InhibitorScreening ConcentrationKinase% Activity RemainingStandard Deviation
CP-690550 (Tasocitinib)0.10µMMKK11056
CP-690550 (Tasocitinib)0.10µMMKK21103
CP-690550 (Tasocitinib)0.10µMMKK6978
CP-690550 (Tasocitinib)0.10µMERK1974
CP-690550 (Tasocitinib)0.10µMERK29710
CP-690550 (Tasocitinib)0.10µMJNK1803
CP-690550 (Tasocitinib)0.10µMJNK2944
CP-690550 (Tasocitinib)0.10µMJNK311912
CP-690550 (Tasocitinib)0.10µMp38 alpha MAPK1001
CP-690550 (Tasocitinib)0.10µMp38 beta MAPK10612
CP-690550 (Tasocitinib)0.10µMp38 gamma MAPK1156
CP-690550 (Tasocitinib)0.10µMp38 delta MAPK1017
CP-690550 (Tasocitinib)0.10µMERK81216
CP-690550 (Tasocitinib)0.10µMRSK1966
CP-690550 (Tasocitinib)0.10µMRSK2913
CP-690550 (Tasocitinib)0.10µMPDK110714
CP-690550 (Tasocitinib)0.10µMPKB alpha 1151
CP-690550 (Tasocitinib)0.10µMPKB beta 859
CP-690550 (Tasocitinib)0.10µMSGK1922
CP-690550 (Tasocitinib)0.10µMS6K1880
CP-690550 (Tasocitinib)0.10µMPKA944
CP-690550 (Tasocitinib)0.10µMROCK 29515
CP-690550 (Tasocitinib)0.10µMPRK2502
CP-690550 (Tasocitinib)0.10µMPKC alpha 960
CP-690550 (Tasocitinib)0.10µMPKC gamma 10021
CP-690550 (Tasocitinib)0.10µMPKC zeta 9911
CP-690550 (Tasocitinib)0.10µMPKD1924
CP-690550 (Tasocitinib)0.10µMSTK33984
CP-690550 (Tasocitinib)0.10µMMSK18310
CP-690550 (Tasocitinib)0.10µMMNK110011
CP-690550 (Tasocitinib)0.10µMMNK2972
CP-690550 (Tasocitinib)0.10µMMAPKAP-K2 827
CP-690550 (Tasocitinib)0.10µMMAPKAP-K3914
CP-690550 (Tasocitinib)0.10µMPRAK11310
CP-690550 (Tasocitinib)0.10µMCAMKK beta 11610
CP-690550 (Tasocitinib)0.10µMCAMK11112
CP-690550 (Tasocitinib)0.10µMSmMLCK1053
CP-690550 (Tasocitinib)0.10µMPHK962
CP-690550 (Tasocitinib)0.10µMDAPK112311
CP-690550 (Tasocitinib)0.10µMCHK1881
CP-690550 (Tasocitinib)0.10µMCHK2959
CP-690550 (Tasocitinib)0.10µMGSK3 beta 1089
CP-690550 (Tasocitinib)0.10µMCDK2-Cyclin A11637
CP-690550 (Tasocitinib)0.10µMPLK11287
CP-690550 (Tasocitinib)0.10µMAurora A11916
CP-690550 (Tasocitinib)0.10µMAurora B928
CP-690550 (Tasocitinib)0.10µMTLK11003
CP-690550 (Tasocitinib)0.10µMLKB11019
CP-690550 (Tasocitinib)0.10µMAMPK955
CP-690550 (Tasocitinib)0.10µMMARK18210
CP-690550 (Tasocitinib)0.10µMMARK2981
CP-690550 (Tasocitinib)0.10µMMARK39416
CP-690550 (Tasocitinib)0.10µMMARK4932
CP-690550 (Tasocitinib)0.10µMBRSK1927
CP-690550 (Tasocitinib)0.10µMBRSK21013
CP-690550 (Tasocitinib)0.10µMMELK11512
CP-690550 (Tasocitinib)0.10µMNUAK1745
CP-690550 (Tasocitinib)0.10µMCK1 delta 1099
CP-690550 (Tasocitinib)0.10µMCK2977
CP-690550 (Tasocitinib)0.10µMDYRK1A927
CP-690550 (Tasocitinib)0.10µMDYRK21035
CP-690550 (Tasocitinib)0.10µMDYRK31162
CP-690550 (Tasocitinib)0.10µMNEK2a10216
CP-690550 (Tasocitinib)0.10µMNEK6873
CP-690550 (Tasocitinib)0.10µMIKK beta 1052
CP-690550 (Tasocitinib)0.10µMIKK epsilon 878
CP-690550 (Tasocitinib)0.10µMTBK1996
CP-690550 (Tasocitinib)0.10µMPIM11125
CP-690550 (Tasocitinib)0.10µMPIM21025
CP-690550 (Tasocitinib)0.10µMPIM312412
CP-690550 (Tasocitinib)0.10µMSRPK1846
CP-690550 (Tasocitinib)0.10µMEF2K1002
CP-690550 (Tasocitinib)0.10µMEIF2AK3979
CP-690550 (Tasocitinib)0.10µMHIPK11124
CP-690550 (Tasocitinib)0.10µMHIPK21176
CP-690550 (Tasocitinib)0.10µMHIPK31083
CP-690550 (Tasocitinib)0.10µMCLK21081
CP-690550 (Tasocitinib)0.10µMPAK2992
CP-690550 (Tasocitinib)0.10µMPAK410410
CP-690550 (Tasocitinib)0.10µMPAK5867
CP-690550 (Tasocitinib)0.10µMPAK61003
CP-690550 (Tasocitinib)0.10µMMST2797
CP-690550 (Tasocitinib)0.10µMMST4878
CP-690550 (Tasocitinib)0.10µMGCK1097
CP-690550 (Tasocitinib)0.10µMMINK1967
CP-690550 (Tasocitinib)0.10µMMEKK1977
CP-690550 (Tasocitinib)0.10µMMLK1865
CP-690550 (Tasocitinib)0.10µMMLK38312
CP-690550 (Tasocitinib)0.10µMTAO110412
CP-690550 (Tasocitinib)0.10µMASK113011
CP-690550 (Tasocitinib)0.10µMTAK11157
CP-690550 (Tasocitinib)0.10µMIRAK11063
CP-690550 (Tasocitinib)0.10µMIRAK4870
CP-690550 (Tasocitinib)0.10µMRIPK2919
CP-690550 (Tasocitinib)0.10µMOSR11129
CP-690550 (Tasocitinib)0.10µMTTK993
CP-690550 (Tasocitinib)0.10µMMPSK19410
CP-690550 (Tasocitinib)0.10µMSrc925
CP-690550 (Tasocitinib)0.10µMLck739
CP-690550 (Tasocitinib)0.10µMCSK783
CP-690550 (Tasocitinib)0.10µMYES11043
CP-690550 (Tasocitinib)0.10µMABL11610
CP-690550 (Tasocitinib)0.10µMBTK9411
CP-690550 (Tasocitinib)0.10µMJAK240
CP-690550 (Tasocitinib)0.10µMSYK1317
CP-690550 (Tasocitinib)0.10µMZAP701330
CP-690550 (Tasocitinib)0.10µMTIE2991
CP-690550 (Tasocitinib)0.10µMBRK927
CP-690550 (Tasocitinib)0.10µMEPH-A211419
CP-690550 (Tasocitinib)0.10µMEPH-A41093
CP-690550 (Tasocitinib)0.10µMEPH-B1934
CP-690550 (Tasocitinib)0.10µMEPH-B212112
CP-690550 (Tasocitinib)0.10µMEPH-B3855
CP-690550 (Tasocitinib)0.10µMEPH-B41204
CP-690550 (Tasocitinib)0.10µMFGF-R1853
CP-690550 (Tasocitinib)0.10µMHER412119
CP-690550 (Tasocitinib)0.10µMIGF-1R10411
CP-690550 (Tasocitinib)0.10µMIR1059
CP-690550 (Tasocitinib)0.10µMIRR1035
CP-690550 (Tasocitinib)0.10µMTrkA10613
CP-690550 (Tasocitinib)0.10µMVEGFR1995
CP-690550 (Tasocitinib)1.00µMMKK1676
CP-690550 (Tasocitinib)1.00µMMKK211220
CP-690550 (Tasocitinib)1.00µMMKK6892
CP-690550 (Tasocitinib)1.00µMERK11085
CP-690550 (Tasocitinib)1.00µMERK29917
CP-690550 (Tasocitinib)1.00µMJNK1815
CP-690550 (Tasocitinib)1.00µMJNK2889
CP-690550 (Tasocitinib)1.00µMJNK310710
CP-690550 (Tasocitinib)1.00µMp38 alpha MAPK1034
CP-690550 (Tasocitinib)1.00µMp38 beta MAPK1153
CP-690550 (Tasocitinib)1.00µMp38 gamma MAPK1309
CP-690550 (Tasocitinib)1.00µMp38 delta MAPK10817
CP-690550 (Tasocitinib)1.00µMERK81211
CP-690550 (Tasocitinib)1.00µMRSK17623
CP-690550 (Tasocitinib)1.00µMRSK2862
CP-690550 (Tasocitinib)1.00µMPDK11233
CP-690550 (Tasocitinib)1.00µMPKB alpha 1254
CP-690550 (Tasocitinib)1.00µMPKB beta 926
CP-690550 (Tasocitinib)1.00µMSGK110619
CP-690550 (Tasocitinib)1.00µMS6K17716
CP-690550 (Tasocitinib)1.00µMPKA891
CP-690550 (Tasocitinib)1.00µMROCK 2469
CP-690550 (Tasocitinib)1.00µMPRK2220
CP-690550 (Tasocitinib)1.00µMPKC alpha 710
CP-690550 (Tasocitinib)1.00µMPKC gamma 10620
CP-690550 (Tasocitinib)1.00µMPKC zeta 1025
CP-690550 (Tasocitinib)1.00µMPKD110627
CP-690550 (Tasocitinib)1.00µMSTK3310319
CP-690550 (Tasocitinib)1.00µMMSK17615
CP-690550 (Tasocitinib)1.00µMMNK11150
CP-690550 (Tasocitinib)1.00µMMNK26410
CP-690550 (Tasocitinib)1.00µMMAPKAP-K2 9111
CP-690550 (Tasocitinib)1.00µMMAPKAP-K31187
CP-690550 (Tasocitinib)1.00µMPRAK1237
CP-690550 (Tasocitinib)1.00µMCAMKK beta 13915
CP-690550 (Tasocitinib)1.00µMCAMK1931
CP-690550 (Tasocitinib)1.00µMSmMLCK1043
CP-690550 (Tasocitinib)1.00µMPHK8511
CP-690550 (Tasocitinib)1.00µMDAPK11455
CP-690550 (Tasocitinib)1.00µMCHK18613
CP-690550 (Tasocitinib)1.00µMCHK21067
CP-690550 (Tasocitinib)1.00µMGSK3 beta 1102
CP-690550 (Tasocitinib)1.00µMCDK2-Cyclin A694
CP-690550 (Tasocitinib)1.00µMPLK112118
CP-690550 (Tasocitinib)1.00µMAurora A938
CP-690550 (Tasocitinib)1.00µMAurora B696
CP-690550 (Tasocitinib)1.00µMTLK11048
CP-690550 (Tasocitinib)1.00µMLKB1955
CP-690550 (Tasocitinib)1.00µMAMPK831
CP-690550 (Tasocitinib)1.00µMMARK1631
CP-690550 (Tasocitinib)1.00µMMARK2854
CP-690550 (Tasocitinib)1.00µMMARK3334
CP-690550 (Tasocitinib)1.00µMMARK4861
CP-690550 (Tasocitinib)1.00µMBRSK1732
CP-690550 (Tasocitinib)1.00µMBRSK2825
CP-690550 (Tasocitinib)1.00µMMELK745
CP-690550 (Tasocitinib)1.00µMNUAK1302
CP-690550 (Tasocitinib)1.00µMCK1 delta 1054
CP-690550 (Tasocitinib)1.00µMCK2921
CP-690550 (Tasocitinib)1.00µMDYRK1A1021
CP-690550 (Tasocitinib)1.00µMDYRK29914
CP-690550 (Tasocitinib)1.00µMDYRK311018
CP-690550 (Tasocitinib)1.00µMNEK2a10732
CP-690550 (Tasocitinib)1.00µMNEK6905
CP-690550 (Tasocitinib)1.00µMIKK beta 1263
CP-690550 (Tasocitinib)1.00µMIKK epsilon 907
CP-690550 (Tasocitinib)1.00µMTBK18319
CP-690550 (Tasocitinib)1.00µMPIM11018
CP-690550 (Tasocitinib)1.00µMPIM212121
CP-690550 (Tasocitinib)1.00µMPIM31149
CP-690550 (Tasocitinib)1.00µMSRPK1898
CP-690550 (Tasocitinib)1.00µMEF2K1031
CP-690550 (Tasocitinib)1.00µMEIF2AK31148
CP-690550 (Tasocitinib)1.00µMHIPK1904
CP-690550 (Tasocitinib)1.00µMHIPK212821
CP-690550 (Tasocitinib)1.00µMHIPK310914
CP-690550 (Tasocitinib)1.00µMCLK210610
CP-690550 (Tasocitinib)1.00µMPAK21142
CP-690550 (Tasocitinib)1.00µMPAK411616
CP-690550 (Tasocitinib)1.00µMPAK5944
CP-690550 (Tasocitinib)1.00µMPAK611610
CP-690550 (Tasocitinib)1.00µMMST26412
CP-690550 (Tasocitinib)1.00µMMST41090
CP-690550 (Tasocitinib)1.00µMGCK870
CP-690550 (Tasocitinib)1.00µMMINK1909
CP-690550 (Tasocitinib)1.00µMMEKK18380
CP-690550 (Tasocitinib)1.00µMMLK1908
CP-690550 (Tasocitinib)1.00µMMLK3751
CP-690550 (Tasocitinib)1.00µMTAO11034
CP-690550 (Tasocitinib)1.00µMASK11057
CP-690550 (Tasocitinib)1.00µMTAK111334
CP-690550 (Tasocitinib)1.00µMIRAK11114
CP-690550 (Tasocitinib)1.00µMIRAK4801
CP-690550 (Tasocitinib)1.00µMRIPK2923
CP-690550 (Tasocitinib)1.00µMOSR19412
CP-690550 (Tasocitinib)1.00µMTTK1157
CP-690550 (Tasocitinib)1.00µMMPSK18314
CP-690550 (Tasocitinib)1.00µMSrc907
CP-690550 (Tasocitinib)1.00µMLck300
CP-690550 (Tasocitinib)1.00µMCSK847
CP-690550 (Tasocitinib)1.00µMYES1654
CP-690550 (Tasocitinib)1.00µMABL10313
CP-690550 (Tasocitinib)1.00µMBTK966
CP-690550 (Tasocitinib)1.00µMJAK231
CP-690550 (Tasocitinib)1.00µMSYK15216
CP-690550 (Tasocitinib)1.00µMZAP701253
CP-690550 (Tasocitinib)1.00µMTIE210619
CP-690550 (Tasocitinib)1.00µMBRK8018
CP-690550 (Tasocitinib)1.00µMEPH-A21066
CP-690550 (Tasocitinib)1.00µMEPH-A41212
CP-690550 (Tasocitinib)1.00µMEPH-B1934
CP-690550 (Tasocitinib)1.00µMEPH-B29110
CP-690550 (Tasocitinib)1.00µMEPH-B31038
CP-690550 (Tasocitinib)1.00µMEPH-B413146
CP-690550 (Tasocitinib)1.00µMFGF-R1424
CP-690550 (Tasocitinib)1.00µMHER41168
CP-690550 (Tasocitinib)1.00µMIGF-1R1099
CP-690550 (Tasocitinib)1.00µMIR878
CP-690550 (Tasocitinib)1.00µMIRR1023
CP-690550 (Tasocitinib)1.00µMTrkA8711
CP-690550 (Tasocitinib)1.00µMVEGFR15810