSRPK111412
Merck 7 (PDK1)1.00µMEF2K10318
Merck 7 (PDK1)1.00µMEIF2AK31042
Merck 7 (PDK1)1.00µMHIPK11003
Merck 7 (PDK1)1.00µMHIPK2969
Merck 7 (PDK1)1.00µMHIPK31084
Merck 7 (PDK1)1.00µMCLK29518
Merck 7 (PDK1)1.00µMPAK21092
Merck 7 (PDK1)1.00µMPAK41010
Merck 7 (PDK1)1.00µMPAK5927
Merck 7 (PDK1)1.00µMPAK61024
Merck 7 (PDK1)1.00µMMST21054
Merck 7 (PDK1)1.00µMMST41178
Merck 7 (PDK1)1.00µMGCK1016
Merck 7 (PDK1)1.00µMMINK11001
Merck 7 (PDK1)1.00µMMEKK11147
Merck 7 (PDK1)1.00µMMLK11023
Merck 7 (PDK1)1.00µMMLK3973
Merck 7 (PDK1)1.00µMTESK1884
Merck 7 (PDK1)1.00µMTAO11261
Merck 7 (PDK1)1.00µMASK110515
Merck 7 (PDK1)1.00µMTAK11035
Merck 7 (PDK1)1.00µMIRAK11182
Merck 7 (PDK1)1.00µMIRAK410922
Merck 7 (PDK1)1.00µMRIPK21059
Merck 7 (PDK1)1.00µMOSR1960
Merck 7 (PDK1)1.00µMTTK10011
Merck 7 (PDK1)1.00µMMPSK111817
Merck 7 (PDK1)1.00µMSrc1003
Merck 7 (PDK1)1.00µMLck1017
Merck 7 (PDK1)1.00µMCSK986
Merck 7 (PDK1)1.00µMYES110512
Merck 7 (PDK1)1.00µMABL1054
Merck 7 (PDK1)1.00µMBTK1081
Merck 7 (PDK1)1.00µMJAK2992
Merck 7 (PDK1)1.00µMSYK884
Merck 7 (PDK1)1.00µMZAP701063
Merck 7 (PDK1)1.00µMTIE210010
Merck 7 (PDK1)1.00µMBRK12910
Merck 7 (PDK1)1.00µMEPH-A21023
Merck 7 (PDK1)1.00µMEPH-A411319
Merck 7 (PDK1)1.00µMEPH-B1884
Merck 7 (PDK1)1.00µMEPH-B211521
Merck 7 (PDK1)1.00µMEPH-B31197
Merck 7 (PDK1)1.00µMEPH-B48518
Merck 7 (PDK1)1.00µMFGF-R1972
Merck 7 (PDK1)1.00µMHER41006
Merck 7 (PDK1)1.00µMIGF-1R1053
Merck 7 (PDK1)1.00µMIR954
Merck 7 (PDK1)1.00µMIRR1145
Merck 7 (PDK1)1.00µMTrkA985
Merck 7 (PDK1)1.00µMVEGFR11003
Merck 7 (PDK1)10.00µMMKK1951
Merck 7 (PDK1)10.00µMMKK21351
Merck 7 (PDK1)10.00µMMKK610817
Merck 7 (PDK1)10.00µMERK1951
Merck 7 (PDK1)10.00µMERK21012
Merck 7 (PDK1)10.00µMJNK111417
Merck 7 (PDK1)10.00µMJNK2958
Merck 7 (PDK1)10.00µMJNK31014
Merck 7 (PDK1)10.00µMp38 alpha MAPK11411
Merck 7 (PDK1)10.00µMp38 beta MAPK1159
Merck 7 (PDK1)10.00µMp38 gamma MAPK1051
Merck 7 (PDK1)10.00µMp38 delta MAPK942
Merck 7 (PDK1)10.00µMERK8942
Merck 7 (PDK1)10.00µMRSK11141
Merck 7 (PDK1)10.00µMRSK2851
Merck 7 (PDK1)10.00µMPDK171
Merck 7 (PDK1)10.00µMPKB alpha 9016
Merck 7 (PDK1)10.00µMPKB beta 7713
Merck 7 (PDK1)10.00µMSGK11025
Merck 7 (PDK1)10.00µMS6K1983
Merck 7 (PDK1)10.00µMPKA1114
Merck 7 (PDK1)10.00µMROCK 210814
Merck 7 (PDK1)10.00µMPRK21036
Merck 7 (PDK1)10.00µMPKC alpha 967
Merck 7 (PDK1)10.00µMPKC gamma 10231
Merck 7 (PDK1)10.00µMPKC zeta 8810
Merck 7 (PDK1)10.00µMPKD1754
Merck 7 (PDK1)10.00µMSTK337910
Merck 7 (PDK1)10.00µMMSK11061
Merck 7 (PDK1)10.00µMMNK1994
Merck 7 (PDK1)10.00µMMNK211214
Merck 7 (PDK1)10.00µMMAPKAP-K2 9014
Merck 7 (PDK1)10.00µMMAPKAP-K3744
Merck 7 (PDK1)10.00µMPRAK955
Merck 7 (PDK1)10.00µMCAMKK beta 902
Merck 7 (PDK1)10.00µMCAMK1515
Merck 7 (PDK1)10.00µMSmMLCK894
Merck 7 (PDK1)10.00µMPHK11922
Merck 7 (PDK1)10.00µMDAPK1915
Merck 7 (PDK1)10.00µMCHK19519
Merck 7 (PDK1)10.00µMCHK21004
Merck 7 (PDK1)10.00µMGSK3 beta 6412
Merck 7 (PDK1)10.00µMCDK2-Cyclin A9512
Merck 7 (PDK1)10.00µMPLK11212
Merck 7 (PDK1)10.00µMAurora A1032
Merck 7 (PDK1)10.00µMAurora B6412
Merck 7 (PDK1)10.00µMTLK1994
Merck 7 (PDK1)10.00µMLKB1931
Merck 7 (PDK1)10.00µMAMPK9911
Merck 7 (PDK1)10.00µMMARK11076
Merck 7 (PDK1)10.00µMMARK2885
Merck 7 (PDK1)10.00µMMARK38311
Merck 7 (PDK1)10.00µMMARK4834
Merck 7 (PDK1)10.00µMBRSK19214
Merck 7 (PDK1)10.00µMBRSK2795
Merck 7 (PDK1)10.00µMMELK992
Merck 7 (PDK1)10.00µMNUAK19816
Merck 7 (PDK1)10.00µMTSSK1869
Merck 7 (PDK1)10.00µMCK1 delta 11310
Merck 7 (PDK1)10.00µMCK210713
Merck 7 (PDK1)10.00µMTTBK11067
Merck 7 (PDK1)10.00µMDYRK1A794
Merck 7 (PDK1)10.00µMDYRK2839
Merck 7 (PDK1)10.00µMDYRK3934
Merck 7 (PDK1)10.00µMNEK2a9611
Merck 7 (PDK1)10.00µMNEK69811
Merck 7 (PDK1)10.00µMIKK beta 994
Merck 7 (PDK1)10.00µMIKK epsilon 955
Merck 7 (PDK1)10.00µMTBK110217
Merck 7 (PDK1)10.00µMPIM1762
Merck 7 (PDK1)10.00µMPIM2854
Merck 7 (PDK1)10.00µMPIM39510
Merck 7 (PDK1)10.00µMSRPK110110
Merck 7 (PDK1)10.00µMEF2K10711
Merck 7 (PDK1)10.00µMEIF2AK3962
Merck 7 (PDK1)10.00µMHIPK1860
Merck 7 (PDK1)10.00µMHIPK29015
Merck 7 (PDK1)10.00µMHIPK3910
Merck 7 (PDK1)10.00µMCLK2741
Merck 7 (PDK1)10.00µMPAK2796
Merck 7 (PDK1)10.00µMPAK4670
Merck 7 (PDK1)10.00µMPAK5643
Merck 7 (PDK1)10.00µMPAK6890
Merck 7 (PDK1)10.00µMMST210010
Merck 7 (PDK1)10.00µMMST48617
Merck 7 (PDK1)10.00µMGCK941
Merck 7 (PDK1)10.00µMMINK18717
Merck 7 (PDK1)10.00µMMEKK11122
Merck 7 (PDK1)10.00µMMLK1503
Merck 7 (PDK1)10.00µMMLK3463
Merck 7 (PDK1)10.00µMTESK11076
Merck 7 (PDK1)10.00µMTAO11194
Merck 7 (PDK1)10.00µMASK1926
Merck 7 (PDK1)10.00µMTAK1544
Merck 7 (PDK1)10.00µMIRAK11086
Merck 7 (PDK1)10.00µMIRAK411026
Merck 7 (PDK1)10.00µMRIPK2987
Merck 7 (PDK1)10.00µMOSR1833
Merck 7 (PDK1)10.00µMTTK950
Merck 7 (PDK1)10.00µMMPSK11063
Merck 7 (PDK1)10.00µMSrc753
Merck 7 (PDK1)10.00µMLck9111
Merck 7 (PDK1)10.00µMCSK1019
Merck 7 (PDK1)10.00µMYES1955
Merck 7 (PDK1)10.00µMABL984
Merck 7 (PDK1)10.00µMBTK11016
Merck 7 (PDK1)10.00µMJAK21012
Merck 7 (PDK1)10.00µMSYK828
Merck 7 (PDK1)10.00µMZAP7012830
Merck 7 (PDK1)10.00µMTIE2966
Merck 7 (PDK1)10.00µMBRK1190
Merck 7 (PDK1)10.00µMEPH-A28614
Merck 7 (PDK1)10.00µMEPH-A41074
Merck 7 (PDK1)10.00µMEPH-B1904
Merck 7 (PDK1)10.00µMEPH-B212117
Merck 7 (PDK1)10.00µMEPH-B311318
Merck 7 (PDK1)10.00µMEPH-B48716
Merck 7 (PDK1)10.00µMFGF-R17510
Merck 7 (PDK1)10.00µMHER49813
Merck 7 (PDK1)10.00µMIGF-1R1034
Merck 7 (PDK1)10.00µMIR9317
Merck 7 (PDK1)10.00µMIRR10514
Merck 7 (PDK1)10.00µMTrkA7819
Merck 7 (PDK1)10.00µMVEGFR111225