InhibitorScreening ConcentrationKinase% Activity RemainingStandard Deviation
BML-258 (SK1-I)0.10µMMKK19716
BML-258 (SK1-I)0.10µMMKK210410
BML-258 (SK1-I)0.10µMMKK61025
BML-258 (SK1-I)0.10µMERK110823
BML-258 (SK1-I)0.10µMERK2982
BML-258 (SK1-I)0.10µMJNK1986
BML-258 (SK1-I)0.10µMJNK2856
BML-258 (SK1-I)0.10µMJNK3936
BML-258 (SK1-I)0.10µMp38 alpha MAPK958
BML-258 (SK1-I)0.10µMp38 beta MAPK999
BML-258 (SK1-I)0.10µMp38 gamma MAPK934
BML-258 (SK1-I)0.10µMp38 delta MAPK909
BML-258 (SK1-I)0.10µMERK8821
BML-258 (SK1-I)0.10µMRSK1951
BML-258 (SK1-I)0.10µMRSK2873
BML-258 (SK1-I)0.10µMPDK11074
BML-258 (SK1-I)0.10µMPKB alpha 995
BML-258 (SK1-I)0.10µMPKB beta 852
BML-258 (SK1-I)0.10µMSGK1835
BML-258 (SK1-I)0.10µMS6K11148
BML-258 (SK1-I)0.10µMPKA1102
BML-258 (SK1-I)0.10µMROCK 21101
BML-258 (SK1-I)0.10µMPRK2784
BML-258 (SK1-I)0.10µMPKC alpha 960
BML-258 (SK1-I)0.10µMPKC gamma 1016
BML-258 (SK1-I)0.10µMPKC zeta 1062
BML-258 (SK1-I)0.10µMPKD11074
BML-258 (SK1-I)0.10µMSTK331000
BML-258 (SK1-I)0.10µMMSK11106
BML-258 (SK1-I)0.10µMMNK11013
BML-258 (SK1-I)0.10µMMNK21113
BML-258 (SK1-I)0.10µMMAPKAP-K2 9812
BML-258 (SK1-I)0.10µMMAPKAP-K311513
BML-258 (SK1-I)0.10µMPRAK892
BML-258 (SK1-I)0.10µMCAMKK beta 974
BML-258 (SK1-I)0.10µMCAMK110613
BML-258 (SK1-I)0.10µMSmMLCK902
BML-258 (SK1-I)0.10µMPHK995
BML-258 (SK1-I)0.10µMDAPK11097
BML-258 (SK1-I)0.10µMCHK1961
BML-258 (SK1-I)0.10µMCHK2923
BML-258 (SK1-I)0.10µMGSK3 beta 838
BML-258 (SK1-I)0.10µMCDK2-Cyclin A984
BML-258 (SK1-I)0.10µMPLK11061
BML-258 (SK1-I)0.10µMAurora A1163
BML-258 (SK1-I)0.10µMAurora B1002
BML-258 (SK1-I)0.10µMLKB1935
BML-258 (SK1-I)0.10µMAMPK1049
BML-258 (SK1-I)0.10µMMARK111412
BML-258 (SK1-I)0.10µMMARK2895
BML-258 (SK1-I)0.10µMMARK31017
BML-258 (SK1-I)0.10µMMARK49011
BML-258 (SK1-I)0.10µMBRSK11144
BML-258 (SK1-I)0.10µMBRSK21307
BML-258 (SK1-I)0.10µMMELK1082
BML-258 (SK1-I)0.10µMNUAK11052
BML-258 (SK1-I)0.10µMCK1 delta 889
BML-258 (SK1-I)0.10µMCK27812
BML-258 (SK1-I)0.10µMDYRK1A834
BML-258 (SK1-I)0.10µMDYRK21163
BML-258 (SK1-I)0.10µMDYRK3936
BML-258 (SK1-I)0.10µMNEK2a1103
BML-258 (SK1-I)0.10µMNEK6924
BML-258 (SK1-I)0.10µMIKK beta 911
BML-258 (SK1-I)0.10µMIKK epsilon 1063
BML-258 (SK1-I)0.10µMTBK111113
BML-258 (SK1-I)0.10µMPIM11000
BML-258 (SK1-I)0.10µMPIM21036
BML-258 (SK1-I)0.10µMPIM31184
BML-258 (SK1-I)0.10µMSRPK1924
BML-258 (SK1-I)0.10µMEF2K9313
BML-258 (SK1-I)0.10µMHIPK1926
BML-258 (SK1-I)0.10µMHIPK21088
BML-258 (SK1-I)0.10µMHIPK311813
BML-258 (SK1-I)0.10µMCLK21064
BML-258 (SK1-I)0.10µMPAK21132
BML-258 (SK1-I)0.10µMPAK4914
BML-258 (SK1-I)0.10µMPAK51043
BML-258 (SK1-I)0.10µMPAK610511
BML-258 (SK1-I)0.10µMMST2962
BML-258 (SK1-I)0.10µMMST41167
BML-258 (SK1-I)0.10µMGCK862
BML-258 (SK1-I)0.10µMMINK110714
BML-258 (SK1-I)0.10µMMEKK1938
BML-258 (SK1-I)0.10µMMLK11056
BML-258 (SK1-I)0.10µMMLK31028
BML-258 (SK1-I)0.10µMTAO110211
BML-258 (SK1-I)0.10µMASK11158
BML-258 (SK1-I)0.10µMTAK11007
BML-258 (SK1-I)0.10µMIRAK4726
BML-258 (SK1-I)0.10µMRIPK21198
BML-258 (SK1-I)0.10µMTTK954
BML-258 (SK1-I)0.10µMMPSK11042
BML-258 (SK1-I)0.10µMSrc10511
BML-258 (SK1-I)0.10µMLck10611
BML-258 (SK1-I)0.10µMCSK1041
BML-258 (SK1-I)0.10µMYES11231
BML-258 (SK1-I)0.10µMABL1103
BML-258 (SK1-I)0.10µMBTK10725
BML-258 (SK1-I)0.10µMJAK211814
BML-258 (SK1-I)0.10µMSYK1344
BML-258 (SK1-I)0.10µMZAP701162
BML-258 (SK1-I)0.10µMTIE21415
BML-258 (SK1-I)0.10µMBRK1044
BML-258 (SK1-I)0.10µMEPH-A21038
BML-258 (SK1-I)0.10µMEPH-A41004
BML-258 (SK1-I)0.10µMEPH-B112614
BML-258 (SK1-I)0.10µMEPH-B21155
BML-258 (SK1-I)0.10µMEPH-B31040
BML-258 (SK1-I)0.10µMEPH-B41227
BML-258 (SK1-I)0.10µMFGF-R11156
BML-258 (SK1-I)0.10µMHER41276
BML-258 (SK1-I)0.10µMIGF-1R8712
BML-258 (SK1-I)0.10µMIR1077
BML-258 (SK1-I)0.10µMIRR996
BML-258 (SK1-I)0.10µMTrkA1031
BML-258 (SK1-I)0.10µMVEGFR1952
BML-258 (SK1-I)1.00µMMKK11025
BML-258 (SK1-I)1.00µMMKK210312
BML-258 (SK1-I)1.00µMMKK6984
BML-258 (SK1-I)1.00µMERK1979
BML-258 (SK1-I)1.00µMERK2909
BML-258 (SK1-I)1.00µMJNK1943
BML-258 (SK1-I)1.00µMJNK2902
BML-258 (SK1-I)1.00µMJNK31037
BML-258 (SK1-I)1.00µMp38 alpha MAPK8713
BML-258 (SK1-I)1.00µMp38 beta MAPK1062
BML-258 (SK1-I)1.00µMp38 gamma MAPK8011
BML-258 (SK1-I)1.00µMp38 delta MAPK995
BML-258 (SK1-I)1.00µMERK8861
BML-258 (SK1-I)1.00µMRSK1984
BML-258 (SK1-I)1.00µMRSK2951
BML-258 (SK1-I)1.00µMPDK11062
BML-258 (SK1-I)1.00µMPKB alpha 978
BML-258 (SK1-I)1.00µMPKB beta 9013
BML-258 (SK1-I)1.00µMSGK1873
BML-258 (SK1-I)1.00µMS6K11086
BML-258 (SK1-I)1.00µMPKA1062
BML-258 (SK1-I)1.00µMROCK 2945
BML-258 (SK1-I)1.00µMPRK2701
BML-258 (SK1-I)1.00µMPKC alpha 885
BML-258 (SK1-I)1.00µMPKC gamma 1098
BML-258 (SK1-I)1.00µMPKC zeta 1083
BML-258 (SK1-I)1.00µMPKD11124
BML-258 (SK1-I)1.00µMSTK3310011
BML-258 (SK1-I)1.00µMMSK110418
BML-258 (SK1-I)1.00µMMNK19216
BML-258 (SK1-I)1.00µMMNK2983
BML-258 (SK1-I)1.00µMMAPKAP-K2 956
BML-258 (SK1-I)1.00µMMAPKAP-K31191
BML-258 (SK1-I)1.00µMPRAK9912
BML-258 (SK1-I)1.00µMCAMKK beta 8115
BML-258 (SK1-I)1.00µMCAMK110111
BML-258 (SK1-I)1.00µMSmMLCK9512
BML-258 (SK1-I)1.00µMPHK860
BML-258 (SK1-I)1.00µMDAPK110111
BML-258 (SK1-I)1.00µMCHK1927
BML-258 (SK1-I)1.00µMCHK2844
BML-258 (SK1-I)1.00µMGSK3 beta 883
BML-258 (SK1-I)1.00µMCDK2-Cyclin A797
BML-258 (SK1-I)1.00µMPLK1947
BML-258 (SK1-I)1.00µMAurora A1054
BML-258 (SK1-I)1.00µMAurora B1024
BML-258 (SK1-I)1.00µMLKB1890
BML-258 (SK1-I)1.00µMAMPK960
BML-258 (SK1-I)1.00µMMARK111217
BML-258 (SK1-I)1.00µMMARK2979
BML-258 (SK1-I)1.00µMMARK31077
BML-258 (SK1-I)1.00µMMARK4898
BML-258 (SK1-I)1.00µMBRSK11110
BML-258 (SK1-I)1.00µMBRSK21081
BML-258 (SK1-I)1.00µMMELK997
BML-258 (SK1-I)1.00µMNUAK11086
BML-258 (SK1-I)1.00µMCK1 delta 877
BML-258 (SK1-I)1.00µMCK28712
BML-258 (SK1-I)1.00µMDYRK1A916
BML-258 (SK1-I)1.00µMDYRK21243
BML-258 (SK1-I)1.00µMDYRK3981
BML-258 (SK1-I)1.00µMNEK2a1032
BML-258 (SK1-I)1.00µMNEK68612
BML-258 (SK1-I)1.00µMIKK beta 977
BML-258 (SK1-I)1.00µMIKK epsilon 956
BML-258 (SK1-I)1.00µMTBK18239
BML-258 (SK1-I)1.00µMPIM19511
BML-258 (SK1-I)1.00µMPIM21093
BML-258 (SK1-I)1.00µMPIM31216
BML-258 (SK1-I)1.00µMSRPK1893
BML-258 (SK1-I)1.00µMEF2K760
BML-258 (SK1-I)1.00µMHIPK11126
BML-258 (SK1-I)1.00µMHIPK21066
BML-258 (SK1-I)1.00µMHIPK31122
BML-258 (SK1-I)1.00µMCLK210412
BML-258 (SK1-I)1.00µMPAK21031
BML-258 (SK1-I)1.00µMPAK4919
BML-258 (SK1-I)1.00µMPAK51008
BML-258 (SK1-I)1.00µMPAK61087
BML-258 (SK1-I)1.00µMMST2900
BML-258 (SK1-I)1.00µMMST4969
BML-258 (SK1-I)1.00µMGCK722
BML-258 (SK1-I)1.00µMMINK19311
BML-258 (SK1-I)1.00µMMEKK1994
BML-258 (SK1-I)1.00µMMLK11086
BML-258 (SK1-I)1.00µMMLK31064
BML-258 (SK1-I)1.00µMTAO11089
BML-258 (SK1-I)1.00µMASK1993
BML-258 (SK1-I)1.00µMTAK11084
BML-258 (SK1-I)1.00µMIRAK4660
BML-258 (SK1-I)1.00µMRIPK2953
BML-258 (SK1-I)1.00µMTTK914
BML-258 (SK1-I)1.00µMMPSK1988
BML-258 (SK1-I)1.00µMSrc1003
BML-258 (SK1-I)1.00µMLck928
BML-258 (SK1-I)1.00µMCSK10115
BML-258 (SK1-I)1.00µMYES11009
BML-258 (SK1-I)1.00µMABL10611
BML-258 (SK1-I)1.00µMBTK1035
BML-258 (SK1-I)1.00µMJAK2983
BML-258 (SK1-I)1.00µMSYK1056
BML-258 (SK1-I)1.00µMZAP7010610
BML-258 (SK1-I)1.00µMTIE21183
BML-258 (SK1-I)1.00µMBRK938
BML-258 (SK1-I)1.00µMEPH-A2919
BML-258 (SK1-I)1.00µMEPH-A41018
BML-258 (SK1-I)1.00µMEPH-B11087
BML-258 (SK1-I)1.00µMEPH-B210510
BML-258 (SK1-I)1.00µMEPH-B31009
BML-258 (SK1-I)1.00µMEPH-B41018
BML-258 (SK1-I)1.00µMFGF-R111112
BML-258 (SK1-I)1.00µMHER410720
BML-258 (SK1-I)1.00µMIGF-1R862
BML-258 (SK1-I)1.00µMIR10320
BML-258 (SK1-I)1.00µMIRR943
BML-258 (SK1-I)1.00µMTrkA1109
BML-258 (SK1-I)1.00µMVEGFR1815
BML-258 (SK1-I)10.00µMMKK1979
BML-258 (SK1-I)10.00µMMKK210919
BML-258 (SK1-I)10.00µMMKK6991
BML-258 (SK1-I)10.00µMERK1854
BML-258 (SK1-I)10.00µMERK21005
BML-258 (SK1-I)10.00µMJNK19021
BML-258 (SK1-I)10.00µMJNK2885
BML-258 (SK1-I)10.00µMJNK3988
BML-258 (SK1-I)10.00µMp38 alpha MAPK809
BML-258 (SK1-I)10.00µMp38 beta MAPK952
BML-258 (SK1-I)10.00µMp38 gamma MAPK875
BML-258 (SK1-I)10.00µMp38 delta MAPK901
BML-258 (SK1-I)10.00µMERK8770
BML-258 (SK1-I)10.00µMRSK1818
BML-258 (SK1-I)10.00µMRSK28111
BML-258 (SK1-I)10.00µMPDK11229
BML-258 (SK1-I)10.00µMPKB alpha 10724
BML-258 (SK1-I)10.00µMPKB beta 862
BML-258 (SK1-I)10.00µMSGK1784
BML-258 (SK1-I)10.00µMS6K11000
BML-258 (SK1-I)10.00µMPKA10712
BML-258 (SK1-I)10.00µMROCK 21163
BML-258 (SK1-I)10.00µMPRK2581
BML-258 (SK1-I)10.00µMPKC alpha 895
BML-258 (SK1-I)10.00µMPKC gamma 961
BML-258 (SK1-I)10.00µMPKC zeta 925
BML-258 (SK1-I)10.00µMPKD111515
BML-258 (SK1-I)10.00µMSTK338916
BML-258 (SK1-I)10.00µMMSK1951
BML-258 (SK1-I)10.00µMMNK1931
BML-258 (SK1-I)10.00µMMNK210214
BML-258 (SK1-I)10.00µMMAPKAP-K2 914
BML-258 (SK1-I)10.00µMMAPKAP-K31237
BML-258 (SK1-I)10.00µMPRAK903
BML-258 (SK1-I)10.00µMCAMKK beta 902
BML-258 (SK1-I)10.00µMCAMK1895
BML-258 (SK1-I)10.00µMSmMLCK9115
BML-258 (SK1-I)10.00µMPHK760
BML-258 (SK1-I)10.00µMDAPK110318
BML-258 (SK1-I)10.00µMCHK1869
BML-258 (SK1-I)10.00µMCHK2828
BML-258 (SK1-I)10.00µMGSK3 beta 712
BML-258 (SK1-I)10.00µMCDK2-Cyclin A883
BML-258 (SK1-I)10.00µMPLK1963
BML-258 (SK1-I)10.00µMAurora A9215
BML-258 (SK1-I)10.00µMAurora B930
BML-258 (SK1-I)10.00µMLKB1984
BML-258 (SK1-I)10.00µMAMPK946
BML-258 (SK1-I)10.00µMMARK11046
BML-258 (SK1-I)10.00µMMARK2836
BML-258 (SK1-I)10.00µMMARK31050
BML-258 (SK1-I)10.00µMMARK49310
BML-258 (SK1-I)10.00µMBRSK1971
BML-258 (SK1-I)10.00µMBRSK21087
BML-258 (SK1-I)10.00µMMELK9814
BML-258 (SK1-I)10.00µMNUAK11015
BML-258 (SK1-I)10.00µMCK1 delta 814
BML-258 (SK1-I)10.00µMCK2832
BML-258 (SK1-I)10.00µMDYRK1A846
BML-258 (SK1-I)10.00µMDYRK21197
BML-258 (SK1-I)10.00µMDYRK3939
BML-258 (SK1-I)10.00µMNEK2a1087
BML-258 (SK1-I)10.00µMNEK6849
BML-258 (SK1-I)10.00µMIKK beta 1006
BML-258 (SK1-I)10.00µMIKK epsilon 864
BML-258 (SK1-I)10.00µMTBK1931
BML-258 (SK1-I)10.00µMPIM19510
BML-258 (SK1-I)10.00µMPIM2972
BML-258 (SK1-I)10.00µMPIM31072
BML-258 (SK1-I)10.00µMSRPK1839
BML-258 (SK1-I)10.00µMEF2K691
BML-258 (SK1-I)10.00µMHIPK19418
BML-258 (SK1-I)10.00µMHIPK21065
BML-258 (SK1-I)10.00µMHIPK31023
BML-258 (SK1-I)10.00µMCLK29711
BML-258 (SK1-I)10.00µMPAK21138
BML-258 (SK1-I)10.00µMPAK4855
BML-258 (SK1-I)10.00µMPAK51014
BML-258 (SK1-I)10.00µMPAK61035
BML-258 (SK1-I)10.00µMMST2947
BML-258 (SK1-I)10.00µMMST410813
BML-258 (SK1-I)10.00µMGCK719
BML-258 (SK1-I)10.00µMMINK111113
BML-258 (SK1-I)10.00µMMEKK1890
BML-258 (SK1-I)10.00µMMLK11003
BML-258 (SK1-I)10.00µMMLK310912
BML-258 (SK1-I)10.00µMTAO1916
BML-258 (SK1-I)10.00µMASK1940
BML-258 (SK1-I)10.00µMTAK11112
BML-258 (SK1-I)10.00µMIRAK4671
BML-258 (SK1-I)10.00µMRIPK21004
BML-258 (SK1-I)10.00µMTTK864
BML-258 (SK1-I)10.00µMMPSK11004
BML-258 (SK1-I)10.00µMSrc11113
BML-258 (SK1-I)10.00µMLck8411
BML-258 (SK1-I)10.00µMCSK985
BML-258 (SK1-I)10.00µMYES11092
BML-258 (SK1-I)10.00µMABL10910
BML-258 (SK1-I)10.00µMBTK10315
BML-258 (SK1-I)10.00µMJAK210010
BML-258 (SK1-I)10.00µMSYK9213
BML-258 (SK1-I)10.00µMZAP70920
BML-258 (SK1-I)10.00µMTIE21134
BML-258 (SK1-I)10.00µMBRK1042
BML-258 (SK1-I)10.00µMEPH-A2916
BML-258 (SK1-I)10.00µMEPH-A4967
BML-258 (SK1-I)10.00µMEPH-B111518
BML-258 (SK1-I)10.00µMEPH-B21085
BML-258 (SK1-I)10.00µMEPH-B3860
BML-258 (SK1-I)10.00µMEPH-B412313
BML-258 (SK1-I)10.00µMFGF-R11041
BML-258 (SK1-I)10.00µMHER41056
BML-258 (SK1-I)10.00µMIGF-1R9314
BML-258 (SK1-I)10.00µMIR992
BML-258 (SK1-I)10.00µMIRR1005
BML-258 (SK1-I)10.00µMTrkA860
BML-258 (SK1-I)10.00µMVEGFR1834