Kinase Profiling Inhibitor Database

Inhibitor Structure Image Brutto MW Action Reference Reference 2 Patent Commercial Vendor Notes Results
UCN-01 C28H26N4O4 482.5 PKC Reinhardt H.C. (2007) Cancer Cell 11 175 Jiang X. (2004) Mol. Cancer Ther. 3 1221 Sigma Download

Results as Barchart

View results as a bar chart
0.01µM

Results as Table

Screening Concentration: 0.01µM
Kinase % Activity Remaining Standard Deviation
MKK1 74 0
ERK1 112 5
ERK2 88 4
JNK1 79 8
JNK2 92 7
JNK3 106 0
p38 alpha MAPK 105 7
p38 beta MAPK 105 3
p38 gamma MAPK 103 5
p38 delta MAPK 94 2
ERK8 92 2
RSK1 25 2
RSK2 28 4
PDK1 1 0
PKB alpha 79 2
PKB beta 76 4
SGK1 83 0
S6K1 95 3
PKA 62 2
ROCK 2 86 3
PRK2 9 3
PKC alpha 5 0
PKC zeta 78 5
PKD1 83 5
MSK1 67 7
MNK1 84 0
MNK2 103 1
MAPKAP-K2 75 5
MAPKAP-K3 107 4
PRAK 83 1
CAMKK alpha 57 3
CAMKK beta 20 0
CAMK1 86 2
SmMLCK 82 8
PHK 5 1
CHK1 11 1
CHK2 95 1
GSK3 beta 76 5
CDK2-Cyclin A 44 0
PLK1 75 6
Aurora B 58 0
Aurora C 70 5
AMPK 8 0
MARK3 5 1
BRSK2 27 6
MELK 52 8
CK1 delta 96 1
CK2 92 3
DYRK1A 90 8
DYRK2 91 9
DYRK3 84 7
NEK2a 84 1
NEK6 104 2
NEK7 99 0
IKK beta 85 0
PIM1 52 2
PIM2 72 3
PIM3 7 0
SRPK1 70 0
EF2K 104 7
HIPK2 109 3
HIPK3 115 1
PAK4 33 1
PAK5 35 0
PAK6 35 0
MST2 2 0
Src 76 3
Lck 49 8
CSK 80 0

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