Kinase Profiling Inhibitor Database

Inhibitor Structure Image Brutto MW Action Reference Reference 2 Patent Commercial Vendor Notes Results
AG1296 (Tyrphostin) C16H14N2O2 266.29 PDGF Kovalenko M. (1994) Cancer Res. 54 6106 Merck (Calbiochem) Download

Results as Barchart

View results as a bar chart
10µM

Results as Table

Screening Concentration: 10µM
Kinase % Activity Remainingsort descending Standard Deviation
Aurora B 15 1
VEGFR1 50 1
CK1 delta 54 2
MELK 64 6
TBK1 64 4
NEK2a 65 5
PAK4 69 1
IR 70 7
Src 72 2
MNK2 74 0
PAK5 74 2
RSK1 75 2
IRR 75 9
PIM3 79 1
MST2 79 6
BTK 80 10
CK2 80 2
AMPK 80 1
Lck 82 1
MNK1 83 11
DYRK2 84 5
SmMLCK 84 26
IKK epsilon 85 2
ROCK 2 85 3
YES1 85 7
ERK8 86 12
EPH-B3 86 10
PRAK 88 13
CAMKK beta 88 1
SGK1 88 3
DYRK3 91 22
CDK2-Cyclin A 91 8
p38 alpha MAPK 91 5
MKK1 92 10
DYRK1A 93 4
CHK2 93 9
FGF-R1 94 18
PKC zeta 94 1
CHK1 95 0
PRK2 95 9
SRPK1 95 0
p38 beta MAPK 95 4
PKA 96 5
PLK1 96 3
RSK2 97 6
PAK6 97 2
HIPK2 98 0
PKB beta 98 0
EPH-A2 98 14
BRSK2 99 2
SYK 100 2
PHK 101 10
ERK1 101 17
IKK beta 101 3
JNK1 101 11
MSK1 102 1
p38 delta MAPK 102 11
IGF-1R 102 7
MARK3 103 9
EF2K 103 10
PKC alpha 103 5
PKD1 103 9
PKB alpha 104 2
CAMK1 104 3
PIM1 104 8
CSK 105 0
ERK2 105 3
MST4 105 10
S6K1 106 17
MAPKAP-K2 107 11
PIM2 108 1
p38 gamma MAPK 110 6
PDK1 110 5
GSK3 beta 113 4
JNK2 113 10
NEK6 116 27

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